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ECSP15032859A - Derivados de n-(sustituido)-5-fluoro-4-imino-3-metil-2-oxo-3,4-dihidropirimidin-1(2h)-carboxilato - Google Patents

Derivados de n-(sustituido)-5-fluoro-4-imino-3-metil-2-oxo-3,4-dihidropirimidin-1(2h)-carboxilato

Info

Publication number
ECSP15032859A
ECSP15032859A ECIEPI201532859A ECPI201532859A ECSP15032859A EC SP15032859 A ECSP15032859 A EC SP15032859A EC IEPI201532859 A ECIEPI201532859 A EC IEPI201532859A EC PI201532859 A ECPI201532859 A EC PI201532859A EC SP15032859 A ECSP15032859 A EC SP15032859A
Authority
EC
Ecuador
Prior art keywords
imino
oxo
fluoro
derivatives
substituted
Prior art date
Application number
ECIEPI201532859A
Other languages
English (en)
Inventor
W Owen
Beth Lorsbach
Lindsay Stelzer
Chenglin Yao
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of ECSP15032859A publication Critical patent/ECSP15032859A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/22—O-Aryl or S-Aryl esters thereof
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Dentistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

La presente invención se relaciona con el campo de N-(sustituido)-5-fluoro-4-imino-3-metil-2-oxo-3,4-dihidropirimidin-1(2H)-carboxilatos y sus derivados y con el uso de éstos compuestos como fungicidas. También se proporcionan métodos para controlar una enfermedad fúngica como Septoria tritici, que comprende administrar una cantidad efectiva del compuesto fungicida a por lo menos una superficie asociada con la planta, la semilla o la tierra.
ECIEPI201532859A 2012-12-28 2015-07-28 Derivados de n-(sustituido)-5-fluoro-4-imino-3-metil-2-oxo-3,4-dihidropirimidin-1(2h)-carboxilato ECSP15032859A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201261747086P 2012-12-28 2012-12-28

Publications (1)

Publication Number Publication Date
ECSP15032859A true ECSP15032859A (es) 2015-11-30

Family

ID=51022033

Family Applications (1)

Application Number Title Priority Date Filing Date
ECIEPI201532859A ECSP15032859A (es) 2012-12-28 2015-07-28 Derivados de n-(sustituido)-5-fluoro-4-imino-3-metil-2-oxo-3,4-dihidropirimidin-1(2h)-carboxilato

Country Status (18)

Country Link
US (2) US9622474B2 (es)
EP (1) EP2938194B1 (es)
JP (1) JP6324994B2 (es)
KR (1) KR20150103096A (es)
CN (2) CN104902757B (es)
AU (1) AU2013370493B2 (es)
BR (1) BR102013033709B1 (es)
CA (1) CA2893778A1 (es)
CR (1) CR20150382A (es)
DK (1) DK2938194T3 (es)
EC (1) ECSP15032859A (es)
HU (1) HUE047711T2 (es)
IL (1) IL239561B (es)
MX (1) MX2015008441A (es)
PL (1) PL2938194T3 (es)
RU (1) RU2638556C2 (es)
UA (1) UA115462C2 (es)
WO (1) WO2014105844A1 (es)

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CN104902757B (zh) 2012-12-28 2019-01-08 阿达玛马克西姆股份有限公司 N-(取代的)-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-1(2h)-羧酸酯衍生物
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KR20170100547A (ko) 2014-12-30 2017-09-04 다우 아그로사이언시즈 엘엘씨 살진균 활성을 갖는 피콜린아미드
KR20170100549A (ko) 2014-12-30 2017-09-04 다우 아그로사이언시즈 엘엘씨 살진균 활성을 갖는 피콜린아미드 화합물
EP3240424B1 (en) 2014-12-30 2020-09-16 Dow AgroSciences LLC Use of picolinamide compounds as fungicides

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CA2935601C (en) 2013-12-31 2023-03-14 Adama Makhteshim Ltd. 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
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Also Published As

Publication number Publication date
HUE047711T2 (hu) 2020-05-28
DK2938194T3 (da) 2020-01-02
RU2638556C2 (ru) 2017-12-14
BR102013033709A2 (pt) 2015-10-06
EP2938194A4 (en) 2016-08-31
US9908855B2 (en) 2018-03-06
UA115462C2 (uk) 2017-11-10
JP6324994B2 (ja) 2018-05-16
RU2015131095A (ru) 2017-02-06
CN104902757A (zh) 2015-09-09
KR20150103096A (ko) 2015-09-09
IL239561B (en) 2018-01-31
US20160192653A1 (en) 2016-07-07
CN110003118A (zh) 2019-07-12
CA2893778A1 (en) 2014-07-03
MX2015008441A (es) 2015-09-23
HK1214475A1 (en) 2016-07-29
US9622474B2 (en) 2017-04-18
CR20150382A (es) 2015-08-21
JP2016507512A (ja) 2016-03-10
EP2938194B1 (en) 2019-11-27
WO2014105844A1 (en) 2014-07-03
IL239561A0 (en) 2015-08-31
CN104902757B (zh) 2019-01-08
AU2013370493B2 (en) 2017-08-17
EP2938194A1 (en) 2015-11-04
US20170204069A1 (en) 2017-07-20
BR102013033709B1 (pt) 2019-05-14
AU2013370493A1 (en) 2015-07-02
PL2938194T3 (pl) 2020-09-21

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