ES424717A1 - Procedimiento para preparar carboxamidas y tiocarboxamidas. - Google Patents

Procedimiento para preparar carboxamidas y tiocarboxamidas.

Info

Publication number: ES424717A1
Authority: ES; Spain
Prior art keywords: lower alkyl; compound; hydrogen; group; compound obtained
Prior art date: 1973-03-29
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired

Application number

ES424717A

Other languages

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

STWB Inc

Original Assignee

Sterling Drug Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1973-03-29

Filing date

1974-03-28

Publication date

1976-11-01

1973-03-29 Priority claimed from US346005A external-priority patent/US3928380A/en

1974-03-28 Application filed by Sterling Drug Inc filed Critical Sterling Drug Inc

1976-11-01 Publication of ES424717A1 publication Critical patent/ES424717A1/es

Status Expired legal-status Critical Current

Links

150000003857 carboxamides Chemical class 0.000 title abstract 2
238000000034 method Methods 0.000 title abstract 2
125000000217 alkyl group Chemical group 0.000 abstract 27
150000001875 compounds Chemical class 0.000 abstract 24
-1 4- (2, 1, 3-benzothiadiazolyl) -2-benzothiazolyl Chemical group 0.000 abstract 14
229910052739 hydrogen Inorganic materials 0.000 abstract 11
239000001257 hydrogen Substances 0.000 abstract 11
125000002485 formyl group Chemical group [H]C(*)=O 0.000 abstract 7
150000002431 hydrogen Chemical group 0.000 abstract 7
125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 6
125000003545 alkoxy group Chemical group 0.000 abstract 5
239000002253 acid Substances 0.000 abstract 3
125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 3
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 3
125000004029 hydroxymethyl group Chemical group [H]OC([H])([H])* 0.000 abstract 3
UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 2
KAESVJOAVNADME-UHFFFAOYSA-N Pyrrole Chemical compound C=1C=CNC=1 KAESVJOAVNADME-UHFFFAOYSA-N 0.000 abstract 2
150000001447 alkali salts Chemical class 0.000 abstract 2
125000003342 alkenyl group Chemical group 0.000 abstract 2
125000004414 alkyl thio group Chemical group 0.000 abstract 2
239000002168 alkylating agent Substances 0.000 abstract 2
229940100198 alkylating agent Drugs 0.000 abstract 2
239000002585 base Substances 0.000 abstract 2
230000007062 hydrolysis Effects 0.000 abstract 2
238000006460 hydrolysis reaction Methods 0.000 abstract 2
125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
150000003839 salts Chemical class 0.000 abstract 2
125000004530 1,2,4-triazinyl group Chemical group N1=NC(=NC=C1)* 0.000 abstract 1
125000004105 2-pyridyl group Chemical group N1=C([*])C([H])=C([H])C([H])=C1[H] 0.000 abstract 1
125000003349 3-pyridyl group Chemical group N1=C([H])C([*])=C([H])C([H])=C1[H] 0.000 abstract 1
VHUUQVKOLVNVRT-UHFFFAOYSA-N Ammonium hydroxide Chemical compound [NH4+].[OH-] VHUUQVKOLVNVRT-UHFFFAOYSA-N 0.000 abstract 1
BXDZOYLPNAIDOC-UHFFFAOYSA-N N-[5-[(5-tert-butyl-1,3-oxazol-2-yl)methylsulfanyl]-1,3-thiazol-2-yl]-1-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethylamino]-2-oxoethyl]piperidine-4-carboxamide Chemical compound CC(C)(C)c1cnc(CSc2cnc(NC(=O)C3CCN(CC(=O)NCCOCCOCCOCCNc4cccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c45)CC3)s2)o1 BXDZOYLPNAIDOC-UHFFFAOYSA-N 0.000 abstract 1
238000005644 Wolff-Kishner reduction reaction Methods 0.000 abstract 1
125000000641 acridinyl group Chemical group C1(=CC=CC2=NC3=CC=CC=C3C=C12)* 0.000 abstract 1
229910052783 alkali metal Inorganic materials 0.000 abstract 1
150000001340 alkali metals Chemical class 0.000 abstract 1
125000005236 alkanoylamino group Chemical group 0.000 abstract 1
125000004849 alkoxymethyl group Chemical group 0.000 abstract 1
125000004644 alkyl sulfinyl group Chemical group 0.000 abstract 1
125000004390 alkyl sulfonyl group Chemical group 0.000 abstract 1
125000002947 alkylene group Chemical group 0.000 abstract 1
125000000304 alkynyl group Chemical group 0.000 abstract 1
239000000908 ammonium hydroxide Substances 0.000 abstract 1
150000003863 ammonium salts Chemical class 0.000 abstract 1
QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 1
125000004432 carbon atom Chemical group C* 0.000 abstract 1
125000005518 carboxamido group Chemical group 0.000 abstract 1
230000003197 catalytic effect Effects 0.000 abstract 1
238000006243 chemical reaction Methods 0.000 abstract 1
125000004966 cyanoalkyl group Chemical group 0.000 abstract 1
125000000753 cycloalkyl group Chemical group 0.000 abstract 1
150000002148 esters Chemical class 0.000 abstract 1
229910052736 halogen Inorganic materials 0.000 abstract 1
150000002367 halogens Chemical class 0.000 abstract 1
230000003301 hydrolyzing effect Effects 0.000 abstract 1
RAXXELZNTBOGNW-UHFFFAOYSA-N imidazole Natural products C1=CNC=N1 RAXXELZNTBOGNW-UHFFFAOYSA-N 0.000 abstract 1
125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 1
229910052760 oxygen Inorganic materials 0.000 abstract 1
239000001301 oxygen Substances 0.000 abstract 1
125000003884 phenylalkyl group Chemical group 0.000 abstract 1
CYQAYERJWZKYML-UHFFFAOYSA-N phosphorus pentasulfide Chemical compound S1P(S2)(=S)SP3(=S)SP1(=S)SP2(=S)S3 CYQAYERJWZKYML-UHFFFAOYSA-N 0.000 abstract 1
125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1
125000004307 pyrazin-2-yl group Chemical group [H]C1=C([H])N=C(*)C([H])=N1 0.000 abstract 1
125000002206 pyridazin-3-yl group Chemical group [H]C1=C([H])C([H])=C(*)N=N1 0.000 abstract 1
125000000246 pyrimidin-2-yl group Chemical group [H]C1=NC(*)=NC([H])=C1[H] 0.000 abstract 1
125000004527 pyrimidin-4-yl group Chemical group N1=CN=C(C=C1)* 0.000 abstract 1
125000004943 pyrimidin-6-yl group Chemical group N1=CN=CC=C1* 0.000 abstract 1
150000003242 quaternary ammonium salts Chemical class 0.000 abstract 1
LMBFAGIMSUYTBN-MPZNNTNKSA-N teixobactin Chemical compound C([C@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](CCC(N)=O)C(=O)N[C@H]([C@@H](C)CC)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H]1C(N[C@@H](C)C(=O)N[C@@H](C[C@@H]2NC(=N)NC2)C(=O)N[C@H](C(=O)O[C@H]1C)[C@@H](C)CC)=O)NC)C1=CC=CC=C1 LMBFAGIMSUYTBN-MPZNNTNKSA-N 0.000 abstract 1
125000001544 thienyl group Chemical group 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Pyrrole Compounds (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

