HK1089959A1 - Saquinavir mesylate oral dosage form - Google Patents

Saquinavir mesylate oral dosage form

Info

Publication number: HK1089959A1
Authority: HK; Hong Kong
Prior art keywords: dosage form; oral dosage; saquinavir mesylate; mesylate oral; saquinavir
Prior art date: 2003-07-11

Application number

HK06110649.8A

Other languages

English (en)

Inventor

Antonio A Albano

Martin Howard Infeld

Wantanee Phuapradit

Navnit-Hargovindas Shah

Lin Zhang

Original Assignee

Hoffmann La Roche

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-07-11

Filing date

2006-09-25

Publication date

2006-12-15

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34068244&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1089959(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2006-09-25 Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche

2006-12-15 Publication of HK1089959A1 publication Critical patent/HK1089959A1/xx

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1617—Organic compounds, e.g. phospholipids, fats
- A61K9/1623—Sugars or sugar alcohols, e.g. lactose; Derivatives thereof; Homeopathic globules
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1635—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Epidemiology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Molecular Biology (AREA)
Biophysics (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Virology (AREA)
Oncology (AREA)
Communicable Diseases (AREA)
Tropical Medicine & Parasitology (AREA)
AIDS & HIV (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)
Peptides Or Proteins (AREA)

HK06110649.8A 2003-07-11 2006-09-25 Saquinavir mesylate oral dosage form HK1089959A1 (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US48660003P	2003-07-11	2003-07-11
US56820404P	2004-05-05	2004-05-05
PCT/EP2004/007309 WO2005004836A2 (en)	2003-07-11	2004-07-05	Saquinavir mesylate oral dosage form

Publications (1)

Publication Number	Publication Date
HK1089959A1 true HK1089959A1 (en)	2006-12-15

Family

ID=34068244

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
HK06110649.8A HK1089959A1 (en)	2003-07-11	2006-09-25	Saquinavir mesylate oral dosage form

Country Status (24)

Country	Link
US (2)	US20050009811A1 (es)
EP (1)	EP1646369B1 (es)
JP (2)	JP4608488B2 (es)
KR (2)	KR20070087194A (es)
AU (1)	AU2004255436B2 (es)
BR (1)	BRPI0412523A (es)
CA (1)	CA2531486C (es)
CO (1)	CO5640069A2 (es)
CR (1)	CR8172A (es)
EA (1)	EA015349B1 (es)
EC (1)	ECSP066274A (es)
HK (1)	HK1089959A1 (es)
IL (1)	IL172890A (es)
MA (1)	MA27904A1 (es)
MX (1)	MXPA06000363A (es)
MY (1)	MY140413A (es)
NO (1)	NO20060313L (es)
NZ (1)	NZ544585A (es)
PA (1)	PA8606001A1 (es)
PE (1)	PE20050247A1 (es)
RS (1)	RS20060009A (es)
TN (1)	TNSN06003A1 (es)
TW (1)	TWI356711B (es)
WO (1)	WO2005004836A2 (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JP5767429B2 (ja)	1999-11-12	2015-08-19	アッヴィ・インコーポレイテッド	固体分散剤中の結晶化阻害剤
US7364752B1 (en)	1999-11-12	2008-04-29	Abbott Laboratories	Solid dispersion pharamaceutical formulations
WO2005004836A2 (en) *	2003-07-11	2005-01-20	F.Hoffmann-La Roche Ag	Saquinavir mesylate oral dosage form
US8025899B2 (en)	2003-08-28	2011-09-27	Abbott Laboratories	Solid pharmaceutical dosage form
US8377952B2 (en)	2003-08-28	2013-02-19	Abbott Laboratories	Solid pharmaceutical dosage formulation
EP2168573A1 (en) *	2008-09-30	2010-03-31	LEK Pharmaceuticals D.D.	Formulations comprising ezetimibe
WO2013172297A1 (ja)	2012-05-14	2013-11-21	塩野義製薬株式会社	６，７－不飽和－７－カルバモイルモルヒナン誘導体含有製剤
MX2021004553A (es) *	2018-10-23	2021-07-16	Eastern Virginia Medical School	Composiciones farmaceuticas y metodos para fabricar formulaciones de dosificacion solidas bajo demanda.

