[go: up one dir, main page]

EE9900135A - N-(2-bensotiasolüül)-1-piperidiinetaanamiini derivaadid, nende valmistamine ja kasutamine raviks - Google Patents

N-(2-bensotiasolüül)-1-piperidiinetaanamiini derivaadid, nende valmistamine ja kasutamine raviks

Info

Publication number
EE9900135A
EE9900135A EEP199900135A EE9900135A EE9900135A EE 9900135 A EE9900135 A EE 9900135A EE P199900135 A EEP199900135 A EE P199900135A EE 9900135 A EE9900135 A EE 9900135A EE 9900135 A EE9900135 A EE 9900135A
Authority
EE
Estonia
Prior art keywords
piperidinethanamine
benzothiazolyl
therapy
derivatives
preparation
Prior art date
Application number
EEP199900135A
Other languages
English (en)
Estonian (et)
Inventor
Dargazanli Gihad
George Pascal
Lardenois Patrick
Frost Jonathan
Schoemaker Johannes
Renones Maria-Carmen
Magat Pascale
Original Assignee
Synthlabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthlabo filed Critical Synthlabo
Publication of EE9900135A publication Critical patent/EE9900135A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
EEP199900135A 1996-10-01 1997-09-26 N-(2-bensotiasolüül)-1-piperidiinetaanamiini derivaadid, nende valmistamine ja kasutamine raviks EE9900135A (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9611925A FR2753970B1 (fr) 1996-10-01 1996-10-01 Derives de n-(benzothiazol-2-yl) piperidine-1-ethanamine, leur preparation et leur application en therapeutique
PCT/FR1997/001692 WO1998014444A1 (fr) 1996-10-01 1997-09-26 Derives de n-(benzothiazol-2-yl)piperidine-1-ethanamine, leur preparation et leur application en therapeutique

Publications (1)

Publication Number Publication Date
EE9900135A true EE9900135A (et) 1999-12-15

Family

ID=9496217

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP199900135A EE9900135A (et) 1996-10-01 1997-09-26 N-(2-bensotiasolüül)-1-piperidiinetaanamiini derivaadid, nende valmistamine ja kasutamine raviks

Country Status (23)

Country Link
EP (1) EP0929550A1 (zh)
JP (1) JP2001501217A (zh)
KR (1) KR20000048767A (zh)
CN (1) CN1230959A (zh)
AR (1) AR009105A1 (zh)
AU (1) AU722147B2 (zh)
BG (1) BG103271A (zh)
BR (1) BR9711842A (zh)
CA (1) CA2266510A1 (zh)
CO (1) CO4650030A1 (zh)
CZ (1) CZ112699A3 (zh)
EE (1) EE9900135A (zh)
FR (1) FR2753970B1 (zh)
HU (1) HUP9904091A3 (zh)
IL (1) IL128902A (zh)
NO (1) NO991581L (zh)
NZ (1) NZ334553A (zh)
PL (1) PL332648A1 (zh)
SK (1) SK42299A3 (zh)
TR (1) TR199900634T2 (zh)
TW (1) TW438800B (zh)
WO (1) WO1998014444A1 (zh)
ZA (1) ZA978772B (zh)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9725541D0 (en) * 1997-12-02 1998-02-04 Pharmacia & Upjohn Spa Amino-benzothiazole derivatives
US6107313A (en) * 1998-10-02 2000-08-22 Combichem, Inc. Dopamine receptor antagonists
CZ2003182A3 (cs) 2000-06-21 2003-06-18 F. Hoffmann-La Roche Ag Deriváty benzothiazolu
US7087761B2 (en) 2003-01-07 2006-08-08 Hoffmann-La Roche Inc. Cyclization process for substituted benzothiazole derivatives
RU2006117631A (ru) * 2003-10-24 2007-12-10 Ф.Хоффманн-Ля Рош Аг (Ch) Антагонисты рецептора ссr3
PT1753760E (pt) 2004-05-24 2008-02-12 Hoffmann La Roche '' - metoxi - 7 - morfolin - 4 - il - benzotiazol - 2 - il) - amida do ácido 4 - hidroxi - 4 - metil - piperidina - 1 - carboxílico''
JP4633123B2 (ja) 2004-11-05 2011-02-16 エフ.ホフマン−ラ ロシュ アーゲー イソニコチン酸誘導体の製造方法
EP1863818B1 (en) 2005-03-23 2010-03-10 F.Hoffmann-La Roche Ag Acetylenyl-pyrazolo-pvrimidine derivatives as mglur2 antagonists
ES2340321T3 (es) 2005-09-27 2010-06-01 F.Hoffmann-La Roche Ag Oxadiazolilpirazolo-pirimidinas, como antagonistas de mglur2.

