FI791562A - PROCEDURE FOR FRAMSTATION OF AV 4-AMINO-2-PIPERIDINOKINAZOLINE DERIVATIVES - Google Patents

PROCEDURE FOR FRAMSTATION OF AV 4-AMINO-2-PIPERIDINOKINAZOLINE DERIVATIVES

Info

Publication number: FI791562A
Authority: FI; Finland
Prior art keywords: piperidinokinazoline; framstation; derivatives; amino; procedure
Prior art date: 1978-05-18

Application number

FI791562A

Other languages

Finnish (fi)

Other versions

FI64589C (en

FI64589B (en

Inventor

Simon Fraser Campbell

John Christopher Danilewicz

Colin William Greengrass

Rhona Plews

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1978-05-18

Filing date

1979-05-16

Publication date

1979-11-19

1979-05-16 Application filed by Pfizer filed Critical Pfizer

1979-11-19 Publication of FI791562A publication Critical patent/FI791562A/en

1983-08-31 Application granted granted Critical

1983-08-31 Publication of FI64589B publication Critical patent/FI64589B/en

1983-12-12 Publication of FI64589C publication Critical patent/FI64589C/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/60—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D211/62—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals attached in position 4
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/40—Oxygen atoms
- C07D211/44—Oxygen atoms attached in position 4
- C07D211/46—Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/60—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Cardiology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Heart & Thoracic Surgery (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Hydrogenated Pyridines (AREA)
Pyridine Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

FI791562A 1978-05-18 1979-05-16 FRAMEWORK FOR THE PREPARATION OF THERAPEUTIC THERAPEUTIC 4-AMINO-2-PIPERIDINOQUINAZOLE DERIVATIVES FI64589C (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB2035178		1978-05-18
GB2035178		1978-05-18

Publications (3)

Publication Number	Publication Date
FI791562A true FI791562A (en)	1979-11-19
FI64589B FI64589B (en)	1983-08-31
FI64589C FI64589C (en)	1983-12-12

Family

ID=10144517

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
FI791562A FI64589C (en)	1978-05-18	1979-05-16	FRAMEWORK FOR THE PREPARATION OF THERAPEUTIC THERAPEUTIC 4-AMINO-2-PIPERIDINOQUINAZOLE DERIVATIVES

Country Status (30)

Country	Link
US (1)	US4243666A (en)
JP (1)	JPS554370A (en)
AR (2)	AR223487A1 (en)
AT (1)	ATA363379A (en)
AU (1)	AU512947B2 (en)
BE (1)	BE876297A (en)
CA (1)	CA1240325A (en)
CH (1)	CH643553A5 (en)
CS (1)	CS214796B2 (en)
DD (1)	DD143613A5 (en)
DE (1)	DE2919800A1 (en)
DK (1)	DK159079A (en)
ES (2)	ES480671A1 (en)
FI (1)	FI64589C (en)
FR (1)	FR2434162A1 (en)
GR (1)	GR72824B (en)
HU (1)	HU182562B (en)
IL (1)	IL57297A (en)
IN (1)	IN153045B (en)
IT (1)	IT1114222B (en)
LU (1)	LU81284A1 (en)
NL (1)	NL172157C (en)
NO (1)	NO791648L (en)
NZ (1)	NZ190465A (en)
PH (1)	PH14802A (en)
PL (2)	PL121158B1 (en)
PT (1)	PT69622A (en)
SE (1)	SE439306B (en)
YU (2)	YU115279A (en)
ZA (1)	ZA792390B (en)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4607034A (en) *	1979-10-29	1986-08-19	Mitsubishi Yuka Pharmaceutical Co., Ltd.	Quinazoline derivatives and pharmaceutical composition thereof
JPS5962766U (en) *	1982-06-30	1984-04-25	守田　智	Water dispenser for small animals
GB8414518D0 (en) *	1984-06-07	1984-07-11	Pfizer Ltd	Therapeutic agents
US5801195A (en) *	1994-12-30	1998-09-01	Celgene Corporation	Immunotherapeutic aryl amides
US6248888B1 (en)	1997-11-14	2001-06-19	Teva Pharmaceutical Industries Ltd.	Process for the preparation of terazosin hydrochloride dihydrate
CN1494529A (en) *	2001-01-18	2004-05-05	武田药品工业株式会社	The preparation method of benzyl piperidine compound
US6746460B2 (en) *	2002-08-07	2004-06-08	Satiety, Inc.	Intra-gastric fastening devices
EP1685115A1 (en) *	2003-11-03	2006-08-02	Warner-Lambert Company LLC	Novel norepinephrine reuptake inhibitors for the treatment of central nervous system disorders
CL2007002958A1 (en) *	2006-10-12	2008-05-09	Epix Delaware Inc	COMPOUNDS DERIVED FROM HETEROARIL-CARBOXAMIDA, ANTAGONISTS OF THE CHEMIOQUINE RECEPTOR; PHARMACEUTICAL COMPOSITION; AND USE FOR THE TREATMENT OR PREVENTION OF SUCH DISEASES AS REJECTION OF ORGAN TRANSPLANTS, Rheumatoid Arthritis, LUPUS, ENTR
EP2139868B1 (en) *	2007-04-04	2015-07-29	Cipla Limited	Process for preparation of erlotinib and its pharmaceutically acceptable salts
AU2008335135A1 (en) *	2007-12-11	2009-06-18	Cytopathfinder, Inc.	Carboxamide compounds and their use as chemokine receptor agonists
ES2404076T3 (en) *	2008-11-14	2013-05-23	F. Hoffmann-La Roche Ag	Quinazoline derivatives as NK3 receptor antagonists

