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ES8105148A1 - Un procedimiento para la preparacion de una composicion far-maceutica de quinazolinonas analgesicas - Google Patents

Un procedimiento para la preparacion de una composicion far-maceutica de quinazolinonas analgesicas

Info

Publication number
ES8105148A1
ES8105148A1 ES490453A ES490453A ES8105148A1 ES 8105148 A1 ES8105148 A1 ES 8105148A1 ES 490453 A ES490453 A ES 490453A ES 490453 A ES490453 A ES 490453A ES 8105148 A1 ES8105148 A1 ES 8105148A1
Authority
ES
Spain
Prior art keywords
formulation
active agents
myotonolytic
analgesic
preparations
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES490453A
Other languages
English (en)
Other versions
ES490453A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sandoz AG
Original Assignee
Sandoz AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from CH341179A external-priority patent/CH640415A5/de
Application filed by Sandoz AG filed Critical Sandoz AG
Publication of ES490453A0 publication Critical patent/ES490453A0/es
Publication of ES8105148A1 publication Critical patent/ES8105148A1/es
Expired legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

PROCEDIMIENTO DE OBTENCION DE DERIVADOS DE QUINAZOLINONAS. CONSTA DE LAS SIGUIENTES ETAPAS: 1. PREPARACION DE UNA FORMULACION INICIAL COMBINANDO SINERGISTICAMENTE UNA QUINAZOLINONA ANALGESICAMENTE ACTIVA CON UN MIOTONOLITICO EN UN MEDIO DE VEHICULO SOLIDO O LIQUIDO FARMACEUTICAMENTE ACEPTABLE MEDIANTE LA TECNICA DE FORMULACION GALENICA. 2. OPCIONALMENTE SE OBTIENE LA FORMULACION ANTERIOR EN FORMA DE DOSIS. LOS AGENTES ACTIVOS SE ASOCIAN EN UNA PROPORCION DE APROXIMADAMENTE 20:1 A 50:1 PARTES POR PESO. LOS AGENTES ACTIVOS SON EL 1-ISOPROPIL-4-(4-FLUORFENIL)-7-METIL-2-(1H) QUIAZOLINONA Y EL 5-CLORO-4-(2-IMIDAZOLIN-2-IL-AMINO)-2,1,3-BENGOTIADIAZOL. A
ES490453A 1979-04-10 1980-04-10 Un procedimiento para la preparacion de una composicion far-maceutica de quinazolinonas analgesicas Expired ES8105148A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH340979 1979-04-10
CH341179A CH640415A5 (en) 1979-04-10 1979-04-10 Therapeutic preparations for the treatment of pain

Publications (2)

Publication Number Publication Date
ES490453A0 ES490453A0 (es) 1981-05-16
ES8105148A1 true ES8105148A1 (es) 1981-05-16

Family

ID=25692937

Family Applications (1)

Application Number Title Priority Date Filing Date
ES490453A Expired ES8105148A1 (es) 1979-04-10 1980-04-10 Un procedimiento para la preparacion de una composicion far-maceutica de quinazolinonas analgesicas

Country Status (18)

Country Link
US (1) US4442084A (es)
AR (1) AR228255A1 (es)
AU (1) AU538643B2 (es)
CA (1) CA1147261A (es)
DE (1) DE3012837A1 (es)
ES (1) ES8105148A1 (es)
FR (1) FR2453648A1 (es)
GB (1) GB2047534B (es)
HU (1) HU183119B (es)
IE (1) IE49676B1 (es)
IL (1) IL59786A (es)
IT (1) IT1143133B (es)
MY (1) MY8500127A (es)
NL (1) NL8002041A (es)
NZ (1) NZ193379A (es)
PH (1) PH17681A (es)
PT (1) PT71066A (es)
SE (1) SE445708B (es)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2499991A1 (fr) * 1981-02-19 1982-08-20 Sandoz Sa Nouveaux 2,1,3-benzothiadiazoles et 2,1,3-benzoxadiazoles, leur preparation et leur application comme medicaments
GB8306473D0 (en) * 1983-03-09 1983-04-13 Sandoz Ltd Analgesic preparations
GB2135884B (en) * 1983-03-09 1986-09-17 Sandoz Ltd Analgesic preparations containing tizanidine and paracetamol
JPS608274A (ja) * 1983-06-27 1985-01-17 Fujisawa Pharmaceut Co Ltd 新規キナゾリノン誘導体およびその製造法・並びに抗アレルギ−剤
NL8702523A (nl) * 1986-11-03 1988-06-01 Sandoz Ag Farmaceutische preparaten met analgetische werking en werkwijze voor het bereiden of vervaardigen en toepassen van deze preparaten.
DE3738844A1 (de) * 1987-11-16 1989-05-24 Merck Patent Gmbh Analgetikum
US5039999A (en) * 1990-06-26 1991-08-13 Hewlett-Packard Company Accumulator and pressure control for ink-ket pens
DE10146275A1 (de) 2001-09-18 2003-04-24 Gruenenthal Gmbh Kombination ausgewählter Opioide mit Muscarin-Antagonisten zur Therapie der Harninkontinenz
US7799832B2 (en) * 2003-10-23 2010-09-21 Valeant Pharmaceuticals North America Combinations of retigabine and sodium channel inhibitors or sodium channel-influencing active compounds for treating pains

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BG16442A3 (bg) * 1967-10-30 1972-11-20 Max Denzer Метод за получаване на нови о-изопропиламинобензофенони
CH569722A5 (es) * 1971-06-24 1975-11-28 Sandoz Ag
US3759920A (en) * 1971-06-24 1973-09-18 Sandoz Ag Process for the preparation of 1-substituted-phenyl-2(1h)-quinazolinones
BE801898A (en) * 1973-07-04 1974-01-04 Merck Patent Gmbh Insomnia treatment - with synergistic mixt of carisoprodol and methaqualone

Also Published As

Publication number Publication date
MY8500127A (en) 1985-12-31
IE800724L (en) 1980-10-10
GB2047534B (en) 1983-04-20
IE49676B1 (en) 1985-11-27
PH17681A (en) 1984-11-02
CA1147261A (en) 1983-05-31
ES490453A0 (es) 1981-05-16
NZ193379A (en) 1984-07-31
SE445708B (sv) 1986-07-14
AR228255A1 (es) 1983-02-15
PT71066A (en) 1980-05-01
AU5722380A (en) 1980-10-16
FR2453648B1 (es) 1983-06-24
IT8048364A0 (it) 1980-04-08
IT1143133B (it) 1986-10-22
IL59786A0 (en) 1980-06-30
US4442084A (en) 1984-04-10
HU183119B (en) 1984-04-28
AU538643B2 (en) 1984-08-23
GB2047534A (en) 1980-12-03
IL59786A (en) 1984-02-29
NL8002041A (nl) 1980-10-14
DE3012837A1 (de) 1980-10-30
FR2453648A1 (fr) 1980-11-07
SE8002642L (sv) 1980-10-11

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