ES424717A 1973-03-29 1974-03-28 Procedimiento para preparar carboxamidas y tiocarboxamidas. Expired ES424717A1 (es)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US346005A US3928380A (en)	1973-03-29	1973-03-29	1,1{40 -Spirobis(cyclopenta-{8 4,5-c{9 pyrroles)

Publications (1)

Publication Number	Publication Date
ES424717A1 true ES424717A1 (es)	1976-11-01

Family

ID=23357526

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
ES424717A Expired ES424717A1 (es)	1973-03-29	1974-03-28	Procedimiento para preparar carboxamidas y tiocarboxamidas.
ES447116A Expired ES447116A1 (es)	1973-03-29	1976-04-15	Un procedimiento para preparar 2,4,5,6-tetrahidrociclopenta-(c)pirrol-4-carbonitrilos.

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
ES447116A Expired ES447116A1 (es)	1973-03-29	1976-04-15	Un procedimiento para preparar 2,4,5,6-tetrahidrociclopenta-(c)pirrol-4-carbonitrilos.

Country Status (6)

Country	Link
AR (1)	AR213064A1 (es)
ES (2)	ES424717A1 (es)
IE (1)	IE39694B1 (es)
IL (2)	IL44490A (es)
PH (1)	PH12366A (es)
SE (1)	SE7609982L (es)

1974
- 1974-03-25 IL IL44490A patent/IL44490A/xx unknown
- 1974-03-26 IE IE656/74A patent/IE39694B1/xx unknown
- 1974-03-28 ES ES424717A patent/ES424717A1/es not_active Expired
- 1974-03-29 PH PH7415680A patent/PH12366A/en unknown
- 1974-03-29 AR AR253065A patent/AR213064A1/es active
1976
- 1976-04-15 ES ES447116A patent/ES447116A1/es not_active Expired
- 1976-08-11 IL IL50239A patent/IL50239A0/xx unknown
- 1976-09-09 SE SE7609982A patent/SE7609982L/xx unknown

Also Published As

Publication number	Publication date
IE39694B1 (en)	1978-12-06
ES447116A1 (es)	1977-10-16
PH12366A (en)	1979-01-29
IL44490A (en)	1978-09-29
IL50239A0 (en)	1976-10-31
AR213064A1 (es)	1978-12-15
IE39694L (en)	1974-09-29
IL44490A0 (en)	1974-06-30
SE7609982L (sv)	1977-12-30

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