[go: up one dir, main page]

FI956298L - 3-fenyl-isokinolin-1(2H)-oner, och framställning och terapeutisk användning av dessa - Google Patents

3-fenyl-isokinolin-1(2H)-oner, och framställning och terapeutisk användning av dessa Download PDF

Info

Publication number
FI956298L
FI956298L FI956298A FI956298A FI956298L FI 956298 L FI956298 L FI 956298L FI 956298 A FI956298 A FI 956298A FI 956298 A FI956298 A FI 956298A FI 956298 L FI956298 L FI 956298L
Authority
FI
Finland
Prior art keywords
phenylisoquinolin
ones
preparation
therapeutic use
therapeutic
Prior art date
Application number
FI956298A
Other languages
English (en)
Finnish (fi)
Other versions
FI956298A0 (sv
Inventor
Mireille Sevrin
Benoit Marabout
Jacques Froissant
Catherine Guinot
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of FI956298A0 publication Critical patent/FI956298A0/sv
Publication of FI956298L publication Critical patent/FI956298L/sv

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D217/00Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/22Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D217/00Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/22Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
    • C07D217/24Oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/16Otologicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
FI956298A 1994-12-29 1995-12-28 3-fenyl-isokinolin-1(2H)-oner, och framställning och terapeutisk användning av dessa FI956298L (sv)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9415837A FR2728900B1 (fr) 1994-12-29 1994-12-29 Derives de 3-phenylisoquinolein-1(2h)-one, leur preparation et leur application en therapeutique

Publications (2)

Publication Number Publication Date
FI956298A0 FI956298A0 (sv) 1995-12-28
FI956298L true FI956298L (sv) 1996-06-30

Family

ID=9470390

Family Applications (1)

Application Number Title Priority Date Filing Date
FI956298A FI956298L (sv) 1994-12-29 1995-12-28 3-fenyl-isokinolin-1(2H)-oner, och framställning och terapeutisk användning av dessa

Country Status (22)

Country Link
US (1) US5665733A (sv)
EP (1) EP0719764B1 (sv)
JP (1) JPH08239365A (sv)
KR (1) KR960022472A (sv)
CN (1) CN1131150A (sv)
AR (1) AR002016A1 (sv)
AT (1) ATE172966T1 (sv)
AU (1) AU698595B2 (sv)
BR (1) BR9506106A (sv)
CA (1) CA2166234A1 (sv)
CO (1) CO4700298A1 (sv)
CZ (1) CZ348995A3 (sv)
DE (1) DE69505780D1 (sv)
FI (1) FI956298L (sv)
FR (1) FR2728900B1 (sv)
HU (1) HU215394B (sv)
IL (1) IL116590A0 (sv)
NO (1) NO955326L (sv)
NZ (1) NZ280765A (sv)
PL (1) PL312079A1 (sv)
SK (1) SK165795A3 (sv)
ZA (1) ZA9511046B (sv)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2750427B1 (fr) * 1996-06-28 1998-08-07 Synthelabo Derives de 1-oxo-1, 2-dihydroisoquinoleine-4-propanamide, leur preparation et leur application en therapeutique
FR2772758B1 (fr) * 1997-12-22 2000-02-04 Synthelabo Derives de 1-oxo-1,2-dihydroisoquinoleine-4-propanamide, leur preparation et leur application en therapeutique
ES2361924T3 (es) * 2002-12-20 2011-06-24 X-Ceptor Therapeutics, Inc. Derivados de isoquinolinona y su uso como agentes terapéuticos.
GB0420722D0 (en) * 2004-09-17 2004-10-20 Addex Pharmaceuticals Sa Novel allosteric modulators
KR20090035744A (ko) * 2006-08-10 2009-04-10 페레르 인터내쇼날 에스.에이. Gaba 수용체의 친화력을 갖는 1h-퀴놀린-4-원 화합물,제조방법, 사용방법 및 조성물
EP1886996A1 (en) * 2006-08-10 2008-02-13 Ferrer Internacional, S.A. 1H-Quinolin-4-one compounds, with affinity for the GABA receptor, processes, uses and compositions
US8741917B2 (en) 2009-01-15 2014-06-03 Rutgers, The State University Of New Jersey Benzo [C] phenanthridines as antimicrobial agents
US20120059026A1 (en) 2009-04-30 2012-03-08 University Of Medicine And Dentistry Of New Jersey Antimicrobial agents
FR2956816B1 (fr) * 2010-03-01 2012-05-18 Univ Joseph Fourier Utilisation de quinolones pour la preparation de medicaments, nouvelles quinolones et leur procede de synthese
US8933096B2 (en) 2010-06-09 2015-01-13 Rugers, The State University of New Jersey Antimicrobial agents
CA2803890A1 (en) 2010-06-25 2011-12-29 Rutgers, The State University Of New Jersey Antimicrobial agents
WO2013106756A2 (en) 2012-01-13 2013-07-18 Rutgers, The State University Of New Jersey Antimicrobial agents
US9475783B2 (en) 2012-03-21 2016-10-25 Rutgers, The State University Of New Jersey Antimicrobial agents
US9458150B2 (en) 2013-11-08 2016-10-04 Rutgers, The State University Of New Jersey Antimicrobial agents
US10513528B2 (en) 2016-02-25 2019-12-24 Taxis Pharmaceuticals, Inc. Synthetic processes and intermediates
CA3058183A1 (en) 2017-03-30 2018-10-04 Taxis Pharmaceuticals, Inc. Synthetic processes and synthetic intermediates
TW202202495A (zh) * 2020-03-26 2022-01-16 匈牙利商羅特格登公司 作為gamma-胺基丁酸A受體次單元alpha 5受體調節劑之㖠啶及吡啶并〔3,4-c〕嗒𠯤衍生物
EP4126858A1 (en) * 2020-03-26 2023-02-08 Richter Gedeon Nyrt. Dihydro-2-pyrrolo[3,4-c]pyridine derivatives as gabaa a5 receptor modulators

