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FR2414511A1 - Nouveaux 1, 2, 3, 4-tetrahydropyrido(4', 3' : 4,5)thiazolo(3,2-a)benzimidazoles utiles notamment comme anti-inflammatoires et leur procede de preparation - Google Patents

Nouveaux 1, 2, 3, 4-tetrahydropyrido(4', 3' : 4,5)thiazolo(3,2-a)benzimidazoles utiles notamment comme anti-inflammatoires et leur procede de preparation

Info

Publication number
FR2414511A1
FR2414511A1 FR7836900A FR7836900A FR2414511A1 FR 2414511 A1 FR2414511 A1 FR 2414511A1 FR 7836900 A FR7836900 A FR 7836900A FR 7836900 A FR7836900 A FR 7836900A FR 2414511 A1 FR2414511 A1 FR 2414511A1
Authority
FR
France
Prior art keywords
inflammatory
tetrahydropyrido
thiazolo
preparation
new
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7836900A
Other languages
English (en)
Other versions
FR2414511B1 (fr
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
ER Squibb and Sons LLC
Original Assignee
ER Squibb and Sons LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ER Squibb and Sons LLC filed Critical ER Squibb and Sons LLC
Publication of FR2414511A1 publication Critical patent/FR2414511A1/fr
Application granted granted Critical
Publication of FR2414511B1 publication Critical patent/FR2414511B1/fr
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
    • C07D513/14—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D211/74—Oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Les médicaments selon l'invention sont des 1,2,3,4-tétrahydropyridoØ4',3':4,5õthiazoloØ3,2-aõbenzimidazoles utiles notamment comme anti-inflammatoires de formule générale :
FR7836900A 1978-01-16 1978-12-29 Nouveaux 1, 2, 3, 4-tetrahydropyrido(4', 3' : 4,5)thiazolo(3,2-a)benzimidazoles utiles notamment comme anti-inflammatoires et leur procede de preparation Granted FR2414511A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/869,737 US4122083A (en) 1978-01-16 1978-01-16 1,2,3,4-Tetrahydropyrido[4',3':4.5]thiazolo-[3,2-a]benzimidazoles

Publications (2)

Publication Number Publication Date
FR2414511A1 true FR2414511A1 (fr) 1979-08-10
FR2414511B1 FR2414511B1 (fr) 1981-02-27

Family

ID=25354170

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7836900A Granted FR2414511A1 (fr) 1978-01-16 1978-12-29 Nouveaux 1, 2, 3, 4-tetrahydropyrido(4', 3' : 4,5)thiazolo(3,2-a)benzimidazoles utiles notamment comme anti-inflammatoires et leur procede de preparation

Country Status (6)

Country Link
US (1) US4122083A (fr)
JP (1) JPS54100370A (fr)
DE (1) DE2856792A1 (fr)
FR (1) FR2414511A1 (fr)
GB (1) GB2012747B (fr)
IT (1) IT1114703B (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1131226A (fr) * 1978-09-28 1982-09-07 Tomohiko Munakata Composes heterocycliques
US7485637B2 (en) * 2005-01-04 2009-02-03 Hoffmann-La Roche Inc. Benzoyl-tetrahydropiperidine derivatives

Also Published As

Publication number Publication date
GB2012747B (en) 1982-08-04
IT7947620A0 (it) 1979-01-12
IT1114703B (it) 1986-01-27
JPS54100370A (en) 1979-08-08
US4122083A (en) 1978-10-24
DE2856792A1 (de) 1979-07-19
GB2012747A (en) 1979-08-01
FR2414511B1 (fr) 1981-02-27

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