HK1039113A1 - Benzothieno Ä3,2-CÜpyridines as alpha2 antagonists - Google Patents

Benzothieno Ä3,2-CÜpyridines as alpha2 antagonists

Info

Publication number: HK1039113A1
Authority: HK; Hong Kong
Prior art keywords: cüpyridines; benzothieno; alpha2 antagonists; alpha2; antagonists
Prior art date: 1998-10-06

Application number

HK01108819A

Other languages

English (en)

Inventor

Ludo Edmond Josephine Kennis

Serge Maria Aloysius Pieters

Francois Paul Bischoff

Original Assignee

Janssen Pharmaceutica Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-10-06

Filing date

2001-12-15

Publication date

2002-04-12

2001-12-15 Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv

2002-04-12 Publication of HK1039113A1 publication Critical patent/HK1039113A1/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Diabetes (AREA)
Psychiatry (AREA)
Pain & Pain Management (AREA)
Endocrinology (AREA)
Psychology (AREA)
Hospice & Palliative Care (AREA)
Emergency Medicine (AREA)
Hematology (AREA)
Obesity (AREA)
Reproductive Health (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

HK01108819A 1998-10-06 2001-12-15 Benzothieno Ä3,2-CÜpyridines as alpha2 antagonists HK1039113A1 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP98203363		1998-10-06
PCT/EP1999/007418 WO2000020422A1 (en)	1998-10-06	1999-10-01	BENZOTHIENO[3,2-c]PYRIDINES AS α2 ANTAGONISTS

Publications (1)

Publication Number	Publication Date
HK1039113A1 true HK1039113A1 (en)	2002-04-12

Family

ID=8234188

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
HK01108819A HK1039113A1 (en)	1998-10-06	2001-12-15	Benzothieno Ä3,2-CÜpyridines as alpha2 antagonists

Country Status (28)

Country	Link
US (2)	US6426350B1 (xx)
EP (1)	EP1117667B1 (xx)
JP (1)	JP4580555B2 (xx)
KR (1)	KR20010071828A (xx)
CN (1)	CN1158287C (xx)
AR (1)	AR023678A1 (xx)
AT (1)	ATE363485T1 (xx)
AU (1)	AU760226B2 (xx)
BG (1)	BG64625B1 (xx)
BR (1)	BR9913110A (xx)
CA (1)	CA2346084C (xx)
CZ (1)	CZ20011103A3 (xx)
DE (1)	DE69936219T2 (xx)
EE (1)	EE04835B1 (xx)
ES (1)	ES2288025T3 (xx)
HK (1)	HK1039113A1 (xx)
HU (1)	HUP0103612A3 (xx)
ID (1)	ID28280A (xx)
IL (2)	IL142442A0 (xx)
NO (1)	NO20011309D0 (xx)
NZ (1)	NZ509911A (xx)
PL (1)	PL347184A1 (xx)
RU (1)	RU2222542C2 (xx)
SK (1)	SK4312001A3 (xx)
TR (1)	TR200100954T2 (xx)
TW (1)	TWI251595B (xx)
UA (1)	UA70334C2 (xx)
WO (1)	WO2000020422A1 (xx)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP2305284A3 (en) *	2002-03-08	2012-11-14	Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V.	Use of EGFR transactivation inhibitors in human cancer
JP2005521728A (ja) *	2002-04-03	2005-07-21	オリオンコーポレーション	ＣＮＳ関連疾患のためのα２−アドレナリン受容体アンタゴニストの使用
CN1972938B (zh)	2004-04-12	2010-09-29	大正制药株式会社	环状胺化合物

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3752820A (en) *	1972-03-20	1973-08-14	Colgate Palmolive Co	Substituted-1,2,3,4-tetrahydrobenzothieno(3,2-c)pyridine derivatives
FR2570701B1 (fr) *	1984-09-27	1987-05-22	Synthelabo	Derives de furo(3,2-c)pyridines, leur preparation et leur application en therapeutique
US4686226A (en) *	1985-09-03	1987-08-11	Merck & Co., Inc.	Substituted benzo[b]furo- and benzo[b]thieno quinolizines
EP0339959A3 (en) *	1988-04-27	1991-03-20	Glaxo Group Limited	Lactam derivatives
US5100891A (en) *	1991-01-18	1992-03-31	Hoechst-Roussel Pharmaceuticals Inc.	Substituted 1,2,3,4-tetrahydrocyclopent[b]indoles, 1,2,3,3a,4,8a-hexahydrocyclopent[B]indoles and related compounds
DE69531476T2 (de) *	1994-09-12	2004-06-09	Lilly Industries Ltd., Basingstoke	Serotonergische Modulatoren
JP3274579B2 (ja) *	1995-01-12	2002-04-15	住友製薬株式会社	脳血管障害に伴う精神症候治療剤
UA52681C2 (uk)	1997-04-08	2003-01-15	Янссен Фармацевтика Н.В.	Похідні 1,2,3,4-тетрагідро-бензофуро[3,2,-c]піридину, спосіб їх одержання та фармацевтична композиція на їх основі

