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ES534186A0 - Un procedimiento para la preparacion de derivados peptidicos - Google Patents

Un procedimiento para la preparacion de derivados peptidicos

Info

Publication number
ES534186A0
ES534186A0 ES534186A ES534186A ES534186A0 ES 534186 A0 ES534186 A0 ES 534186A0 ES 534186 A ES534186 A ES 534186A ES 534186 A ES534186 A ES 534186A ES 534186 A0 ES534186 A0 ES 534186A0
Authority
ES
Spain
Prior art keywords
procedure
preparation
peptidic derivatives
peptidic
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES534186A
Other languages
English (en)
Other versions
ES8601236A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB838318855A external-priority patent/GB8318855D0/en
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Publication of ES8601236A1 publication Critical patent/ES8601236A1/es
Publication of ES534186A0 publication Critical patent/ES534186A0/es
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06086Dipeptides with the first amino acid being basic
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/0215Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing natural amino acids, forming a peptide bond via their side chain functional group, e.g. epsilon-Lys, gamma-Glu
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08Tripeptides
    • C07K5/0815Tripeptides with the first amino acid being basic
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ES534186A 1983-07-12 1984-07-11 Un procedimiento para la preparacion de derivados peptidicos Granted ES534186A0 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB838318855A GB8318855D0 (en) 1983-07-12 1983-07-12 Peptide derivatives
GB848411635A GB8411635D0 (en) 1983-07-12 1984-05-08 Peptide derivatives

Publications (2)

Publication Number Publication Date
ES8601236A1 ES8601236A1 (es) 1985-11-01
ES534186A0 true ES534186A0 (es) 1985-11-01

Family

ID=26286589

Family Applications (1)

Application Number Title Priority Date Filing Date
ES534186A Granted ES534186A0 (es) 1983-07-12 1984-07-11 Un procedimiento para la preparacion de derivados peptidicos

Country Status (11)

Country Link
US (1) US4623639A (es)
EP (1) EP0133225B1 (es)
AU (1) AU578898B2 (es)
CA (1) CA1267499A (es)
DE (1) DE3474670D1 (es)
DK (1) DK304684A (es)
ES (1) ES534186A0 (es)
IE (1) IE57747B1 (es)
IL (1) IL72345A (es)
NZ (1) NZ208796A (es)
PH (1) PH23381A (es)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3481913D1 (de) * 1983-04-27 1990-05-17 Ici America Inc Prolin-derivate.
DD248961A1 (de) * 1984-05-22 1987-08-26 Akad Wissenschaften Ddr Verfahren zur herstellung wundheilungsfoerdernder praeparationen
HU192646B (en) * 1984-12-21 1987-06-29 Gyogyszerkutato Intezet Process for preparing new n-alkyl-peptide aldehydes
GB8613704D0 (en) * 1986-06-05 1986-07-09 Ici America Inc Difluoro keto compounds
US5736520A (en) * 1988-10-07 1998-04-07 Merrell Pharmaceuticals Inc. Peptidase inhibitors
ZA897514B (en) * 1988-10-07 1990-06-27 Merrell Dow Pharma Novel peptidase inhibitors
WO1990012805A1 (en) * 1989-04-15 1990-11-01 Zaidan Hojin Biseibutsu Kagaku Kenkyu Kai Postostatin and related compound thereof, or their salts
DK53291D0 (da) * 1991-03-25 1991-03-25 Carlbiotech Ltd As Smaa peptider og peptidrelaterede stoffer samt farmaceutiske praeparater indeholdende saadanne forbindelser
US5714470A (en) * 1991-08-22 1998-02-03 Merrell Pharmaceuticals, Inc. Orally-active elastase inhibitors
US5478811A (en) * 1991-08-22 1995-12-26 Merrell Dow Pharmaceuticals Inc. Orally-active elastase inhibitors
IL108031A0 (en) * 1992-12-22 1994-04-12 Procter & Gamble Difluoro pentapeptide derivatives and pharmaceutical compositions containing them
AU696292B2 (en) * 1994-06-02 1998-09-03 Merrell Pharmaceuticals Inc. Acylated enol derivatives as prodrugs of elastase inhibitors
DE69513167T2 (de) * 1994-06-02 2000-06-15 Merrell Pharmaceuticals Inc., Cincinnati Perfluoroalkyll ketone, inhibitoren von elastase und prozess zur deren herstellung
US6172044B1 (en) 1995-12-01 2001-01-09 Aventis Pharmaceuticals Inc. Acylated enol derivative of α-ketoesters and α-ketoamides
US5948886A (en) * 1996-11-20 1999-09-07 Hoechst Marion Roussel, Inc. Acylated enol derivatives of α-ketoesters and α-ketoamides
JP2022538360A (ja) * 2019-07-01 2022-09-01 ビーエーエスエフ ソシエタス・ヨーロピア 酵素を安定化するためのペプチドアセタール

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3481913D1 (de) * 1983-04-27 1990-05-17 Ici America Inc Prolin-derivate.

Also Published As

Publication number Publication date
IE57747B1 (en) 1993-03-24
PH23381A (en) 1989-07-26
ES8601236A1 (es) 1985-11-01
CA1267499A (en) 1990-04-03
EP0133225A2 (de) 1985-02-20
US4623639A (en) 1986-11-18
IL72345A (en) 1988-05-31
EP0133225B1 (de) 1988-10-19
NZ208796A (en) 1989-01-27
DK304684D0 (da) 1984-06-21
IL72345A0 (en) 1984-11-30
AU578898B2 (en) 1988-11-10
AU3039384A (en) 1985-01-17
IE841782L (en) 1985-01-12
DE3474670D1 (en) 1988-11-24
DK304684A (da) 1985-01-13
EP0133225A3 (en) 1985-10-02

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19970303