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4753801A (en) *	1985-10-25	1988-06-28	Eli Lilly And Company	Sustained release tablets
JP2642486B2 (ja) *	1989-08-04	1997-08-20	田辺製薬株式会社	難溶性薬物の超微粒子化法
GB8927913D0 (en) *	1989-12-11	1990-02-14	Hoffmann La Roche	Amino acid derivatives
EP0616841B1 (en) *	1992-10-09	1998-12-23	Kanegafuchi Kagaku Kogyo Kabushiki Kaisha	Production method for fine granulate
TW390813B (en) *	1994-04-29	2000-05-21	Merck & Co Inc	Wet granulation formulation for bisphosphonic acids
US5585115A (en) *	1995-01-09	1996-12-17	Edward H. Mendell Co., Inc.	Pharmaceutical excipient having improved compressability
US5608085A (en) *	1995-02-27	1997-03-04	The University Of Tennessee Research Corporation	Synthesis of optically active calanolides A and B and enantiomers and related compounds
US6177460B1 (en) *	1995-04-12	2001-01-23	The Procter & Gamble Company	Method of treatment for cancer or viral infections
US6039975A (en) *	1995-10-17	2000-03-21	Hoffman-La Roche Inc.	Colon targeted delivery system
US6045829A (en) *	1997-02-13	2000-04-04	Elan Pharma International Limited	Nanocrystalline formulations of human immunodeficiency virus (HIV) protease inhibitors using cellulosic surface stabilizers
US6514530B2 (en) *	1997-09-09	2003-02-04	Alza Corporation	Dosage form comprising means for changing drug delivery shape
AU3705799A (en) *	1998-04-09	1999-11-01	F. Hoffmann-La Roche Ag	Process for the manufacture of (sub)micron sized particles by dissolving in compressed gas and surfactants
HUP0104721A3 (en) *	1998-12-17	2006-07-28	Alza Corp Mountain View	Conversion of liquid filled gelatin capsules into controlled release systems by multiple coatings
US7674480B2 (en) *	2000-06-23	2010-03-09	Teva Pharmaceutical Industries Ltd.	Rapidly expanding composition for gastric retention and controlled release of therapeutic agents, and dosage forms including the composition
EP1247456A3 (en) *	2001-02-28	2003-12-10	Pfizer Products Inc.	Palatable pharmaceutical compositions for companion animals
US20030068356A1 (en) *	2001-07-10	2003-04-10	Pather S. Indiran	Sequential drug delivery systems
WO2005004836A2 (en) *	2003-07-11	2005-01-20	F.Hoffmann-La Roche Ag	Saquinavir mesylate oral dosage form

2004
- 2004-07-05 WO PCT/EP2004/007309 patent/WO2005004836A2/en active IP Right Grant
- 2004-07-05 NZ NZ544585A patent/NZ544585A/en not_active IP Right Cessation
- 2004-07-05 MX MXPA06000363A patent/MXPA06000363A/es active IP Right Grant
- 2004-07-05 EP EP04763093.4A patent/EP1646369B1/en not_active Expired - Lifetime
- 2004-07-05 JP JP2006519808A patent/JP4608488B2/ja not_active Expired - Lifetime
- 2004-07-05 CA CA2531486A patent/CA2531486C/en not_active Expired - Lifetime
- 2004-07-05 AU AU2004255436A patent/AU2004255436B2/en not_active Ceased
- 2004-07-05 BR BRPI0412523-1A patent/BRPI0412523A/pt not_active IP Right Cessation
- 2004-07-05 KR KR1020077016817A patent/KR20070087194A/ko not_active Application Discontinuation
- 2004-07-05 EA EA200600156A patent/EA015349B1/ru not_active IP Right Cessation
- 2004-07-05 RS YUP-2006/0009A patent/RS20060009A/sr unknown
- 2004-07-05 KR KR1020067000732A patent/KR100767271B1/ko active IP Right Grant
- 2004-07-07 PE PE2004000651A patent/PE20050247A1/es not_active Application Discontinuation
- 2004-07-07 TW TW093120382A patent/TWI356711B/zh not_active IP Right Cessation
- 2004-07-07 PA PA20048606001A patent/PA8606001A1/es unknown
- 2004-07-08 US US10/886,765 patent/US20050009811A1/en not_active Abandoned
- 2004-07-09 MY MYPI20042754A patent/MY140413A/en unknown
2005
- 2005-12-29 IL IL172890A patent/IL172890A/en not_active IP Right Cessation
2006
- 2006-01-05 CR CR8172A patent/CR8172A/es unknown
- 2006-01-06 TN TNP2006000003A patent/TNSN06003A1/en unknown
- 2006-01-06 MA MA28709A patent/MA27904A1/fr unknown
- 2006-01-06 CO CO06001295A patent/CO5640069A2/es not_active Application Discontinuation
- 2006-01-09 EC EC2006006274A patent/ECSP066274A/es unknown
- 2006-01-20 NO NO20060313A patent/NO20060313L/no not_active Application Discontinuation
- 2006-09-25 HK HK06110649.8A patent/HK1089959A1/xx not_active IP Right Cessation
2008
- 2008-10-31 US US12/262,607 patent/US20090054481A1/en not_active Abandoned
2010
- 2010-08-13 JP JP2010181350A patent/JP2010280707A/ja active Pending

