ES2191207T3 - Compuestos de carbapenem triciclicos. - Google Patents
Compuestos de carbapenem triciclicos.Info
- Publication number
- ES2191207T3 ES2191207T3 ES97951174T ES97951174T ES2191207T3 ES 2191207 T3 ES2191207 T3 ES 2191207T3 ES 97951174 T ES97951174 T ES 97951174T ES 97951174 T ES97951174 T ES 97951174T ES 2191207 T3 ES2191207 T3 ES 2191207T3
- Authority
- ES
- Spain
- Prior art keywords
- group
- tricycle
- formula
- elements
- constituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- YZBQHRLRFGPBSL-RXMQYKEDSA-N carbapenem Chemical class C1C=CN2C(=O)C[C@H]21 YZBQHRLRFGPBSL-RXMQYKEDSA-N 0.000 title 1
- QQONPFPTGQHPMA-UHFFFAOYSA-N Propene Chemical group CC=C QQONPFPTGQHPMA-UHFFFAOYSA-N 0.000 abstract 1
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 1
- 230000000844 anti-bacterial effect Effects 0.000 abstract 1
- 239000002131 composite material Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 125000001570 methylene group Chemical group [H]C([H])([*:1])[*:2] 0.000 abstract 1
- 229910052717 sulfur Inorganic materials 0.000 abstract 1
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Chemical compound O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D477/00—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- Animal Behavior & Ethology (AREA)
- Oncology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Steroid Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
LA PRESENTE INVENCION SE REFIERE A UN COMPUESTO DE LA FORMULA (I), SALES Y ESTERES METABOLICAMENTE LABILES DE DICHO COMPUESTO QUE TENGAN UNA ACTIVIDAD ANTIBACTERIANA, ASI COMO PROCEDIMIENTOS PARA SU PREPARACION Y USO EN MEDICINA. EN LA FORMULA, R REPRESENTA UN ARILO POSIBLEMENTE SUSTITUIDO O UN GRUPO HETEROARILO; A REPRESENTA UNA CADENA DE PROPILENO O ES UNA CADENA CONSTITUIDA DE 3 ELEMENTOS, DE LOS CUALES UNO PERTENECE AL GRUPO CONSTITUIDO POR UN ATOMO DE OXIGENO, POR UN ATOMO DE AZUFRE, DEL GRUPO NH O POR UN DERIVADO SUSTITUIDO DEL GRUPO, SIENDO LOS OTROS DOS ELEMENTOS DE LOS GRUPOS METILENO.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB9623684.9A GB9623684D0 (en) | 1996-11-14 | 1996-11-14 | Chemical compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2191207T3 true ES2191207T3 (es) | 2003-09-01 |
Family
ID=10802915
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES97951174T Expired - Lifetime ES2191207T3 (es) | 1996-11-14 | 1997-11-12 | Compuestos de carbapenem triciclicos. |
Country Status (17)
| Country | Link |
|---|---|
| EP (1) | EP0937078B1 (es) |
| JP (1) | JP2001503765A (es) |
| KR (1) | KR20000053258A (es) |
| AR (1) | AR010585A1 (es) |
| AT (1) | ATE232532T1 (es) |
| AU (1) | AU727328B2 (es) |
| BR (1) | BR9713982A (es) |
| CA (1) | CA2271732A1 (es) |
| DE (1) | DE69719054T2 (es) |
| ES (1) | ES2191207T3 (es) |
| GB (1) | GB9623684D0 (es) |
| HR (1) | HRP970611A2 (es) |
| PE (1) | PE14099A1 (es) |
| TR (1) | TR199901705T2 (es) |
| TW (1) | TW438802B (es) |
| WO (1) | WO1998021210A1 (es) |
