HU9502832D0 - Cyclic compounds useful as inhibitors of platelet glycoprotein iib/iiia - Google Patents

Cyclic compounds useful as inhibitors of platelet glycoprotein iib/iiia

Info

Publication number: HU9502832D0
Authority: HU; Hungary
Prior art keywords: iiia; inhibitors; compounds useful; cyclic compounds; glycoprotein iib
Prior art date: 1993-03-29

Application number

HU9502832A

Other languages

Hungarian (hu)

Other versions

HUT72896A (en

Inventor

William Frank Degrado

Shaker Ahmed Mousa

Anju Parthasarathy

Michael Sworin

Sharon Anne Jackson

Maria Rafalski

Original Assignee

Du Pont Merck Pharma

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1993-03-29

Filing date

1994-03-28

Publication date

1995-11-28

1994-03-28 Application filed by Du Pont Merck Pharma filed Critical Du Pont Merck Pharma

1995-11-28 Publication of HU9502832D0 publication Critical patent/HU9502832D0/en

1996-06-28 Publication of HUT72896A publication Critical patent/HUT72896A/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/745—Blood coagulation or fibrinolysis factors
- C07K14/75—Fibrinogen
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Hematology (AREA)
Medicinal Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Zoology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Diabetes (AREA)
Pharmacology & Pharmacy (AREA)
Bioinformatics & Cheminformatics (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Toxicology (AREA)
Chemical Kinetics & Catalysis (AREA)
Gastroenterology & Hepatology (AREA)
Biochemistry (AREA)
Biophysics (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Peptides Or Proteins (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

HU9502832A 1993-03-29 1994-03-28 Cyclic compounds useful as inhibitors of platelet glycoprotein iib/iiia HUT72896A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US3844893A	1993-03-29	1993-03-29

Publications (2)

Publication Number	Publication Date
HU9502832D0 true HU9502832D0 (en)	1995-11-28
HUT72896A HUT72896A (en)	1996-06-28

Family

ID=21900014

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
HU9502832A HUT72896A (en)	1993-03-29	1994-03-28	Cyclic compounds useful as inhibitors of platelet glycoprotein iib/iiia

Country Status (10)

Country	Link
EP (1)	EP0691987A1 (en)
JP (1)	JPH08508498A (en)
AU (1)	AU6415894A (en)
CA (1)	CA2159070A1 (en)
FI (1)	FI954556A (en)
HU (1)	HUT72896A (en)
NO (1)	NO953832L (en)
NZ (1)	NZ263456A (en)
PL (1)	PL310896A1 (en)
WO (1)	WO1994022910A1 (en)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CA2159072A1 (en) *	1993-03-29	1994-10-13	Lin-Hua Zhang	Novel processes and intermediate compounds for the preparation of platelet glycoprotein iib/iiia inhibitors
US5879657A (en) *	1993-03-30	1999-03-09	The Dupont Merck Pharmaceutical Company	Radiolabeled platelet GPIIb/IIIa receptor antagonists as imaging agents for the diagnosis of thromboembolic disorders
CA2272317C (en) *	1996-11-27	2001-01-30	Rhone-Poulenc Rorer Pharmaceuticals Inc.	Pharmaceutical composition comprising a compound having anti-xa activity and a platelet aggregation antagonist compound
US6010911A (en) *	1997-04-30	2000-01-04	Medtronic, Inc.	Apparatus for performing a heparin-independent high sensitivity platelet function evaluation technique
US6537520B1 (en)	1998-03-31	2003-03-25	Bristol-Myers Squibb Pharma Company	Pharmaceuticals for the imaging of angiogenic disorders
GB0623607D0 (en)	2006-11-27	2007-01-03	Haemostatix Ltd	Tissue adhesive
JP5649825B2 (en)	2007-01-31	2015-01-07	デイナファーバーキャンサーインスティチュート，インコーポレイテッド	Stabilized p53 peptides and methods of use thereof
CA2682174C (en)	2007-03-28	2021-04-06	President And Fellows Of Harvard College	Stitched polypeptides
US11673914B2 (en)	2009-11-10	2023-06-13	Allegro Pharmaceuticals, LLC	Peptide therapies for reduction of macular thickening
BR112012011731A2 (en) *	2009-11-10	2020-08-25	Allegro Pharmaceuticals, Inc.	compositions and methods for inhibiting cell adhesion or targeting diagnostic or therapeutic agents to rgd binding sites
PL2603600T3 (en)	2010-08-13	2019-06-28	Aileron Therapeutics, Inc.	Peptidomimetic macrocycles
JP6106159B2 (en)	2011-05-09	2017-03-29	アレグロファーマシューティカルズインコーポレイテッドＡｌｌｅｇｒｏＰｈａｒｍａｃｅｕｔｉｃａｌｓ，Ｉｎｃ．	Pharmaceutical composition comprising RG-cysteic acid peptide
AR088392A1 (en)	2011-10-18	2014-05-28	Aileron Therapeutics Inc	PEPTIDOMIMETIC MACROCICLES
CN104144695A (en)	2012-02-15	2014-11-12	爱勒让治疗公司	Triazole-crosslinked and thioether-crosslinked peptidomimetic macrocycles
RU2017145921A (en)	2012-02-15	2019-02-21	Эйлерон Терапьютикс, Инк.	PEPTIDOMIMETIC MACROCYCLES
KR20150082307A (en)	2012-11-01	2015-07-15	에일러론 테라퓨틱스 인코포레이티드	Disubstituted amino acids and methods of preparation and use thereof
SG11201702175YA (en)	2014-09-24	2017-04-27	Aileron Therapeutics Inc	Peptidomimetic macrocycles and formulations thereof
SG10201902594QA (en)	2014-09-24	2019-04-29	Aileron Therapeutics Inc	Peptidomimetic macrocycles and uses thereof
KR20170129879A (en)	2015-03-20	2017-11-27	에일러론 테라퓨틱스 인코포레이티드	Peptidomimetic macrocycles and their uses
CN108368161A (en)	2015-09-10	2018-08-03	艾瑞朗医疗公司	Peptidomimetic macrocyclic compound as MCL-1 conditioning agents