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1156973A (en) *	1965-07-06	1969-07-02		Quinazoline Derivatives
US3511836A (en) *	1967-12-13	1970-05-12	Pfizer & Co C	2,4,6,7-tetra substituted quinazolines
FR2321890A1 (en) *	1975-08-26	1977-03-25	Synthelabo	Hypotensive amino-quinazoline derivs. - with substd. piperidine or piperazine substit.
DK140695C (en) *	1976-05-07	1980-05-12	Synthelabo	ANALOGY PROCEDURE FOR PREPARING 2,4-DIAMINO-6,7-DIMETHOXYQUINAZOLINE DERIVATIVES OR ACID ADDITION SALTS

1979
- 1979-04-18 DK DK159079A patent/DK159079A/en not_active IP Right Cessation
- 1979-05-14 US US06/038,509 patent/US4243666A/en not_active Expired - Lifetime
- 1979-05-16 BE BE0/195197A patent/BE876297A/en unknown
- 1979-05-16 IL IL57297A patent/IL57297A/en unknown
- 1979-05-16 NO NO791648A patent/NO791648L/en unknown
- 1979-05-16 PL PL1979223844A patent/PL121158B1/en unknown
- 1979-05-16 GR GR59104A patent/GR72824B/el unknown
- 1979-05-16 YU YU01152/79A patent/YU115279A/en unknown
- 1979-05-16 PH PH22500A patent/PH14802A/en unknown
- 1979-05-16 NL NLAANVRAGE7903853,A patent/NL172157C/en not_active IP Right Cessation
- 1979-05-16 DE DE19792919800 patent/DE2919800A1/en not_active Ceased
- 1979-05-16 NZ NZ190465A patent/NZ190465A/en unknown
- 1979-05-16 IT IT22720/79A patent/IT1114222B/en active
- 1979-05-16 CS CS793372A patent/CS214796B2/en unknown
- 1979-05-16 AT AT0363379A patent/ATA363379A/en not_active IP Right Cessation
- 1979-05-16 FI FI791562A patent/FI64589C/en not_active IP Right Cessation
- 1979-05-16 AR AR276536A patent/AR223487A1/en active
- 1979-05-16 AU AU47101/79A patent/AU512947B2/en not_active Ceased
- 1979-05-16 IN IN337/DEL/79A patent/IN153045B/en unknown
- 1979-05-16 PL PL1979215626A patent/PL120651B1/en unknown
- 1979-05-17 HU HU79PI678A patent/HU182562B/en unknown
- 1979-05-17 CA CA000327839A patent/CA1240325A/en not_active Expired
- 1979-05-17 FR FR7912635A patent/FR2434162A1/en active Granted
- 1979-05-17 SE SE7904358A patent/SE439306B/en not_active IP Right Cessation
- 1979-05-17 JP JP6100079A patent/JPS554370A/en active Granted
- 1979-05-17 PT PT69622A patent/PT69622A/en unknown
- 1979-05-17 LU LU81284A patent/LU81284A1/en unknown
- 1979-05-17 ES ES480671A patent/ES480671A1/en not_active Expired
- 1979-05-17 CH CH459879A patent/CH643553A5/en not_active IP Right Cessation
- 1979-05-17 ZA ZA792390A patent/ZA792390B/en unknown
- 1979-05-18 DD DD79213010A patent/DD143613A5/en unknown
1980
- 1980-02-01 ES ES488210A patent/ES8101584A1/en not_active Expired
- 1980-10-28 AR AR283021A patent/AR224784A1/en active
1982
- 1982-11-16 YU YU02563/82A patent/YU256382A/en unknown

