FR1439514A - Procédé de préparation de 3-oxo-4.6-bis-déhydro-6-halogéno-9beta. 10alpha-stéroïdes - Google Patents

Procédé de préparation de 3-oxo-4.6-bis-déhydro-6-halogéno-9beta. 10alpha-stéroïdes

Info

Publication number: FR1439514A
Authority: FR; France
Prior art keywords: 9beta; 10alpha; dehydro; halogeno; steroids
Prior art date: 1965-01-22
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired

Application number

FR22465A

Other languages

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Koninklijke Philips NV

Original Assignee

Philips Gloeilampenfabrieken NV

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1965-01-22

Filing date

1965-06-26

Publication date

1966-05-20

1965-01-22 Priority claimed from GB291965A external-priority patent/GB1139411A/en

1965-05-31 Priority claimed from CH846564A external-priority patent/CH454842A/de

1965-06-26 Application filed by Philips Gloeilampenfabrieken NV filed Critical Philips Gloeilampenfabrieken NV

1966-05-20 Application granted granted Critical

1966-05-20 Publication of FR1439514A publication Critical patent/FR1439514A/fr

Status Expired legal-status Critical Current

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/568—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/568—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
- A61K31/569—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone substituted in position 17 alpha, e.g. ethisterone
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J15/00—Stereochemically pure steroids containing carbon, hydrogen, halogen or oxygen having a partially or totally inverted skeleton, e.g. retrosteroids, L-isomers
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J5/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J75/00—Processes for the preparation of steroids in general

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Epidemiology (AREA)
Pharmacology & Pharmacy (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Steroid Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

FR22465A 1965-01-22 1965-06-26 Procédé de préparation de 3-oxo-4.6-bis-déhydro-6-halogéno-9beta. 10alpha-stéroïdes Expired FR1439514A (fr)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB291965A GB1139411A (en)	1965-01-22	1965-01-22	Preparation of 10-‡-methyl steroids
CH846564A CH454842A (de)	1965-05-31	1965-05-31	Verfahren zur Herstellung von neuen 9B,10a-Steroiden

Publications (1)

Publication Number	Publication Date
FR1439514A true FR1439514A (fr)	1966-05-20

Family

ID=25703347

Family Applications (3)

Application Number	Title	Priority Date	Filing Date
FR20951A Expired FR4631M (fr)	1965-01-22	1965-06-16
FR22045A Expired FR1446515A (fr)	1965-01-22	1965-06-24	Procédé pour la préparation de nouveaux 9beta, 10alpha-stéroïdes
FR22465A Expired FR1439514A (fr)	1965-01-22	1965-06-26	Procédé de préparation de 3-oxo-4.6-bis-déhydro-6-halogéno-9beta. 10alpha-stéroïdes

Family Applications Before (2)

Application Number	Title	Priority Date	Filing Date
FR20951A Expired FR4631M (fr)	1965-01-22	1965-06-16
FR22045A Expired FR1446515A (fr)	1965-01-22	1965-06-24	Procédé pour la préparation de nouveaux 9beta, 10alpha-stéroïdes

Country Status (14)

Country	Link
US (2)	US3304314A (fr)
AT (1)	AT261129B (fr)
BE (2)	BE665762A (fr)
BR (1)	BR6570589D0 (fr)
CH (1)	CH464188A (fr)
DE (2)	DE1518994A1 (fr)
DK (2)	DK120337B (fr)
ES (1)	ES314639A1 (fr)
FI (1)	FI41743B (fr)
FR (3)	FR4631M (fr)
GB (1)	GB1087920A (fr)
IL (2)	IL23629A (fr)
NL (2)	NL6508148A (fr)
SE (1)	SE331277B (fr)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
BE667121A (fr) *	1964-10-28
IL23629A (en) *	1965-01-22	1969-01-29	Hoffmann La Roche	9beta,10alpha-steroids and process for the manufacture thereof
GB1228801A (fr) *	1967-07-11	1971-04-21
US3937700A (en) *	1970-03-04	1976-02-10	U.S. Philips Corporation	Novel 1,2-methylene-17α-acyloxy (or improved hydroxy)-9β, 10α-steroid compounds of the pregnane series, pharmaceutic preparations on the basis of the novel compounds and methods of producing said compounds and preparations
US4898694A (en) *	1987-11-25	1990-02-06	Schwartz Arthur G	17-Hydroxy-steroids
US20070082876A1 (en) *	2005-09-30	2007-04-12	Solvay Pharmaceuticals Gmbh	Novel C18 modified retrosteroids as progesterone receptor modulator compounds
US20070212751A1 (en) *	2006-01-18	2007-09-13	Solvay Pharmaceuticals Gmbh	Microbial method for the 11beta hydroxylation of 9beta, 10alpha-steriods

