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GB9707659D0 - Hepatitis C NS3 Protease inhibitors - Google Patents

Hepatitis C NS3 Protease inhibitors

Info

Publication number
GB9707659D0
GB9707659D0 GBGB9707659.0A GB9707659A GB9707659D0 GB 9707659 D0 GB9707659 D0 GB 9707659D0 GB 9707659 A GB9707659 A GB 9707659A GB 9707659 D0 GB9707659 D0 GB 9707659D0
Authority
GB
United Kingdom
Prior art keywords
hepatitis
protease inhibitors
protease
inhibitors
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
GBGB9707659.0A
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Pasteur Holding Ltd
Original Assignee
Peptide Therapeutics Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Peptide Therapeutics Ltd filed Critical Peptide Therapeutics Ltd
Priority to GBGB9707659.0A priority Critical patent/GB9707659D0/en
Publication of GB9707659D0 publication Critical patent/GB9707659D0/en
Priority to PCT/GB1998/001126 priority patent/WO1998046630A1/en
Priority to JP54364898A priority patent/JP2001521516A/en
Priority to EP98917395A priority patent/EP0975662A1/en
Priority to AU70635/98A priority patent/AU7063598A/en
Pending legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10Tetrapeptides
    • C07K5/1021Tetrapeptides with the first amino acid being acidic
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Molecular Biology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Virology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
GBGB9707659.0A 1997-04-16 1997-04-16 Hepatitis C NS3 Protease inhibitors Pending GB9707659D0 (en)

Priority Applications (5)

Application Number Priority Date Filing Date Title
GBGB9707659.0A GB9707659D0 (en) 1997-04-16 1997-04-16 Hepatitis C NS3 Protease inhibitors
PCT/GB1998/001126 WO1998046630A1 (en) 1997-04-16 1998-04-16 Hepatitis c ns3 protease inhibitors
JP54364898A JP2001521516A (en) 1997-04-16 1998-04-16 Hepatitis C NS3 protease inhibitor
EP98917395A EP0975662A1 (en) 1997-04-16 1998-04-16 Hepatitis c ns3 protease inhibitors
AU70635/98A AU7063598A (en) 1997-04-16 1998-04-16 Hepatitis c ns3 protease inhibitors

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9707659.0A GB9707659D0 (en) 1997-04-16 1997-04-16 Hepatitis C NS3 Protease inhibitors

Publications (1)

Publication Number Publication Date
GB9707659D0 true GB9707659D0 (en) 1997-06-04

Family

ID=10810848

Family Applications (1)

Application Number Title Priority Date Filing Date
GBGB9707659.0A Pending GB9707659D0 (en) 1997-04-16 1997-04-16 Hepatitis C NS3 Protease inhibitors

Country Status (5)

Country Link
EP (1) EP0975662A1 (en)
JP (1) JP2001521516A (en)
AU (1) AU7063598A (en)
GB (1) GB9707659D0 (en)
WO (1) WO1998046630A1 (en)

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* Cited by examiner, † Cited by third party
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US6608027B1 (en) 1999-04-06 2003-08-19 Boehringer Ingelheim (Canada) Ltd Macrocyclic peptides active against the hepatitis C virus
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US7122627B2 (en) 1999-07-26 2006-10-17 Bristol-Myers Squibb Company Lactam inhibitors of Hepatitis C virus NS3 protease
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US6846806B2 (en) 2000-10-23 2005-01-25 Bristol-Myers Squibb Company Peptide inhibitors of Hepatitis C virus NS3 protein
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US7119072B2 (en) 2002-01-30 2006-10-10 Boehringer Ingelheim (Canada) Ltd. Macrocyclic peptides active against the hepatitis C virus
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ATE481106T1 (en) 2002-05-20 2010-10-15 Bristol Myers Squibb Co HETEROCYCLIC SULFONAMIDE HEPATITIS C VIRUS INHIBITORS
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US7642235B2 (en) 2003-09-22 2010-01-05 Boehringer Ingelheim International Gmbh Macrocyclic peptides active against the hepatitis C virus
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US7470664B2 (en) 2005-07-20 2008-12-30 Merck & Co., Inc. HCV NS3 protease inhibitors
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EP0732399A3 (en) * 1990-03-05 1997-03-12 Cephalon Inc Chymotrypsin-like proteases and their inhibitors
IT1277914B1 (en) * 1995-08-22 1997-11-12 Angeletti P Ist Richerche Bio PROCEDURE TO PRODUCE - IN PURE FORM AND IN HIGH QUANTITIES - POLYPEPTIDES WITH THE PROTEOLYTIC ACTIVITY OF THE NS3 PROTEASE OF HCV, AND
ATE212037T1 (en) * 1996-10-18 2002-02-15 Vertex Pharma INHIBITORS OF SERINE PROTEASES, IN PARTICULAR THE NS3 PROTEASE OF THE HEPATITIS C VIRUS

Also Published As

Publication number Publication date
EP0975662A1 (en) 2000-02-02
JP2001521516A (en) 2001-11-06
WO1998046630A1 (en) 1998-10-22
AU7063598A (en) 1998-11-11

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