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1260474A (en) * 1984-12-03 1989-09-26 Raymond A. Stokbroekx Benzoxazol- and benzothiazolamine derivatives
KR930005004B1 (ko) * 1985-04-15 1993-06-11 쟈안센 파아마슈우티카 엔. 부이. 치환된 n-[(4-피페리디닐)알킬]이환 축합 옥사졸아민 및 티아졸아민의 제조방법

Also Published As

Publication number Publication date
FR2753970B1 (fr) 1998-10-30
BR9711842A (pt) 1999-08-24
IL128902A (en) 2001-07-24
NO991581L (no) 1999-06-01
BG103271A (en) 2000-05-31
NZ334553A (en) 2000-11-24
SK42299A3 (en) 1999-12-10
TR199900634T2 (xx) 1999-06-21
NO991581D0 (no) 1999-03-30
AU4463897A (en) 1998-04-24
AR009105A1 (es) 2000-03-08
CA2266510A1 (en) 1998-04-09
ZA978772B (en) 1998-03-27
CO4650030A1 (es) 1998-09-03
HUP9904091A2 (hu) 2000-05-28
CN1230959A (zh) 1999-10-06
HUP9904091A3 (en) 2000-07-28
KR20000048767A (ko) 2000-07-25
CZ112699A3 (cs) 1999-06-16
IL128902A0 (en) 2000-02-17
FR2753970A1 (fr) 1998-04-03
JP2001501217A (ja) 2001-01-30
WO1998014444A1 (fr) 1998-04-09
EP0929550A1 (fr) 1999-07-21
AU722147B2 (en) 2000-07-20
TW438800B (en) 2001-06-07
PL332648A1 (en) 1999-09-27

Similar Documents

Publication Publication Date Title
FI955235A0 (fi) Oksatsolidiinionijohdannaiset, niiden valmistus ja käyttö
EE04566B1 (et) Epotilooni derivaadid ja nende kasutamine meditsiinis
FI953479A0 (fi) 1-aryylipyrimidiinijohdannaiset ja niiden farmaseuttinen käyttö
EE9800459A (et) Spiro-piperidiini derivaadid ja nende kasutamine terapeutiliste toimeainetena
FI944600A (fi) Imidatsol-4-yylipiperidiinijohdannaisia, niiden valmistus ja niiden käyttö terapiassa
FI951370A0 (fi) Tiatsolidinin ja oksatsolidinin johdannaiset, niiden valmistus ja lääkinnällinen käyttö
EE05003B1 (et) Dihdro-1,3,5-triasiinamino derivaadid ja nende kasutamine ravis
EE9600172A (et) Puriin-6-ooni derivaadid, nende valmistamismeetod, kasutamine ravimite valmistamiseks ja ravimid
EE200000037A (et) Atsüülpiperasinüülpürimidiinide derivaadid, nende valmistamine ja kasutamine ravimitena
EE200100470A (et) Püridopüranoasepiini derivaadid, nende valmistamine ja terapeutiline kasutamine
NO955305L (no) Optisk aktive benzotiepinderivater, deres fremstilling og anvendelse
EE9700288A (et) Asatsükloalkaani derivaadid, nende valmistamine ja kasutamine ravis
EE9900218A (et) 1,4-diasabitsüklo[2.2.2]okt-2-üülmetüülbensoaadi derivaadid, nende valmistamine ja kasutamine raviks
EE200000056A (et) 4-okso-3,5-dihüdro-4H-püridasino[4.5-b]indool-1-etaanamiidi derivaadid, nende valmistamine ja kasutamine raviks
DK1025100T3 (da) 3-substituerede tetrahydropyridopyrimidinonderivater, fremstilling og anvendelsen heraf
EE9900135A (et) N-(2-bensotiasolüül)-1-piperidiinetaanamiini derivaadid, nende valmistamine ja kasutamine raviks
FI961977A (fi) N-substituoidut atsabisykloalkaanijohdannaiset, niiden valmistus ja käyttö
DK0835254T3 (da) Oxazolidinonderivater, deres fremstilling og deres terapeutiske anvendelse
EE9800333A (et) Uued furaandiarüülmetülideeni derivaadid, nende valmistamise meetod ja kasutamine teraapias
EE200000207A (et) 8-asabitsüklo[3.2.1]oktaan-3-metaanamiini derivaadid, nende valmistamine ja terapeutiline kasutamine
FI971317A0 (fi) Uusia heterosyklisiä, substituoituja imidatsolokinoksalinoneja, niiden valmistus ja käyttö
EE200000018A (et) 6-pürrolidiin-2-üülpüridiinid, nende valmistamine ja terapeutiline kasutamine
EE9800153A (et) 5-naftalen-1-üül-1,3-dioksaani derivaadid, nende valmistamine ja terapeutiline kasutamine
EE200100363A (et) ((Aminoiminometüül)amino)alkaankarboksamiidid ja nende kasutamine ravis
NO950560L (no) Piperazinderivater, deres fremstilling og terapautiske anvendelse