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ECSP088379A - Tabletas dispersables que comprenden deferasirox - Google Patents

Tabletas dispersables que comprenden deferasirox

Info

Publication number
ECSP088379A
ECSP088379A EC2008008379A ECSP088379A ECSP088379A EC SP088379 A ECSP088379 A EC SP088379A EC 2008008379 A EC2008008379 A EC 2008008379A EC SP088379 A ECSP088379 A EC SP088379A EC SP088379 A ECSP088379 A EC SP088379A
Authority
EC
Ecuador
Prior art keywords
available tablets
tablet
deferasirox
percent
pharmaceutically acceptable
Prior art date
Application number
EC2008008379A
Other languages
English (en)
Inventor
Jean Pierre Cassiere
Florian Battung
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of ECSP088379A publication Critical patent/ECSP088379A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0087Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/06Antianaemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2095Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente invención pertenece a una tableta dispersable que comprende: (a) el Compuesto I de la Fórmula (I), o una sal farmacéuticamente aceptable del mismo, presente en una cantidad del 42 por ciento al 65 por ciento en peso, basándose en el peso total de la tableta, y (b) cuando menos un excipiente farmacéuticamente aceptable adecuado para la preparación de tabletas dispersables, y para el procesamiento con el fin de fabricar dicha tableta dispersable.
EC2008008379A 2005-10-19 2008-04-17 Tabletas dispersables que comprenden deferasirox ECSP088379A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0553182 2005-10-19

Publications (1)

Publication Number Publication Date
ECSP088379A true ECSP088379A (es) 2008-05-30

Family

ID=36616771

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2008008379A ECSP088379A (es) 2005-10-19 2008-04-17 Tabletas dispersables que comprenden deferasirox

Country Status (17)

Country Link
US (1) US20080311194A1 (es)
EP (1) EP1940360A1 (es)
JP (1) JP2009512652A (es)
KR (1) KR20080056225A (es)
CN (1) CN101291655A (es)
AU (1) AU2006303514B2 (es)
BR (1) BRPI0617715A2 (es)
CA (1) CA2625112A1 (es)
EC (1) ECSP088379A (es)
IL (1) IL190397A0 (es)
MA (1) MA29841B1 (es)
NO (1) NO20082265L (es)
NZ (1) NZ567155A (es)
RU (1) RU2008119410A (es)
TN (1) TNSN08173A1 (es)
WO (1) WO2007045445A1 (es)
ZA (1) ZA200802670B (es)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2062572A1 (en) 2007-11-19 2009-05-27 Teva Pharmaceutical Industries Ltd. Pharmaceutical compositions
WO2010035282A1 (en) * 2008-09-24 2010-04-01 Matrix Laboratories Limited Pharmaceutical compositions comprising deferasirox
WO2012003987A1 (en) 2010-07-08 2012-01-12 Ratiopharm Gmbh Oral dosage form of deferasirox
CA2812505A1 (en) * 2010-10-01 2012-04-05 Cipla Limited Pharmaceutical composition
WO2014181108A1 (en) * 2013-05-10 2014-11-13 Cipla Limited Low dose pharmaceutical composition
JP2015536970A (ja) 2012-11-12 2015-12-24 シプラ・リミテッド デフェラシロクス及びデフェリプロンを含む固定用量医薬組成物
AP2015008668A0 (en) * 2013-03-08 2015-08-31 Novartis Ag Oral formulations of deferasirox
TR201909052T4 (tr) 2014-05-20 2019-07-22 Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi Deferasiroks içeren suda dağılabilen tablet formülasyonu.
EP2987482A1 (en) 2014-08-22 2016-02-24 Santa Farma Ilaç Sanayi A.S. Soluble and dispersible pharamaceutical deferasirox formulation
WO2016167729A1 (en) 2015-04-16 2016-10-20 Öğün Yusuf Toktamiş Dispersible tablets comprising deferasirox
EP3095443A1 (en) * 2015-05-21 2016-11-23 Abdi Ibrahim Ilac Sanayi ve Ticaret A.S. Pharmaceutical composition comprising deferasirox
AU2016280280B2 (en) * 2015-06-17 2021-09-02 AustinPx, LLC Improved formulations of deferasirox and methods of making the same
EP3481390A4 (en) * 2016-07-05 2020-03-04 Jubilant Generics Limited PHARMACEUTICAL COMPOSITION WITH IMMEDIATE RELEASE OF IRON CHELATE IMAGERS
EP3518904A1 (en) 2016-09-30 2019-08-07 Synthon B.V. Pharmaceutical composition comprising deferasirox
WO2018208242A1 (en) 2017-05-10 2018-11-15 İlko Ilaç Sanayi Ve Ticaret Anonim Şirketi Formulation of deferasirox tablet for oral suspension composition with better processability
EP3675832A1 (en) 2017-09-01 2020-07-08 Jordan Sweden Medical and Sterilization Company Fast self dispersible dosage forms of deferasirox
WO2019108157A1 (en) * 2017-11-28 2019-06-06 Biofarma Ilac Sanayi Ve Ticaret A.S. A scored tablet formulation in a dispersible form comprising deferasirox
TR201722910A2 (tr) 2017-12-29 2019-07-22 Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi Deferasi̇roks i̇çeren suda dağilabi̇len tablet formülasyonlari
WO2022240279A1 (es) * 2021-05-10 2022-11-17 Garcia Perez Miguel Angel Tableta dispersable con deferasirox en forma de dispersión sólida

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9215908D0 (en) * 1992-07-27 1992-09-09 Wellcome Found Water dispersible tablets
TW533205B (en) * 1996-06-25 2003-05-21 Novartis Ag Substituted 3,5-diphenyl-l,2,4-triazoles and their pharmaceutical composition
GB0223978D0 (en) * 2002-10-15 2002-11-20 Novartis Ag Organic compound

Also Published As

Publication number Publication date
NZ567155A (en) 2010-06-25
RU2008119410A (ru) 2009-11-27
EP1940360A1 (en) 2008-07-09
JP2009512652A (ja) 2009-03-26
US20080311194A1 (en) 2008-12-18
NO20082265L (no) 2008-05-16
CA2625112A1 (en) 2007-04-26
IL190397A0 (en) 2008-11-03
BRPI0617715A2 (pt) 2011-08-02
KR20080056225A (ko) 2008-06-20
CN101291655A (zh) 2008-10-22
AU2006303514B2 (en) 2010-06-24
ZA200802670B (en) 2009-10-28
WO2007045445A1 (en) 2007-04-26
MA29841B1 (fr) 2008-10-03
TNSN08173A1 (en) 2009-10-30
AU2006303514A1 (en) 2007-04-26

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