Also Published As

Publication number	Publication date
AU2004255436B2 (en)	2006-11-30
EA015349B1 (ru)	2011-06-30
US20050009811A1 (en)	2005-01-13
TWI356711B (en)	2012-01-21
NO20060313L (no)	2006-02-09
WO2005004836A3 (en)	2005-05-12
CR8172A (es)	2006-10-04
CA2531486C (en)	2012-10-02
US20090054481A1 (en)	2009-02-26
TNSN06003A1 (en)	2007-10-03
KR100767271B1 (ko)	2007-10-17
MXPA06000363A (es)	2006-03-28
CO5640069A2 (es)	2006-05-31
CA2531486A1 (en)	2005-01-20
PE20050247A1 (es)	2005-04-13
MY140413A (en)	2009-12-31
IL172890A0 (en)	2006-06-11
EP1646369B1 (en)	2019-04-10
EP1646369A2 (en)	2006-04-19
JP2010280707A (ja)	2010-12-16
JP4608488B2 (ja)	2011-01-12
TW200505504A (en)	2005-02-16
ECSP066274A (es)	2006-10-25
IL172890A (en)	2013-11-28
MA27904A1 (fr)	2006-05-02
PA8606001A1 (es)	2005-03-03
NZ544585A (en)	2008-04-30
BRPI0412523A (pt)	2006-09-19
JP2009501694A (ja)	2009-01-22
RS20060009A (en)	2008-06-05
EA200600156A1 (ru)	2006-08-25
AU2004255436A1 (en)	2005-01-20
WO2005004836A2 (en)	2005-01-20
KR20070087194A (ko)	2007-08-27
KR20060056320A (ko)	2006-05-24

Publication	Publication Date	Title
EP1581188A4 (en)	2006-04-05	DOSAGE FORM WITH PHARMACEUTICAL SAFETY
HK1107768A1 (en)	2008-04-18	Solid drug for oral use
GB0324886D0 (en)	2003-11-26	Medicinal compounds
GB0302671D0 (en)	2003-03-12	Pharmaceutical formulations
GB0303396D0 (en)	2003-03-19	Medicinal compounds
EP1553925A4 (en)	2012-09-05	ORAL DOSAGE FORM WITH MODIFIED RELEASE
AU2003238670A8 (en)	2003-10-27	Fast disintegrating oral dosage forms
ZA200509379B (en)	2006-11-29	Memantine oral dosage forms
HK1089959A1 (en)	2006-12-15	Saquinavir mesylate oral dosage form
GB0300531D0 (en)	2003-02-12	Pharmaceutical compositions
IL172824A0 (en)	2006-06-11	Pharmaceutical formulations
EP1648411A4 (en)	2010-03-10	PHARMACEUTICAL COMPOSITIONS
GB0302672D0 (en)	2003-03-12	Pharmaceutical formulations
GB0328490D0 (en)	2004-01-14	Medicinal compounds
HK1092715A1 (en)	2007-02-16	Melt-formulated, multi-particulate oral dosage form
EP1655029A4 (en)	2010-01-13	MEDICINAL COMPOSITIONS
GB0316341D0 (en)	2003-08-13	Pharmaceutical formulations
EP1361866A4 (en)	2007-10-17	EMULSIONS AS SOLID DOSAGE FORMS FOR ORAL ADMINISTRATION
HK1094676A1 (en)	2007-04-04	Solid pharmaceutical preparation form
ZA200603126B (en)	2007-02-28	Pharmaceutical compositions for therapeutic use
GB0305579D0 (en)	2003-04-16	Pharmaceutical compositions
PL373776A1 (en)	2005-10-03	Oral pharmaceutical compound
GB0315019D0 (en)	2003-07-30	Dosage form
GB0316335D0 (en)	2003-08-13	Pharmaceutical formulations
GB0218994D0 (en)	2002-09-25	Oral pharmaceutical compositions

Legal Events

Date	Code	Title	Description
2024-07-19	PE	Patent expired	Effective date: 20240704