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
NL252417A (fr) *	1959-06-08
US3258473A (en) *	1963-10-04	1966-06-28	Syntex Corp	17-dihaloacetate esters of 17alpha-hydroxy-21-desoxypregnane derivatives
IL23629A (en) *	1965-01-22	1969-01-29	Hoffmann La Roche	9beta,10alpha-steroids and process for the manufacture thereof

1965
- 1965-05-30 IL IL6523629A patent/IL23629A/xx unknown
- 1965-06-03 DE DE19651518994 patent/DE1518994A1/de active Pending
- 1965-06-16 FR FR20951A patent/FR4631M/fr not_active Expired
- 1965-06-22 BE BE665762D patent/BE665762A/xx unknown
- 1965-06-22 BR BR170589/65A patent/BR6570589D0/pt unknown
- 1965-06-23 CH CH876665A patent/CH464188A/de unknown
- 1965-06-23 FI FI1505/65A patent/FI41743B/fi active
- 1965-06-23 GB GB26557/65A patent/GB1087920A/en not_active Expired
- 1965-06-23 SE SE08369/65A patent/SE331277B/xx unknown
- 1965-06-23 IL IL6523785A patent/IL23785A/xx unknown
- 1965-06-23 DK DK319165AA patent/DK120337B/da unknown
- 1965-06-24 AT AT573665A patent/AT261129B/de active
- 1965-06-24 US US466818A patent/US3304314A/en not_active Expired - Lifetime
- 1965-06-24 FR FR22045A patent/FR1446515A/fr not_active Expired
- 1965-06-24 US US466817A patent/US3423433A/en not_active Expired - Lifetime
- 1965-06-24 DE DE19651543274 patent/DE1543274A1/de active Pending
- 1965-06-25 DK DK324365AA patent/DK123352B/da unknown
- 1965-06-25 ES ES0314639A patent/ES314639A1/es not_active Expired
- 1965-06-25 NL NL6508148A patent/NL6508148A/xx unknown
- 1965-06-25 NL NL6508179A patent/NL6508179A/xx unknown
- 1965-06-26 FR FR22465A patent/FR1439514A/fr not_active Expired
- 1965-06-28 BE BE666060A patent/BE666060A/xx unknown

Also Published As

Publication number	Publication date
US3423433A (en)	1969-01-21
FR1446515A (fr)	1966-07-22
BE666060A (fr)	1965-12-28
BE665762A (fr)	1965-12-22
BR6570589D0 (pt)	1973-08-02
DK123352B (da)	1972-06-12
NL6508179A (fr)	1965-12-27
IL23629A (en)	1969-01-29
NL6508148A (fr)	1966-06-27
IL23785A (en)	1969-09-25
GB1087920A (en)	1967-10-18
DE1518994A1 (de)	1969-09-25
AT261129B (de)	1968-04-10
ES314639A1 (es)	1966-02-16
US3304314A (en)	1967-02-14
CH464188A (de)	1968-10-31
SE331277B (fr)	1970-12-21
FR4631M (fr)	1966-11-28
FI41743B (fr)	1969-10-31
DE1543274A1 (de)	1969-07-24
DK120337B (da)	1971-05-17

Publication	Publication Date	Title
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CH457480A (fr)	1968-06-15	Procédé de préparation de nitroparaphénylènediamines
FR1439514A (fr)	1966-05-20	Procédé de préparation de 3-oxo-4.6-bis-déhydro-6-halogéno-9beta. 10alpha-stéroïdes
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OA02691A (fr)	1970-12-15	Procédé de préparation de 2-alcanoyl-4-halogéno-5-acylaminophénols.