Also Published As

Publication number Publication date
ZA9511046B (en) 1996-07-11
CZ348995A3 (en) 1996-07-17
FR2728900A1 (fr) 1996-07-05
CN1131150A (zh) 1996-09-18
HUT74187A (en) 1996-11-28
AU4071295A (en) 1996-07-04
CA2166234A1 (en) 1996-06-30
HU9503848D0 (en) 1996-02-28
FR2728900B1 (fr) 1997-01-31
JPH08239365A (ja) 1996-09-17
PL312079A1 (en) 1996-07-08
KR960022472A (ko) 1996-07-18
EP0719764A1 (fr) 1996-07-03
CO4700298A1 (es) 1998-12-29
FI956298A0 (sv) 1995-12-28
ATE172966T1 (de) 1998-11-15
HU215394B (hu) 1998-12-28
EP0719764B1 (fr) 1998-11-04
AR002016A1 (es) 1998-01-07
BR9506106A (pt) 1997-12-23
NZ280765A (en) 1996-08-27
AU698595B2 (en) 1998-11-05
IL116590A0 (en) 1996-03-31
SK165795A3 (en) 1996-07-03
US5665733A (en) 1997-09-09
DE69505780D1 (de) 1998-12-10
NO955326L (no) 1996-07-01
NO955326D0 (no) 1995-12-28

Similar Documents

Publication Publication Date Title
FI955235L (sv) Oxazolidindionderivat, deras framställning och användning
DE69529598D1 (de) Arzneimittelenthaltende Manschette
EE200000658A (et) CD23 antikehad, nende derivaadid ja nende terapeutiline kasutamine
DK1019358T4 (da) 3,3-diarylpropylaminer, deres anvendelse og fremstilling
EE04151B1 (et) Atsüülpiperasinüülpürimidiinide derivaadid, nendevalmistamine ja kasutamine ravimitena
FI956298L (sv) 3-fenyl-isokinolin-1(2H)-oner, och framställning och terapeutisk användning av dessa
EE200000621A (et) Pikornaviirusevastased ühendid, nende valmistamine ja kasutamine
EE04497B1 (et) Püridopüranoasepiini derivaadid, nende valmistamine ja terapeutiline kasutamine
FI972245A0 (sv) Mesomonojodsubstituerade tetramakrocykliska föreningar samt förfarande för framställning och användning därav
ID18679A (id) Penggunaan terapi lanjutan
FI970997L (sv) Bensocykloalkenföreningar, deras framställning och användning
NO992676D0 (no) 1,4-diazabicyklo[2,2,2]okt-2-ylmetylderivater, deres fremstilling og terapeutiske anvendelse
NO962477D0 (no) Benzamidderivater, deres fremstilling og deres terapautiske anvendelse
EE200000207A (et) 8-asabitsüklo[3.2.1]oktaan-3-metaanamiini derivaadid, nende valmistamine ja terapeutiline kasutamine
FI956015L (sv) Användning av 5-acyl-1,4-dihydropyridiner
FI970750L (sv) Indol-2,3-dion-oximderivat, framställning och användning av dem
EE200000018A (et) 6-pürrolidiin-2-üülpüridiinid, nende valmistamine ja terapeutiline kasutamine
FI971317A (sv) Nya heterocykliska, substituerade imidazolokinoxalinoner, framställning och användning av dem
FI956251L (sv) 1-oxo-2-(fenylsulfonylamino)-pentylpiperidinderivat, framställning och terapeutisk användning av dessa
ATE198192T1 (de) Benzolsulfonamidderivate, ihre herstellung und ihre therapeutische verwendung
FI965172L (sv) Nya amido-kinoxalindioner, framställning och användning av dem
FI954141L (sv) Oxazolokinolinonderivat, deras framställning och deras användning i terapi
EE9800153A (et) 5-naftalen-1-üül-1,3-dioksaani derivaadid, nende valmistamine ja terapeutiline kasutamine
NO950560D0 (no) Piperazinderivater, deres fremstilling og terapautiske anvendelse
EE9900560A (et) 5-naftaleen-1-üül-1,3-dioksaani derivaadid, nende valmistamine ja terapeutiline kasutamine

Legal Events

Date Code Title Description
FD Application lapsed