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FI824474L - Nya derivat av bicykliska aminosyror, aemnen som innehaoller dessa och deras anvaendning samt nya bicykliska aminosyror saosom mellansteg och foerfarande foer deras framstaellning - Google Patents

Nya derivat av bicykliska aminosyror, aemnen som innehaoller dessa och deras anvaendning samt nya bicykliska aminosyror saosom mellansteg och foerfarande foer deras framstaellning

Info

Publication number
FI824474L
FI824474L FI824474A FI824474A FI824474L FI 824474 L FI824474 L FI 824474L FI 824474 A FI824474 A FI 824474A FI 824474 A FI824474 A FI 824474A FI 824474 L FI824474 L FI 824474L
Authority
FI
Finland
Prior art keywords
aminosyror
nya
och
deras
mellansteg
Prior art date
Application number
FI824474A
Other languages
English (en)
Other versions
FI80017B (fi
FI824474A0 (fi
FI80017C (fi
Inventor
Hansjoerg Urbach
Rainer Henning
Volker Teetz
Rolf Geiger
Reinhard Becker
Holger Gaul
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=25798350&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FI824474(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from DE19813151690 external-priority patent/DE3151690A1/de
Priority claimed from DE19823210701 external-priority patent/DE3210701A1/de
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of FI824474A0 publication Critical patent/FI824474A0/fi
Publication of FI824474L publication Critical patent/FI824474L/fi
Priority to FI883456A priority Critical patent/FI80675C/fi
Publication of FI80017B publication Critical patent/FI80017B/fi
Application granted granted Critical
Publication of FI80017C publication Critical patent/FI80017C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/32—Oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20—Oxygen atoms
    • C07D215/22—Oxygen atoms attached in position 2 or 4
    • C07D215/227—Oxygen atoms attached in position 2 or 4 only one oxygen atom which is attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10—Antioedematous agents; Diuretics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/32—Oxygen atoms
    • C07D209/34—Oxygen atoms in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/022—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
    • C07K5/0222—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Cardiology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Peptides Or Proteins (AREA)
  • Indole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
FI824474A 1981-12-29 1982-12-27 Foerfarande foer framstaellning av azabicykloalkankarboxylsyraderivat. FI80017C (fi)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FI883456A FI80675C (fi) 1981-12-29 1988-07-21 Azabicykloalkankarboxylsyraderivat och foerfarande foer deras framstaellning.

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE3151690 1981-12-29
DE19813151690 DE3151690A1 (de) 1981-12-29 1981-12-29 "neue derivate bicyclischer aminosaeuren, verfahren zu ihrer herstellung, diese enthaltende mittel und deren verwendung sowie neue bicyclische aminosaeuren als zwischenstufen und verfahren zu deren herstellung"
DE19823210701 DE3210701A1 (de) 1982-03-24 1982-03-24 2-azabicycloalkan-3-carbonsaeuren und verfahren zu ihrer herstellung
DE3210701 1982-03-24

Publications (4)

Publication Number Publication Date
FI824474A0 FI824474A0 (fi) 1982-12-27
FI824474L true FI824474L (fi) 1983-06-30
FI80017B FI80017B (fi) 1989-12-29
FI80017C FI80017C (fi) 1990-04-10

Family

ID=25798350

Family Applications (1)

Application Number Title Priority Date Filing Date
FI824474A FI80017C (fi) 1981-12-29 1982-12-27 Foerfarande foer framstaellning av azabicykloalkankarboxylsyraderivat.

Country Status (27)

Country Link
US (3) US5008400A (fi)
EP (1) EP0084164B1 (fi)
JP (3) JPS58118569A (fi)
KR (1) KR890003424B1 (fi)
AR (1) AR247571A1 (fi)
AU (1) AU559140B2 (fi)
BG (1) BG60936B2 (fi)
CA (1) CA1341296C (fi)
CS (1) CS409591A3 (fi)
DE (2) DE3275293D1 (fi)
DK (2) DK170444B1 (fi)
DZ (1) DZ490A1 (fi)
ES (2) ES8308850A1 (fi)
FI (1) FI80017C (fi)
GR (1) GR78413B (fi)
HK (1) HK74989A (fi)
HU (1) HU194167B (fi)
IE (1) IE55867B1 (fi)
IL (1) IL67572A (fi)
LU (1) LU88263I2 (fi)
MA (1) MA19672A1 (fi)
NL (1) NL930048I2 (fi)
NO (1) NO156786C (fi)
NZ (1) NZ202903A (fi)
PH (2) PH18918A (fi)
PT (1) PT76052B (fi)
SG (1) SG1389G (fi)

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KR890003424B1 (ko) 1989-09-20
AU559140B2 (en) 1987-02-26
BG60936B2 (bg) 1996-06-28
US4933361A (en) 1990-06-12
AR247571A1 (es) 1995-01-31
DK119992D0 (da) 1992-09-28
HU194167B (en) 1988-01-28
CS409591A3 (en) 1992-04-15
EP0084164A3 (en) 1983-10-12
EP0084164A2 (de) 1983-07-27
IE823065L (en) 1983-06-29
PT76052A (de) 1983-01-01
JPH064586B2 (ja) 1994-01-19
NO156786C (no) 1987-11-25
GR78413B (fi) 1984-09-27
ES8402271A1 (es) 1984-01-16
US5101039A (en) 1992-03-31
NO824394L (no) 1983-06-30
DK171232B1 (da) 1996-08-05
ES518574A0 (es) 1983-10-01
PT76052B (de) 1985-11-28
NO156786B (no) 1987-08-17
IE55867B1 (en) 1991-02-14
US5008400A (en) 1991-04-16
NL930048I1 (nl) 1993-09-01
ES521740A0 (es) 1984-01-16
NZ202903A (en) 1988-01-08
MA19672A1 (fr) 1983-07-01
JPH0587504B2 (fi) 1993-12-16
AU9193182A (en) 1983-07-07
CA1341296C (en) 2001-09-25
DE3280014D1 (en) 1989-12-14
KR840002810A (ko) 1984-07-21
FI80017B (fi) 1989-12-29
SG1389G (en) 1989-06-02
JPH01301659A (ja) 1989-12-05
LU88263I2 (fi) 1994-02-03
NL930048I2 (nl) 1994-01-03
PH18918A (en) 1985-11-06
IL67572A0 (en) 1983-05-15
DK576782A (da) 1983-06-30
HK74989A (en) 1989-09-22
JPS58118569A (ja) 1983-07-14
DK119992A (da) 1992-09-28
IL67572A (en) 1992-08-18
DK170444B1 (da) 1995-09-04
DZ490A1 (fr) 2004-09-13
FI824474A0 (fi) 1982-12-27
ES8308850A1 (es) 1983-10-01
JPH01301695A (ja) 1989-12-05
FI80017C (fi) 1990-04-10
DE3275293D1 (en) 1987-03-05
EP0084164B1 (de) 1987-01-28
PH19771A (en) 1986-06-27

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