FR2409267A1 - Derives de 4-amino-2-piperidinoquinazoline, leur procede de production et composition pharmaceutique les contenant - Google Patents
Derives de 4-amino-2-piperidinoquinazoline, leur procede de production et composition pharmaceutique les contenantInfo
- Publication number
- FR2409267A1 FR2409267A1 FR7832235A FR7832235A FR2409267A1 FR 2409267 A1 FR2409267 A1 FR 2409267A1 FR 7832235 A FR7832235 A FR 7832235A FR 7832235 A FR7832235 A FR 7832235A FR 2409267 A1 FR2409267 A1 FR 2409267A1
- Authority
- FR
- France
- Prior art keywords
- derivatives
- piperidinoquinazoline
- amino
- pharmaceutical composition
- composition containing
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/40—Oxygen atoms
- C07D211/44—Oxygen atoms attached in position 4
- C07D211/46—Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB4758377 | 1977-11-16 | ||
| GB7844533A GB2010824B (en) | 1977-11-16 | 1978-11-15 | Therapeutic agents |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| FR2409267A1 true FR2409267A1 (fr) | 1979-06-15 |
| FR2409267B1 FR2409267B1 (de) | 1981-02-27 |
Family
ID=26266083
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR7832235A Granted FR2409267A1 (fr) | 1977-11-16 | 1978-11-15 | Derives de 4-amino-2-piperidinoquinazoline, leur procede de production et composition pharmaceutique les contenant |
Country Status (12)
| Country | Link |
|---|---|
| JP (1) | JPS5481282A (de) |
| AT (1) | AT365183B (de) |
| AU (1) | AU509348B2 (de) |
| BE (1) | BE872023A (de) |
| CA (1) | CA1088068A (de) |
| CH (1) | CH637131A5 (de) |
| DE (1) | DE2849392A1 (de) |
| FR (1) | FR2409267A1 (de) |
| GB (1) | GB2010824B (de) |
| LU (1) | LU80531A1 (de) |
| NL (1) | NL174646C (de) |
| SE (1) | SE7811770L (de) |
Cited By (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2447919A1 (fr) * | 1979-01-31 | 1980-08-29 | Pfizer | Nouvelles quinazolines anti-hypertensives, leur procede de production et composition pharmaceutique les contenant |
| FR2481278A1 (fr) * | 1980-04-28 | 1981-10-30 | Synthelabo | Nouveaux derives de piperidine, leur procede de preparation et leur application en therapeutique |
| FR2514353A2 (fr) * | 1980-04-28 | 1983-04-15 | Synthelabo | Derives de piperidine et leur application en therapeutique |
| FR2597479A1 (fr) * | 1986-03-13 | 1987-10-23 | Kotobuki Seiyaku Co Ltd | Derives de la quinazoline utilises comme agents anti-hypertensifs, et procede de preparation de ces composes. |
-
1978
- 1978-10-24 CA CA314,082A patent/CA1088068A/en not_active Expired
- 1978-11-14 NL NLAANVRAGE7811236,A patent/NL174646C/xx not_active IP Right Cessation
- 1978-11-14 AU AU41576/78A patent/AU509348B2/en not_active Expired
- 1978-11-14 BE BE191743A patent/BE872023A/xx not_active IP Right Cessation
- 1978-11-14 DE DE19782849392 patent/DE2849392A1/de not_active Withdrawn
- 1978-11-14 SE SE7811770A patent/SE7811770L/xx unknown
- 1978-11-15 JP JP14094678A patent/JPS5481282A/ja active Granted
- 1978-11-15 LU LU80531A patent/LU80531A1/fr unknown
- 1978-11-15 FR FR7832235A patent/FR2409267A1/fr active Granted
- 1978-11-15 AT AT0816678A patent/AT365183B/de active
- 1978-11-15 CH CH1175578A patent/CH637131A5/de not_active IP Right Cessation
- 1978-11-15 GB GB7844533A patent/GB2010824B/en not_active Expired
Cited By (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2447919A1 (fr) * | 1979-01-31 | 1980-08-29 | Pfizer | Nouvelles quinazolines anti-hypertensives, leur procede de production et composition pharmaceutique les contenant |
| FR2481278A1 (fr) * | 1980-04-28 | 1981-10-30 | Synthelabo | Nouveaux derives de piperidine, leur procede de preparation et leur application en therapeutique |
| FR2514353A2 (fr) * | 1980-04-28 | 1983-04-15 | Synthelabo | Derives de piperidine et leur application en therapeutique |
| FR2597479A1 (fr) * | 1986-03-13 | 1987-10-23 | Kotobuki Seiyaku Co Ltd | Derives de la quinazoline utilises comme agents anti-hypertensifs, et procede de preparation de ces composes. |
Also Published As
| Publication number | Publication date |
|---|---|
| SE7811770L (sv) | 1979-05-17 |
| ATA816678A (de) | 1981-05-15 |
| NL174646C (nl) | 1984-07-16 |
| GB2010824B (en) | 1982-06-16 |
| FR2409267B1 (de) | 1981-02-27 |
| NL7811236A (nl) | 1979-05-18 |
| CH637131A5 (de) | 1983-07-15 |
| AT365183B (de) | 1981-12-28 |
| LU80531A1 (fr) | 1980-06-05 |
| JPS5623991B2 (de) | 1981-06-03 |
| NL174646B (nl) | 1984-02-16 |
| GB2010824A (en) | 1979-07-04 |
| BE872023A (fr) | 1979-05-14 |
| AU509348B2 (en) | 1980-05-08 |
| DE2849392A1 (de) | 1979-05-23 |
| AU4157678A (en) | 1979-05-24 |
| CA1088068A (en) | 1980-10-21 |
| JPS5481282A (en) | 1979-06-28 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| ST | Notification of lapse |