GEP19971013B - Novel pyridyl and pyrimidyl derivatives process for preparing thereof, and treatment method for mental disorder - Google Patents
Novel pyridyl and pyrimidyl derivatives process for preparing thereof, and treatment method for mental disorderInfo
- Publication number
- GEP19971013B GEP19971013B GEAP19931054A GEAP1993001054A GEP19971013B GE P19971013 B GEP19971013 B GE P19971013B GE AP19931054 A GEAP19931054 A GE AP19931054A GE AP1993001054 A GEAP1993001054 A GE AP1993001054A GE P19971013 B GEP19971013 B GE P19971013B
- Authority
- GE
- Georgia
- Prior art keywords
- hydrogen
- lower alkyl
- halogen
- chem
- preparing
- Prior art date
Links
- 208000020016 psychiatric disease Diseases 0.000 title abstract 2
- 125000004076 pyridyl group Chemical group 0.000 title abstract 2
- 125000000714 pyrimidinyl group Chemical group 0.000 title abstract 2
- 238000004519 manufacturing process Methods 0.000 title 1
- 238000000034 method Methods 0.000 title 1
- 229910052739 hydrogen Chemical group 0.000 abstract 7
- 239000001257 hydrogen Chemical group 0.000 abstract 7
- 125000000217 alkyl group Chemical group 0.000 abstract 6
- 229910052736 halogen Inorganic materials 0.000 abstract 4
- 150000002367 halogens Chemical group 0.000 abstract 4
- 150000002431 hydrogen Chemical group 0.000 abstract 3
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical group [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 1
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 1
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
- 125000000325 methylidene group Chemical group [H]C([H])=* 0.000 abstract 1
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 1
- 229910052760 oxygen Inorganic materials 0.000 abstract 1
- 239000001301 oxygen Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
The present invention concerns novel compounds of the general formula: <CHEM> wherein R1 is halogen or hydrogen and R2 is halogen; X is either oxygen, sulfor or methylene R3 and R4 are the same or different and selected from hydrogen and lower alkyl; n is 2 or 3; A is selected from the following pyrimidyl or pyridyl groups <CHEM> wherein R5 is selected from hydrogen, lower alkyl or halogen; R6 and R7 are the same or different and selected from hydrogen, halogen, lower alkyl, electron donor groups such as lower alkoxy or hydroxy, electron acceptor groups such as cyano, nitro, trifluoromethyl, COOR8, CONR9R10 or CO-B; wherein R8 is hydrogen or lower alkyl; R9 and R10 are the same or different and selected from hydrogen, lower alkyl and cycloalkyl; B is selected from <CHEM> wherein m is 1, 2, 3 or 4.; R11 is selected from hydrogen or lower alkyl, and the pharmacologically active salts thereof. The new compounds are useful for treating mental disorders.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE8803429A SE8803429D0 (en) | 1988-09-28 | 1988-09-28 | NOVEL PYRIDYL AND PYRIMIDYL DERIVATIVES |
Publications (1)
Publication Number | Publication Date |
---|---|
GEP19971013B true GEP19971013B (en) | 1997-11-26 |
Family
ID=74237092
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
GEAP19931054A GEP19971013B (en) | 1988-09-28 | 1993-07-16 | Novel pyridyl and pyrimidyl derivatives process for preparing thereof, and treatment method for mental disorder |
Country Status (2)
Country | Link |
---|---|
GE (1) | GEP19971013B (en) |
UA (1) | UA26426A (en) |
-
1989
- 1989-09-27 UA UA4742280A patent/UA26426A/en unknown
-
1993
- 1993-07-16 GE GEAP19931054A patent/GEP19971013B/en unknown
Also Published As
Publication number | Publication date |
---|---|
UA26426A (en) | 1999-08-30 |
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