EA200870236A1 - Моногидрат римонабанта, способ его получения и фармацевтические композиции на его основе - Google Patents
Моногидрат римонабанта, способ его получения и фармацевтические композиции на его основеInfo
- Publication number
- EA200870236A1 EA200870236A1 EA200870236A EA200870236A EA200870236A1 EA 200870236 A1 EA200870236 A1 EA 200870236A1 EA 200870236 A EA200870236 A EA 200870236A EA 200870236 A EA200870236 A EA 200870236A EA 200870236 A1 EA200870236 A1 EA 200870236A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- monohydrate
- rhimnabant
- basis
- production
- pharmaceutical compositions
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 150000004682 monohydrates Chemical class 0.000 title 1
- 229960003015 rimonabant Drugs 0.000 abstract 1
- -1 rimonabant monohydrate Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Diabetes (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Biomedical Technology (AREA)
- Child & Adolescent Psychology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Настоящее изобретение относится к моногидрату римонабанта, к способу его получения и к содержащей его фармацевтической композиции.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0601253A FR2897060B1 (fr) | 2006-02-08 | 2006-02-08 | Le monohydrate de rimonabant, son procede de preparation et les compositions pharmaceutiques en contenant |
PCT/FR2007/000201 WO2007090949A1 (fr) | 2006-02-08 | 2007-02-05 | Le monohydrate de rimonabant, son procede de preparation et les compositions pharmaceutiques en contenant |
Publications (1)
Publication Number | Publication Date |
---|---|
EA200870236A1 true EA200870236A1 (ru) | 2009-02-27 |
Family
ID=37075667
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200870236A EA200870236A1 (ru) | 2006-02-08 | 2007-02-05 | Моногидрат римонабанта, способ его получения и фармацевтические композиции на его основе |
Country Status (20)
Country | Link |
---|---|
US (1) | US20090048449A1 (ru) |
EP (1) | EP1984341A1 (ru) |
JP (1) | JP2009526025A (ru) |
KR (1) | KR20080093042A (ru) |
CN (1) | CN101405271A (ru) |
AR (1) | AR059327A1 (ru) |
AU (1) | AU2007213649A1 (ru) |
BR (1) | BRPI0707711A2 (ru) |
CA (1) | CA2641494A1 (ru) |
DO (1) | DOP2007000023A (ru) |
EA (1) | EA200870236A1 (ru) |
FR (1) | FR2897060B1 (ru) |
GT (1) | GT200700014A (ru) |
IL (1) | IL192963A0 (ru) |
MA (1) | MA30312B1 (ru) |
NO (1) | NO20083521L (ru) |
TW (1) | TW200804343A (ru) |
UY (1) | UY30137A1 (ru) |
WO (1) | WO2007090949A1 (ru) |
ZA (1) | ZA200806713B (ru) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2057144A4 (en) * | 2006-09-01 | 2010-06-02 | Hetero Drugs Ltd | NEW POLYMORPHIC FROM RIMONABANT |
WO2008056377A2 (en) * | 2006-11-06 | 2008-05-15 | Cadila Healthcare Limited | Polymorphic forms of rimonabant |
HUE043014T2 (hu) * | 2014-12-08 | 2019-07-29 | Crystal Pharmatech Co Ltd | Valzartánt és AHU 377-et tartalmazó trinátrium szupramolekuláris komplex kristályos formái, és az ezekhez tartozó eljárások |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2713225B1 (fr) * | 1993-12-02 | 1996-03-01 | Sanofi Sa | N-pipéridino-3-pyrazolecarboxamide substitué. |
FR2831883B1 (fr) * | 2001-11-08 | 2004-07-23 | Sanofi Synthelabo | Forme polymorphe du rimonabant, son procede de preparation et les compositions pharmaceutiques en contenant |
JP4746931B2 (ja) * | 2005-07-22 | 2011-08-10 | 株式会社日立製作所 | フラットディスプレイパネルモジュール及びフラットディスプレイ装置 |
EP2057144A4 (en) * | 2006-09-01 | 2010-06-02 | Hetero Drugs Ltd | NEW POLYMORPHIC FROM RIMONABANT |
WO2008035023A1 (en) * | 2006-09-19 | 2008-03-27 | Cipla Limited | Polymorphs of rimonabant |
-
2006
- 2006-02-08 FR FR0601253A patent/FR2897060B1/fr not_active Expired - Fee Related
-
2007
- 2007-02-01 DO DO2007000023A patent/DOP2007000023A/es unknown
- 2007-02-05 CN CNA200780004742XA patent/CN101405271A/zh active Pending
- 2007-02-05 KR KR1020087019391A patent/KR20080093042A/ko not_active Withdrawn
- 2007-02-05 EP EP07730917A patent/EP1984341A1/fr not_active Withdrawn
- 2007-02-05 JP JP2008553793A patent/JP2009526025A/ja active Pending
- 2007-02-05 ZA ZA200806713A patent/ZA200806713B/xx unknown
- 2007-02-05 BR BRPI0707711-4A patent/BRPI0707711A2/pt not_active IP Right Cessation
- 2007-02-05 EA EA200870236A patent/EA200870236A1/ru unknown
- 2007-02-05 CA CA002641494A patent/CA2641494A1/fr not_active Abandoned
- 2007-02-05 AU AU2007213649A patent/AU2007213649A1/en not_active Abandoned
- 2007-02-05 WO PCT/FR2007/000201 patent/WO2007090949A1/fr active Application Filing
- 2007-02-06 AR ARP070100477A patent/AR059327A1/es unknown
- 2007-02-06 GT GT200700014A patent/GT200700014A/es unknown
- 2007-02-08 TW TW096104722A patent/TW200804343A/zh unknown
- 2007-02-08 UY UY30137A patent/UY30137A1/es not_active Application Discontinuation
-
2008
- 2008-07-22 IL IL192963A patent/IL192963A0/en unknown
- 2008-08-06 US US12/186,753 patent/US20090048449A1/en not_active Abandoned
- 2008-08-13 NO NO20083521A patent/NO20083521L/no not_active Application Discontinuation
- 2008-08-26 MA MA31195A patent/MA30312B1/fr unknown
Also Published As
Publication number | Publication date |
---|---|
ZA200806713B (en) | 2009-10-28 |
IL192963A0 (en) | 2009-02-11 |
KR20080093042A (ko) | 2008-10-17 |
CA2641494A1 (fr) | 2007-08-16 |
AR059327A1 (es) | 2008-03-26 |
DOP2007000023A (es) | 2008-02-15 |
FR2897060B1 (fr) | 2008-07-25 |
FR2897060A1 (fr) | 2007-08-10 |
WO2007090949A1 (fr) | 2007-08-16 |
MA30312B1 (fr) | 2009-04-01 |
TW200804343A (en) | 2008-01-16 |
BRPI0707711A2 (pt) | 2011-05-10 |
JP2009526025A (ja) | 2009-07-16 |
AU2007213649A1 (en) | 2007-08-16 |
UY30137A1 (es) | 2007-09-28 |
GT200700014A (es) | 2007-09-19 |
US20090048449A1 (en) | 2009-02-19 |
EP1984341A1 (fr) | 2008-10-29 |
NO20083521L (no) | 2008-10-24 |
CN101405271A (zh) | 2009-04-08 |
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EA200870236A1 (ru) | Моногидрат римонабанта, способ его получения и фармацевтические композиции на его основе |