Also Published As

Publication number	Publication date
IN153045B (en)	1984-05-26
NL172157B (en)	1983-02-16
ES480671A1 (en)	1980-08-16
AR223487A1 (en)	1981-08-31
FR2434162B1 (en)	1983-04-22
DK159079A (en)	1979-11-19
BE876297A (en)	1979-11-16
PL223844A1 (en)	1981-01-02
DE2919800A1 (en)	1979-11-22
IT7922720A0 (en)	1979-05-16
GR72824B (en)	1983-12-06
HU182562B (en)	1984-02-28
PL121158B1 (en)	1982-04-30
ZA792390B (en)	1980-07-30
NL7903853A (en)	1979-11-20
ATA363379A (en)	1983-05-15
JPS5623992B2 (en)	1981-06-03
US4243666A (en)	1981-01-06
FR2434162A1 (en)	1980-03-21
IL57297A (en)	1983-02-23
NL172157C (en)	1983-07-18
FI64589C (en)	1983-12-12
CH643553A5 (en)	1984-06-15
LU81284A1 (en)	1980-12-16
ES488210A0 (en)	1980-12-16
AU512947B2 (en)	1980-11-06
CS214796B2 (en)	1982-05-28
YU115279A (en)	1983-04-30
AU4710179A (en)	1979-11-22
DD143613A5 (en)	1980-09-03
PL215626A1 (en)	1980-08-25
SE439306B (en)	1985-06-10
PH14802A (en)	1981-12-14
FI64589B (en)	1983-08-31
JPS554370A (en)	1980-01-12
ES8101584A1 (en)	1980-12-16
PT69622A (en)	1979-06-01
NZ190465A (en)	1981-05-01
IL57297A0 (en)	1979-09-30
YU256382A (en)	1983-04-30
CA1240325A (en)	1988-08-09
PL120651B1 (en)	1982-03-31
IT1114222B (en)	1986-01-27
SE7904358L (en)	1979-11-19
AR224784A1 (en)	1982-01-15
NO791648L (en)	1979-11-20

Publication	Publication Date	Title
NO790358L (en)	1979-08-07	PROCEDURE FOR THE PREPARATION OF ALKYLENDIAMIN DERIVATIVES
FI800008A (en)	1980-07-05	FRAMEWORK FOR FRAMSTATION OF PEPTIDYLARGININALDEHYD DERIVATIVES
FI792824A (en)	1980-03-30	FRAMEWORK FOR OILIZATION OF OXIDERING INHIBITION
ES494635A0 (en)	1981-08-16	PROCEDURE FOR THE PREPARATION OF TIADIAZOLE DERIVATIVES
NO791831L (en)	1979-12-04	PROCEDURE FOR THE PREPARATION OF AMINOTIAZOLES
NO792404L (en)	1980-01-29	PROCEDURE FOR THE PREPARATION OF IMIDAZOLD DERIVATIVES
NO151201C (en)	1985-02-27	PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY EFFECTIVE ANTIGENDATIVE DERIVATIVES
NO150155C (en)	1984-08-29	PROCEDURE FOR THE PREPARATION OF 2-PYRROLIDON COMPOUNDS
NO151895C (en)	1985-06-26	PROCEDURE FOR THE PREPARATION OF PYRIDO-INDOLD DERIVATIVES
NO791139L (en)	1979-10-08	PROCEDURE FOR THE PREPARATION OF LYSERGOLD DERIVATIVES
FI791562A (en)	1979-11-19	PROCEDURE FOR FRAMSTATION OF AV 4-AMINO-2-PIPERIDINOKINAZOLINE DERIVATIVES
SE7902238L (en)	1979-09-21	PROCEDURE FOR DETERMINATION OF ALFA-AMYLAS
NO791604L (en)	1979-11-16	PROCEDURE FOR PREPARING DI-O-N-ALKYL-GLYCEROL DERIVATIVES
SE7803035L (en)	1978-09-30	PROCEDURE FOR THE PREPARATION OF TIENOPYRIDINE DERIVATIVES
NO784382L (en)	1979-07-02	PROCEDURE FOR THE PREPARATION OF TIAZOLDIN DERIVATIVES
SE7707407L (en)	1977-12-29	PROCEDURE FOR PREPARATION OF CEFAM DERIVATIVES
FI793307A (en)	1980-04-28	PROCEDURE FOR FRAMSTATION OF 6-PIPERIDINO-2,4-DIAMINOPYRIMIDIN-3-OXIDE
FI793221A (en)	1980-04-20	FRAMEWORK FOR FRAMEWORK OF SUBSTITUTIONS
NO793164L (en)	1980-04-09	PROCEDURE FOR THE PREPARATION OF SODIUM AMOXYCILLAN
NO152254C (en)	1985-08-28	PROCEDURE FOR THE PREPARATION OF CARBZOLD DERIVATIVES
NO147310C (en)	1983-03-16	PROCEDURE FOR THE PREPARATION OF SUBSTITUTED ANTITUMORANTRACYCLINES
NO791599L (en)	1979-11-20	PROCEDURE FOR THE MANUFACTURE OF DIBENZYLETERS
NO794090L (en)	1980-06-19	PROCEDURE FOR THE PREPARATION OF CHLORODIOXIDE
NO780389L (en)	1978-08-07	PROCEDURE FOR THE PREPARATION OF ERYTROMYCIN DERIVATIVES
NO790972L (en)	1979-09-25	PROCEDURE FOR ISOMERIZATION OF DERIVATIVES OF 3-VINYL-PIPERIDINE

Legal Events

Date	Code	Title	Description
2004-08-31	MM	Patent lapsed	Owner name: PFIZER CORPORATION