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2636066B1 (en) *	1988-09-02	1991-10-25	Centre Nat Rech Scient	CYCLOPEPTIDE DERIVATIVES FOR USE AS SELECTIVE INHIBITORS AGAINST ACTIVE SERINE PROTEASES
US5384309A (en) *	1989-07-17	1995-01-24	Genentech, Inc.	Cyclized peptides and their use as platelet aggregation inhibitors
AU6470590A (en) *	1989-10-23	1991-04-26	Smithkline Beecham Corporation	Cyclic anti-aggregatory peptides
IL103252A (en) *	1991-09-30	1997-03-18	Du Pont Merck Pharma	CYCLIC COMPOUNDS USEFUL AS INHIBITORS OF PLATELET GLYCOPROTEIN IIb/IIIa AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

1994
- 1994-03-28 PL PL94310896A patent/PL310896A1/en unknown
- 1994-03-28 CA CA002159070A patent/CA2159070A1/en not_active Abandoned
- 1994-03-28 EP EP94911703A patent/EP0691987A1/en not_active Withdrawn
- 1994-03-28 NZ NZ263456A patent/NZ263456A/en not_active IP Right Cessation
- 1994-03-28 WO PCT/US1994/003223 patent/WO1994022910A1/en not_active Application Discontinuation
- 1994-03-28 HU HU9502832A patent/HUT72896A/en unknown
- 1994-03-28 AU AU64158/94A patent/AU6415894A/en not_active Abandoned
- 1994-03-28 JP JP6522195A patent/JPH08508498A/en not_active Ceased
1995
- 1995-09-26 FI FI954556A patent/FI954556A/en unknown
- 1995-09-28 NO NO953832A patent/NO953832L/en unknown

Also Published As

Publication number	Publication date
FI954556A0 (en)	1995-09-26
FI954556A (en)	1995-09-26
NZ263456A (en)	1996-11-26
EP0691987A1 (en)	1996-01-17
NO953832L (en)	1995-11-28
AU6415894A (en)	1994-10-24
WO1994022910A1 (en)	1994-10-13
JPH08508498A (en)	1996-09-10
PL310896A1 (en)	1996-01-08
NO953832D0 (en)	1995-09-28
CA2159070A1 (en)	1994-10-13
HUT72896A (en)	1996-06-28

Publication	Publication Date	Title
HU9502832D0 (en)	1995-11-28	Cyclic compounds useful as inhibitors of platelet glycoprotein iib/iiia
AU2025192A (en)	1992-12-30	Peptide mimetic compounds useful as platelet aggregation inhibitors
AU3143793A (en)	1993-07-19	Peptide mimetic compounds useful as platelet aggregation inhibitors
AU1400095A (en)	1995-07-17	Compounds containing basic and acidic termini useful as fibrinogen receptor antagonists
ZA93550B (en)	1994-07-26	Azabricyclic compounds as calcium channel antagonists
AU3364493A (en)	1993-09-01	Compounds as calcium channel antagonists
EP0511866A3 (en)	1993-03-17	Process for the crystallization of cyclic lipopeptides
ITMI932056A1 (en)	1995-03-27	LOCK FOR CONTAINERS SUCH AS BAGS OR SIMILAR
GB9216384D0 (en)	1992-09-16	Improvements relating to packaging
GB9317297D0 (en)	1993-10-06	Biocidal compositions containing organoboron compounds
ZA93549B (en)	1994-09-22	Azabicyclo compounds as calcium channel antagonists
ZA927515B (en)	1994-03-30	Cyclic compounds useful as inhibitors of platelet glycoprotein IIb/IIIa
GB9423929D0 (en)	1995-01-11	Substituted benzene compounds as tranferase inhibitors
AU1398595A (en)	1995-07-10	Peptide analogs of the factor ixa platelet binding site
GB9209374D0 (en)	1992-06-17	Improvements relating to sealable containers
WO1994022911A3 (en)	1995-01-12	A PROCESS AND INTERMEDIATE COMPOUNDS USEFUL FOR THE PREPARATION OF PLATELET GLYCOPROTEIN IIb/IIIa INHIBITORS CONTAINING Nα-METHYLARGININE
GB2257958B (en)	1995-03-15	Improvements relating to packaging
GB9302184D0 (en)	1993-03-24	Improvements relating to the formation of cartosn
GB9222377D0 (en)	1992-12-09	Improvements relating to packaging containers
GB9205505D0 (en)	1992-04-29	Cyclic compounds
GB9320958D0 (en)	1993-12-01	Improvements relating to packaging of articles
GB9214278D0 (en)	1992-08-19	Improvements relating to packaging
GB2275466B (en)	1997-01-22	Improvements relating to containers
GB9321861D0 (en)	1993-12-15	Platelet derived growth factor analogues
GB9324788D0 (en)	1994-01-19	Improvements relating to packaging

Legal Events

Date	Code	Title	Description
1998-01-28	DFC4	Cancellation of temporary prot. due to refusal