1999
- 1999-01-10 UA UA2001031998A patent/UA70334C2/uk unknown
- 1999-10-01 EE EEP200100206A patent/EE04835B1/xx not_active IP Right Cessation
- 1999-10-01 IL IL14244299A patent/IL142442A0/xx active IP Right Grant
- 1999-10-01 DE DE69936219T patent/DE69936219T2/de not_active Expired - Lifetime
- 1999-10-01 PL PL99347184A patent/PL347184A1/xx not_active Application Discontinuation
- 1999-10-01 JP JP2000574534A patent/JP4580555B2/ja not_active Expired - Fee Related
- 1999-10-01 WO PCT/EP1999/007418 patent/WO2000020422A1/en active IP Right Grant
- 1999-10-01 ID IDW20010781A patent/ID28280A/id unknown
- 1999-10-01 US US09/806,432 patent/US6426350B1/en not_active Expired - Lifetime
- 1999-10-01 CA CA2346084A patent/CA2346084C/en not_active Expired - Fee Related
- 1999-10-01 ES ES99947469T patent/ES2288025T3/es not_active Expired - Lifetime
- 1999-10-01 CN CNB998116777A patent/CN1158287C/zh not_active Expired - Fee Related
- 1999-10-01 TW TW088116899A patent/TWI251595B/zh not_active IP Right Cessation
- 1999-10-01 KR KR1020017000400A patent/KR20010071828A/ko active Search and Examination
- 1999-10-01 TR TR2001/00954T patent/TR200100954T2/xx unknown
- 1999-10-01 RU RU2001111753/04A patent/RU2222542C2/ru not_active IP Right Cessation
- 1999-10-01 NZ NZ509911A patent/NZ509911A/xx unknown
- 1999-10-01 SK SK431-2001A patent/SK4312001A3/sk unknown
- 1999-10-01 AT AT99947469T patent/ATE363485T1/de not_active IP Right Cessation
- 1999-10-01 HU HU0103612A patent/HUP0103612A3/hu unknown
- 1999-10-01 BR BR9913110-2A patent/BR9913110A/pt not_active Application Discontinuation
- 1999-10-01 AU AU60899/99A patent/AU760226B2/en not_active Ceased
- 1999-10-01 CZ CZ20011103A patent/CZ20011103A3/cs unknown
- 1999-10-01 EP EP99947469A patent/EP1117667B1/en not_active Expired - Lifetime
- 1999-10-05 AR ARP990105039A patent/AR023678A1/es active IP Right Grant
2001
- 2001-03-12 BG BG105331A patent/BG64625B1/bg unknown
- 2001-03-15 NO NO20011309A patent/NO20011309D0/no not_active Application Discontinuation
- 2001-04-04 IL IL142442A patent/IL142442A/en not_active IP Right Cessation
- 2001-12-15 HK HK01108819A patent/HK1039113A1/xx not_active IP Right Cessation
2002
- 2002-04-16 US US10/123,338 patent/US6774129B2/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
CA2346084A1 (en)	2000-04-13
CZ20011103A3 (cs)	2001-12-12
JP4580555B2 (ja)	2010-11-17
DE69936219T2 (de)	2008-02-07
DE69936219D1 (de)	2007-07-12
ES2288025T3 (es)	2007-12-16
EP1117667B1 (en)	2007-05-30
ATE363485T1 (de)	2007-06-15
US20020169178A1 (en)	2002-11-14
US6774129B2 (en)	2004-08-10
IL142442A (en)	2006-10-05
KR20010071828A (ko)	2001-07-31
HUP0103612A3 (en)	2003-03-28
BR9913110A (pt)	2001-05-08
ID28280A (id)	2001-05-10
BG64625B1 (bg)	2005-09-30
IL142442A0 (en)	2002-03-10
EE04835B1 (et)	2007-06-15
NZ509911A (en)	2002-09-27
HUP0103612A2 (hu)	2002-01-28
AU760226B2 (en)	2003-05-08
CN1158287C (zh)	2004-07-21
PL347184A1 (en)	2002-03-25
AU6089999A (en)	2000-04-26
BG105331A (en)	2001-11-30
RU2222542C2 (ru)	2004-01-27
EP1117667A1 (en)	2001-07-25
TR200100954T2 (tr)	2001-12-21
NO20011309L (no)	2001-03-15
US6426350B1 (en)	2002-07-30
CN1321159A (zh)	2001-11-07
AR023678A1 (es)	2002-09-04
SK4312001A3 (en)	2001-12-03
JP2002526546A (ja)	2002-08-20
TWI251595B (en)	2006-03-21
WO2000020422A1 (en)	2000-04-13
CA2346084C (en)	2010-01-26
NO20011309D0 (no)	2001-03-15
UA70334C2 (en)	2004-10-15
EE200100206A (et)	2002-06-17

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PL353372A1 (en)	2003-11-17	Substituted heterocyclyl-2h-chromenes
HK1039113A1 (en)	2002-04-12	Benzothieno Ä3,2-CÜpyridines as alpha2 antagonists
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GB9918623D0 (en)	1999-10-13	Lathe
PL343921A1 (en)	2001-05-21	Toolhead
ZA200203582B (en)	2003-11-26	Bicyclic imidazo-5-yl-amine derivatives.
TW401868U (en)	2000-08-11	Improved drill
ZA200200734B (en)	2003-01-28	Spiro compounds.

Legal Events

Date	Code	Title	Description
2011-05-20	PC	Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)	Effective date: 20101001