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GR880100175A - Process of preparing 3-piperidinyl-1,2- benzisoxazoles - Google Patents

Process of preparing 3-piperidinyl-1,2- benzisoxazoles

Info

Publication number
GR880100175A
GR880100175A GR88100175A GR880100175A GR880100175A GR 880100175 A GR880100175 A GR 880100175A GR 88100175 A GR88100175 A GR 88100175A GR 880100175 A GR880100175 A GR 880100175A GR 880100175 A GR880100175 A GR 880100175A
Authority
GR
Greece
Prior art keywords
piperidinyl
benzisoxazoles
preparing
oxyms
halogenphenyl
Prior art date
Application number
GR88100175A
Other languages
Greek (el)
Other versions
GR1000667B (en
Inventor
Edmond Josephine Ludo Kennis
Jan Vandenberk
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of GR880100175A publication Critical patent/GR880100175A/en
Publication of GR1000667B publication Critical patent/GR1000667B/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

The present invention refers to a preparation method of 3-piperidinyl-1.2-benzisoxazoles by cycling of properly substituted (2-halogenphenyl) (4-piperidinyl) methanol oxyms.
GR880100175A 1988-03-21 1988-03-21 Process of preparing 3-piperidinyl-1,2- benzisoxazoles GR1000667B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GR88100175 1988-03-21

Publications (2)

Publication Number Publication Date
GR880100175A true GR880100175A (en) 1990-01-19
GR1000667B GR1000667B (en) 1992-09-25

Family

ID=10938709

Family Applications (1)

Application Number Title Priority Date Filing Date
GR880100175A GR1000667B (en) 1988-03-21 1988-03-21 Process of preparing 3-piperidinyl-1,2- benzisoxazoles

Country Status (1)

Country Link
GR (1) GR1000667B (en)

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4355037A (en) * 1981-11-12 1982-10-19 Hoechst-Roussel Pharmaceuticals 3-(4-Piperidyl)-1,2-benzisoxales
EP0196132A2 (en) * 1985-03-27 1986-10-01 Janssen Pharmaceutica N.V. 1,2-Benzisoxazol-3-yl and 1,2-benzisothiazol-3-yl derivatives

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4355037A (en) * 1981-11-12 1982-10-19 Hoechst-Roussel Pharmaceuticals 3-(4-Piperidyl)-1,2-benzisoxales
EP0196132A2 (en) * 1985-03-27 1986-10-01 Janssen Pharmaceutica N.V. 1,2-Benzisoxazol-3-yl and 1,2-benzisothiazol-3-yl derivatives

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
CLAIMS SEARCHED: ALL *
JOURNAL OF MEDICINAL CHEMISTRY, vol. 28, no. 6, June 1985, pages 761-769, American Chemical Society, Washington, DC, US; J.T. STRUPCZEWSKI et al.: "Synthesis and neuroleptic activity of 3-(1-substituted-4-piperidinyl)-1,2-benzisoxazoles" *

Also Published As

Publication number Publication date
GR1000667B (en) 1992-09-25

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