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EA200200853A1 - Применение 2-метилтиазолидин-3,3-дикарбоновой кислоты (2-мтдк) и/или ее физиологически совместимых солей для лечения и/или предупреждения рака - Google Patents

Применение 2-метилтиазолидин-3,3-дикарбоновой кислоты (2-мтдк) и/или ее физиологически совместимых солей для лечения и/или предупреждения рака

Info

Publication number
EA200200853A1
EA200200853A1 EA200200853A EA200200853A EA200200853A1 EA 200200853 A1 EA200200853 A1 EA 200200853A1 EA 200200853 A EA200200853 A EA 200200853A EA 200200853 A EA200200853 A EA 200200853A EA 200200853 A1 EA200200853 A1 EA 200200853A1
Authority
EA
Eurasian Patent Office
Prior art keywords
treatment
mtdk
application
compatible salts
cancer prevention
Prior art date
Application number
EA200200853A
Other languages
English (en)
Other versions
EA004592B1 (ru
Inventor
Руди Зузило
Ханс Роммельшпахер
Original Assignee
Руди Зузило
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Руди Зузило filed Critical Руди Зузило
Publication of EA200200853A1 publication Critical patent/EA200200853A1/ru
Publication of EA004592B1 publication Critical patent/EA004592B1/ru

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/4261,3-Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Настоящее изобретение относится к применению 2-метилтиазолидин-2,4-дикарбоновой кислоты (2-МТДК) и/или ее физиологически совместимых солей для лечения и/или предупреждения рака.Отчет о международном поиске был опубликован 2002.05.30.
EA200200853A 2000-02-15 2001-02-15 Применение 2-метилтиазолидин-3,3-дикарбоновой кислоты (2-мтдк) и/или ее физиологически совместимых солей для лечения и/или предупреждения рака EA004592B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10008159A DE10008159B4 (de) 2000-02-15 2000-02-15 Verwendung von 2-Methyl-thiazolidin-2,4-dicarbonsäure und/oder ihrer physiologisch verträglichen Salze als Antikrebsmittel
PCT/DE2001/000656 WO2001060343A2 (de) 2000-02-15 2001-02-15 Verwendung von 2-methyl-thiazolidin-2,4-dicarbonsäure und/oder ihrer physiologisch verträglichen salze zur herstellung eines medikaments zur behandlung von krebserkrankungen

Publications (2)

Publication Number Publication Date
EA200200853A1 true EA200200853A1 (ru) 2003-02-27
EA004592B1 EA004592B1 (ru) 2004-06-24

Family

ID=7631906

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200200853A EA004592B1 (ru) 2000-02-15 2001-02-15 Применение 2-метилтиазолидин-3,3-дикарбоновой кислоты (2-мтдк) и/или ее физиологически совместимых солей для лечения и/или предупреждения рака

Country Status (15)

Country Link
US (2) US6943185B2 (ru)
EP (1) EP1255538B1 (ru)
JP (1) JP2003522782A (ru)
CN (1) CN1400899A (ru)
AT (1) ATE252383T1 (ru)
AU (1) AU783933B2 (ru)
CA (1) CA2399709C (ru)
DE (2) DE10008159B4 (ru)
EA (1) EA004592B1 (ru)
ES (1) ES2208571T3 (ru)
MX (1) MXPA02007903A (ru)
PL (1) PL357179A1 (ru)
PT (1) PT1255538E (ru)
TR (1) TR200302134T4 (ru)
WO (1) WO2001060343A2 (ru)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20050197406A1 (en) * 1999-04-14 2005-09-08 Li Chiang J. Method of treatment of lung cancer
DE10008159B4 (de) * 2000-02-15 2005-08-18 Rudy Dr. Susilo Verwendung von 2-Methyl-thiazolidin-2,4-dicarbonsäure und/oder ihrer physiologisch verträglichen Salze als Antikrebsmittel
NZ531890A (en) * 2002-02-28 2006-02-24 Japan Tobacco Inc Ester compound and medicinal use thereof
WO2005021486A1 (ja) * 2003-08-29 2005-03-10 Japan Tobacco Inc. エステル誘導体及びその医薬用途
DE102004021658A1 (de) * 2004-05-03 2005-12-01 Rudy Dr. Susilo Kombinationspräparate enthaltend 2-Methylthiazolidin-2,4-dicarbonsäure
US20060030623A1 (en) * 2004-07-16 2006-02-09 Noboru Furukawa Agent for the treatment or prevention of diabetes, obesity or arteriosclerosis
US8101774B2 (en) * 2004-10-18 2012-01-24 Japan Tobacco Inc. Ester derivatives and medicinal use thereof
CA2582767C (en) * 2004-10-25 2011-05-24 Japan Tobacco Inc. Solid formulation with improved solubility and stability and method for producing said formulation
JP5439849B2 (ja) * 2008-02-28 2014-03-12 味の素株式会社 システイン誘導体
JP5378713B2 (ja) * 2008-06-19 2013-12-25 日本理化学薬品株式会社 外用組成物

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19711052C2 (de) * 1997-03-03 1999-09-23 Hans Rommelspacher Verwendung von 2-Methyl-thiazolidin-2,4-dicarbonsäure als Mukolytikum
DE19711053C2 (de) 1997-03-03 1999-09-02 Rommelspacher Kombinationspräparat aus 2-Methyl-thiazolidin-2,4-dicarbonsäure und Paracetamol
DE10008159B4 (de) * 2000-02-15 2005-08-18 Rudy Dr. Susilo Verwendung von 2-Methyl-thiazolidin-2,4-dicarbonsäure und/oder ihrer physiologisch verträglichen Salze als Antikrebsmittel

Also Published As

Publication number Publication date
PT1255538E (pt) 2004-03-31
TR200302134T4 (tr) 2004-01-21
EP1255538A2 (de) 2002-11-13
ES2208571T3 (es) 2004-06-16
US20050187271A1 (en) 2005-08-25
JP2003522782A (ja) 2003-07-29
EP1255538B1 (de) 2003-10-22
ATE252383T1 (de) 2003-11-15
PL357179A1 (en) 2004-07-26
DE10008159A1 (de) 2001-09-06
CN1400899A (zh) 2003-03-05
US6943185B2 (en) 2005-09-13
AU3919001A (en) 2001-08-27
CA2399709A1 (en) 2001-08-23
DE50100833D1 (de) 2003-11-27
MXPA02007903A (es) 2004-09-10
WO2001060343A3 (de) 2002-05-30
WO2001060343A2 (de) 2001-08-23
AU783933B2 (en) 2005-12-22
US20030149085A1 (en) 2003-08-07
DE10008159B4 (de) 2005-08-18
CA2399709C (en) 2007-05-15
EA004592B1 (ru) 2004-06-24

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Legal Events

Date Code Title Description
MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ KZ KG MD TJ TM