FI55334B - Foerfarande foer framstaellning av som mellanprodukter vid framstaellning av triazolobensodiazepiner anvaenda 2-alkoxi-5-fenyl-3h-1,4-bensodiazepinderivat - Google Patents
Foerfarande foer framstaellning av som mellanprodukter vid framstaellning av triazolobensodiazepiner anvaenda 2-alkoxi-5-fenyl-3h-1,4-bensodiazepinderivatInfo
- Publication number
- FI55334B FI55334B FI896/71A FI89671A FI55334B FI 55334 B FI55334 B FI 55334B FI 896/71 A FI896/71 A FI 896/71A FI 89671 A FI89671 A FI 89671A FI 55334 B FI55334 B FI 55334B
- Authority
- FI
- Finland
- Prior art keywords
- triazolobensodiazepiner
- benzodiazepinderivat
- anvaenda
- framstation
- alcoxy
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
- C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
- C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
- C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
- C07D243/20—Nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FI752812A FI57938C (fi) | 1970-03-27 | 1975-10-09 | Foerfarande foer framstaellning av 2-hydrazino-5-fenyl-3h-1;4-benzodiazepinderivat |
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2580570A JPS5010316B1 (fi) | 1970-03-27 | 1970-03-27 | |
JP2580470A JPS4811112B1 (fi) | 1970-03-27 | 1970-03-27 | |
JP3495070A JPS5011920B1 (fi) | 1970-04-23 | 1970-04-23 | |
JP4663770A JPS4924060B1 (fi) | 1970-05-28 | 1970-05-28 |
Publications (2)
Publication Number | Publication Date |
---|---|
FI55334B true FI55334B (fi) | 1979-03-30 |
FI55334C FI55334C (fi) | 1979-07-10 |
Family
ID=27458380
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI896/71A FI55334C (fi) | 1970-03-27 | 1971-03-29 | Foerfarande foer framstaellning av som mellanprodukter vid framstaellning av triazolobensodiazepiner anvaenda 2-alkoxi-5-fenyl-3h-1,4-bensodiazepinderivat |
Country Status (14)
Country | Link |
---|---|
US (1) | US4102881A (fi) |
BE (1) | BE764913A (fi) |
CA (2) | CA922317A (fi) |
CH (1) | CH559188A5 (fi) |
DE (1) | DE2114441A1 (fi) |
DK (1) | DK131374B (fi) |
FI (1) | FI55334C (fi) |
FR (1) | FR2085748B1 (fi) |
GB (1) | GB1353486A (fi) |
NL (1) | NL7104132A (fi) |
NO (1) | NO132800C (fi) |
PH (1) | PH9214A (fi) |
SE (1) | SE400968B (fi) |
YU (1) | YU34997B (fi) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3709898A (en) * | 1971-02-09 | 1973-01-09 | Upjohn Co | Process for the production of triazolobenzodiazepines and intermediates |
US3681343A (en) * | 1971-05-11 | 1972-08-01 | Upjohn Co | 6-phenyl-s-triazolo{8 4,3-a{9 {8 1,4{9 {0 benzodiazepines |
US4755508A (en) * | 1984-06-26 | 1988-07-05 | Merck & Co., Inc. | Benzodiazepine analogs and use as antogonists of gastrin and cholecystokinin |
US5939414A (en) * | 1996-10-31 | 1999-08-17 | Merck & Co., Inc. | Benzodiazepine hydrazide derivatives as inhibitors of HIV integrase |
AU4917397A (en) * | 1996-10-31 | 1998-05-22 | Merck & Co., Inc. | Benzodiazepine hydrazide derivatives as inhibitors of hiv integrase |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3462418A (en) * | 1963-10-29 | 1969-08-19 | Hoffmann La Roche | Preparation of 1,4-benzodiazepin-2-one-4-oxide from 2-lower alkoxy-1,4-benzodiazepine-4-oxide |
DK120901B (da) * | 1965-09-17 | 1971-08-02 | Rexolin Chem | Fremgangsmåde til fremstilling af 7-chlor-1,3-dihydro-1-methyl-5-phenyl-2H-1,4-benzodiazepin-2-on. |
US3987052A (en) * | 1969-03-17 | 1976-10-19 | The Upjohn Company | 6-Phenyl-4H-s-triazolo[4,3-a][1,4]benzodiazepines |
NO128154B (fi) * | 1969-07-30 | 1973-10-08 | Grindstedvaerket As | |
BE755139A (fr) * | 1969-08-21 | 1971-02-22 | Upjohn Co | Derives de benzodiazepinones, leurs intermediaires, et leur preparatio |
FR2022598A1 (en) * | 1969-11-04 | 1970-07-31 | Pakeda Chemical Ind | Sedative chloro-phenyl-triazolobenzodiazepines |
-
1971
- 1971-03-24 YU YU737/71A patent/YU34997B/xx unknown
- 1971-03-25 FR FR7110689A patent/FR2085748B1/fr not_active Expired
- 1971-03-25 CH CH437571A patent/CH559188A5/xx not_active IP Right Cessation
- 1971-03-25 DE DE19712114441 patent/DE2114441A1/de not_active Withdrawn
- 1971-03-26 PH PH12320*UA patent/PH9214A/en unknown
- 1971-03-26 BE BE764913A patent/BE764913A/xx unknown
- 1971-03-26 NO NO1151/71A patent/NO132800C/no unknown
- 1971-03-26 NL NL7104132A patent/NL7104132A/xx unknown
- 1971-03-26 SE SE7103998A patent/SE400968B/xx unknown
- 1971-03-26 CA CA108803A patent/CA922317A/en not_active Expired
- 1971-03-26 DK DK147671AA patent/DK131374B/da unknown
- 1971-03-29 FI FI896/71A patent/FI55334C/fi active
- 1971-04-19 GB GB2562271*A patent/GB1353486A/en not_active Expired
-
1972
- 1972-11-16 CA CA156599A patent/CA936864A/en not_active Expired
-
1974
- 1974-06-12 US US05/478,823 patent/US4102881A/en not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
FR2085748B1 (fi) | 1974-08-02 |
BE764913A (fr) | 1971-08-16 |
NO132800C (fi) | 1976-01-07 |
FI55334C (fi) | 1979-07-10 |
SE400968B (sv) | 1978-04-17 |
NL7104132A (fi) | 1971-09-29 |
DE2114441A1 (de) | 1971-10-14 |
DK131374B (da) | 1975-07-07 |
CH559188A5 (fi) | 1975-02-28 |
CA936864A (en) | 1973-11-13 |
YU34997B (en) | 1980-06-30 |
GB1353486A (en) | 1974-05-15 |
US4102881A (en) | 1978-07-25 |
NO132800B (fi) | 1975-09-29 |
FR2085748A1 (fi) | 1971-12-31 |
CA922317A (en) | 1973-03-06 |
YU73771A (en) | 1979-12-31 |
PH9214A (en) | 1975-07-10 |
DK131374C (fi) | 1975-12-01 |
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