| ZA (1) | ZA9710207B (es) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2321146A1 (en) | 1998-02-17 | 1999-08-19 | Nippon Kayaku Kabushiki Kaisha | Novel acetamide derivative and use thereof |
| US7601847B2 (en) | 2004-10-26 | 2009-10-13 | Wyeth | Preparation and purification of 4-(indazol-3-yl)phenols |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CZ435990A3 (cs) * | 1989-09-08 | 1999-11-17 | Glaxo S.P.A. | Kyselina 10-(1-hydroxyethyl)-11-oxo-1-azatricyklo/7,2,0,03,8/-undec-2en-2-karboxylová a její deriváty, způsob jejich výroby, použití pro výrobu farmaceutických prostředků a farmaceutické prostředky s jejich obsahem |
| AU636913B2 (en) * | 1989-10-11 | 1993-05-13 | Takeda Chemical Industries Ltd. | Tricyclic carbapenem compounds |
| CA2065079C (en) * | 1991-04-05 | 2003-03-18 | Michiyuki Sendai | Polycyclic carbapenem compounds, their production and use |
| JPH06166688A (ja) * | 1992-10-02 | 1994-06-14 | Takeda Chem Ind Ltd | カルバペネム化合物、その製造法および抗菌組成物 |
| JPH08245628A (ja) * | 1995-01-12 | 1996-09-24 | Takeda Chem Ind Ltd | カルバペネム化合物、その製造法および剤 |
-
1996
- 1996-11-14 GB GBGB9623684.9A patent/GB9623684D0/en active Pending
-
1997
- 1997-11-12 WO PCT/EP1997/006299 patent/WO1998021210A1/en active IP Right Grant
- 1997-11-12 ES ES97951174T patent/ES2191207T3/es not_active Expired - Lifetime
- 1997-11-12 AU AU54815/98A patent/AU727328B2/en not_active Ceased
- 1997-11-12 AR ARP970105280A patent/AR010585A1/es unknown
- 1997-11-12 JP JP52217698A patent/JP2001503765A/ja not_active Ceased
- 1997-11-12 DE DE69719054T patent/DE69719054T2/de not_active Expired - Lifetime
- 1997-11-12 TR TR1999/01705T patent/TR199901705T2/xx unknown
- 1997-11-12 PE PE1997001012A patent/PE14099A1/es not_active Application Discontinuation
- 1997-11-12 EP EP97951174A patent/EP0937078B1/en not_active Expired - Lifetime
- 1997-11-12 AT AT97951174T patent/ATE232532T1/de not_active IP Right Cessation
- 1997-11-12 ZA ZA9710207A patent/ZA9710207B/xx unknown
- 1997-11-12 BR BR9713982-3A patent/BR9713982A/pt not_active IP Right Cessation
- 1997-11-12 KR KR1019990704237A patent/KR20000053258A/ko not_active Application Discontinuation
- 1997-11-12 CA CA002271732A patent/CA2271732A1/en not_active Abandoned
- 1997-11-13 HR HR9623684.9A patent/HRP970611A2/hr not_active Application Discontinuation
- 1997-12-03 TW TW086118192A patent/TW438802B/zh active
Also Published As
| Publication number | Publication date |
|---|---|
| ATE232532T1 (de) | 2003-02-15 |
| JP2001503765A (ja) | 2001-03-21 |
| BR9713982A (pt) | 2000-05-02 |
| PE14099A1 (es) | 1999-03-19 |
| DE69719054D1 (de) | 2003-03-20 |
| EP0937078A1 (en) | 1999-08-25 |
| WO1998021210A1 (en) | 1998-05-22 |
| KR20000053258A (ko) | 2000-08-25 |
| ZA9710207B (en) | 1999-05-12 |
| TW438802B (en) | 2001-06-07 |
| AU5481598A (en) | 1998-06-03 |
| AR010585A1 (es) | 2000-06-28 |
| CA2271732A1 (en) | 1998-05-22 |
| GB9623684D0 (en) | 1997-01-08 |
| DE69719054T2 (de) | 2003-11-27 |
| HRP970611A2 (en) | 1998-10-31 |
| AU727328B2 (en) | 2000-12-07 |
| TR199901705T2 (xx) | 1999-12-21 |
| EP0937078B1 (en) | 2003-02-12 |
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