FR2362121A1 - SOMATOSTATIN APPROVED, AND PREPARATION INTERMEDIARIES - Google Patents
SOMATOSTATIN APPROVED, AND PREPARATION INTERMEDIARIESInfo
- Publication number
- FR2362121A1 FR2362121A1 FR7706775A FR7706775A FR2362121A1 FR 2362121 A1 FR2362121 A1 FR 2362121A1 FR 7706775 A FR7706775 A FR 7706775A FR 7706775 A FR7706775 A FR 7706775A FR 2362121 A1 FR2362121 A1 FR 2362121A1
- Authority
- FR
- France
- Prior art keywords
- preparation
- somatostatin
- intermediaries
- approved
- homologues
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- 102000005157 Somatostatin Human genes 0.000 title abstract 2
- 108010056088 Somatostatin Proteins 0.000 title abstract 2
- NHXLMOGPVYXJNR-ATOGVRKGSA-N somatostatin Chemical compound C([C@H]1C(=O)N[C@H](C(N[C@@H](CO)C(=O)N[C@@H](CSSC[C@@H](C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CC=2C=CC=CC=2)C(=O)N[C@@H](CC=2C=CC=CC=2)C(=O)N[C@@H](CC=2C3=CC=CC=C3NC=2)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N1)[C@@H](C)O)NC(=O)CNC(=O)[C@H](C)N)C(O)=O)=O)[C@H](O)C)C1=CC=CC=C1 NHXLMOGPVYXJNR-ATOGVRKGSA-N 0.000 title abstract 2
- 229960000553 somatostatin Drugs 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/655—Somatostatins
- C07K14/6555—Somatostatins at least 1 amino acid in D-form
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biophysics (AREA)
- Gastroenterology & Hepatology (AREA)
- Zoology (AREA)
- Biochemistry (AREA)
- Toxicology (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Endocrinology (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
L'invention concerne des homologues de somatostatine, leur préparation et les intermédiaires necessaires à cette préparation. On prépare un composé de formule :The invention relates to homologues of somatostatin, their preparation and the intermediates necessary for this preparation. A compound of formula is prepared:
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US66445276A | 1976-03-08 | 1976-03-08 | |
| US05/763,943 US4093574A (en) | 1977-02-02 | 1977-02-02 | Somatostatin analogs and intermediates thereto |
| US05/763,944 US4087390A (en) | 1977-02-02 | 1977-02-02 | Somatostatin analogs and intermediates thereto |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| FR2362121A1 true FR2362121A1 (en) | 1978-03-17 |
Family
ID=27418106
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR7706775A Withdrawn FR2362121A1 (en) | 1976-03-08 | 1977-03-08 | SOMATOSTATIN APPROVED, AND PREPARATION INTERMEDIARIES |
Country Status (6)
| Country | Link |
|---|---|
| JP (1) | JPS52116489A (en) |
| DE (1) | DE2709877A1 (en) |
| FR (1) | FR2362121A1 (en) |
| GB (1) | GB1577414A (en) |
| IL (1) | IL51508A0 (en) |
| NL (1) | NL7702447A (en) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2439181A1 (en) * | 1978-10-02 | 1980-05-16 | Lilly Co Eli | SOMATOSTATIN-RELATED PEPTIDES AND THEIR THERAPEUTIC USE |
-
1977
- 1977-02-21 IL IL51508A patent/IL51508A0/en unknown
- 1977-03-03 GB GB9091/77A patent/GB1577414A/en not_active Expired
- 1977-03-07 NL NL7702447A patent/NL7702447A/en not_active Application Discontinuation
- 1977-03-07 DE DE19772709877 patent/DE2709877A1/en not_active Withdrawn
- 1977-03-08 JP JP2587277A patent/JPS52116489A/en active Pending
- 1977-03-08 FR FR7706775A patent/FR2362121A1/en not_active Withdrawn
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2439181A1 (en) * | 1978-10-02 | 1980-05-16 | Lilly Co Eli | SOMATOSTATIN-RELATED PEPTIDES AND THEIR THERAPEUTIC USE |
| EP0011366A3 (en) * | 1978-10-02 | 1982-02-10 | Eli Lilly And Company | Synthetic peptides, their preparation, pharmaceutical formulations containing them and intermediates for their preparation |
Also Published As
| Publication number | Publication date |
|---|---|
| IL51508A0 (en) | 1977-06-30 |
| DE2709877A1 (en) | 1977-09-15 |
| JPS52116489A (en) | 1977-09-29 |
| GB1577414A (en) | 1980-10-22 |
| NL7702447A (en) | 1977-09-12 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| ST | Notification of lapse |