[go: up one dir, main page]

DK89286D0 - Renininhiberende peptid-aminoalkoholderivater, som ogsaa inhiberer sure proteaser, fremgangsmaade til fremstilling deraf og derivaternes terapeutiske anvendelse - Google Patents

Renininhiberende peptid-aminoalkoholderivater, som ogsaa inhiberer sure proteaser, fremgangsmaade til fremstilling deraf og derivaternes terapeutiske anvendelse

Info

Publication number
DK89286D0
DK89286D0 DK89286A DK89286A DK89286D0 DK 89286 D0 DK89286 D0 DK 89286D0 DK 89286 A DK89286 A DK 89286A DK 89286 A DK89286 A DK 89286A DK 89286 D0 DK89286 D0 DK 89286D0
Authority
DK
Denmark
Prior art keywords
derivatives
aminoal
proteas
procedures
pure
Prior art date
Application number
DK89286A
Other languages
English (en)
Other versions
DK89286A (da
Inventor
Jean Wagnon
Remy Guegan
Colette Lacour
Dino Nisato
Original Assignee
Sanofi Sa
Inst Nat Sante Rech Med
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR8502763A external-priority patent/FR2577931B1/fr
Priority claimed from FR8511728A external-priority patent/FR2585708B1/fr
Application filed by Sanofi Sa, Inst Nat Sante Rech Med filed Critical Sanofi Sa
Publication of DK89286D0 publication Critical patent/DK89286D0/da
Publication of DK89286A publication Critical patent/DK89286A/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/0227—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the (partial) peptide sequence -Phe-His-NH-(X)2-C(=0)-, e.g. Renin-inhibitors with n = 2 - 6; for n > 6 see C07K5/06 - C07K5/10
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/06—Linear peptides containing only normal peptide links having 5 to 11 amino acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/0205—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -NH-(X)3-C(=0)-, e.g. statine or derivatives thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
DK89286A 1985-02-26 1986-02-26 Renininhiberende peptid-aminoalkoholderivater, som ogsaa inhiberer sure proteaser, fremgangsmaade til fremstilling deraf og derivaternes terapeutiske anvendelse DK89286A (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8502763A FR2577931B1 (fr) 1985-02-26 1985-02-26 Derives aminodiols peptidiques inhibiteurs de la renine et des proteases acides, leur procede de preparation et leur application en therapeutique
FR8511728A FR2585708B1 (fr) 1985-07-31 1985-07-31 Derives aminoalcools peptidiques inhibiteurs de la resine et des proteases acides, leur procede de preparation et leur application en therapeutique

Publications (2)

Publication Number Publication Date
DK89286D0 true DK89286D0 (da) 1986-02-26
DK89286A DK89286A (da) 1986-08-27

Family

ID=26224394

Family Applications (1)

Application Number Title Priority Date Filing Date
DK89286A DK89286A (da) 1985-02-26 1986-02-26 Renininhiberende peptid-aminoalkoholderivater, som ogsaa inhiberer sure proteaser, fremgangsmaade til fremstilling deraf og derivaternes terapeutiske anvendelse

Country Status (9)

Country Link
EP (1) EP0214209A1 (da)
KR (1) KR860006487A (da)
AU (1) AU587426B2 (da)
DK (1) DK89286A (da)
ES (1) ES8900018A1 (da)
GR (1) GR860532B (da)
NZ (1) NZ215282A (da)
PT (1) PT82077B (da)
WO (1) WO1986004901A1 (da)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4668663A (en) * 1984-03-27 1987-05-26 Merck & Co., Inc. Renin inhibitors containing homophe8
CA1290097C (en) * 1985-07-24 1991-10-01 Merck & Co., Inc. Peptide enzyme inhibitors
IL83663A0 (en) * 1986-10-27 1988-01-31 Robins Co Inc A H Preparation of 3-pyrrolidinols
NZ222755A (en) * 1986-12-23 1989-11-28 Warner Lambert Co Renin inhibiting acyl peptide derivatives containing two to four amino acid residues, and pharmaceutical compositions
DE3721855A1 (de) * 1987-03-12 1988-09-22 Merck Patent Gmbh Aminosaeurederivate
DE4136443A1 (de) * 1991-11-06 1993-05-13 Boehringer Ingelheim Int Expression der reifen proteinase 2a, ihre partielle reinigung und bereitstellung kompetitiv wirkender substrate
EP1346983A3 (en) * 1998-02-20 2003-12-03 Ortho-Mcneil Pharmaceutical, Inc. Phthalimido arylpiperazines as alpha 1A receptor antagonists useful in the treatment of benign prostatic hyperplasia
ZA991319B (en) * 1998-02-20 2000-11-20 Ortho Mcneil Pharm Inc Novel phthalimido arylpiperazines useful in the treatment of benign prostatic hyperplasia.
TW536538B (en) 1998-02-20 2003-06-11 Ortho Mcneil Pharm Inc Phthalimido arylpiperazines useful in the treatment of benign prostatic hyperplasia
EP2877485B1 (de) 2012-07-24 2018-03-14 Merck Patent GmbH Hydroxystatin-derivate zur behandlung von arthrose

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1245217A (en) * 1981-12-10 1988-11-22 Joshua S. Boger Renin inhibitory peptides having phe su13 xx deletion
US4595677A (en) * 1982-12-03 1986-06-17 Ciba-Geigy Corporation Substituted tetrapeptides
US4668663A (en) * 1984-03-27 1987-05-26 Merck & Co., Inc. Renin inhibitors containing homophe8
US4661473A (en) * 1984-03-27 1987-04-28 Merck & Co., Inc. Renin inhibitors containing peptide isosteres
US4636491A (en) * 1984-03-27 1987-01-13 Merck & Co., Inc. Renin inhibitory peptides having improved solubility
DE3418491A1 (de) * 1984-05-18 1985-11-21 Merck Patent Gmbh, 6100 Darmstadt Diaminosaeurederivate

Also Published As

Publication number Publication date
AU5410086A (en) 1986-09-04
PT82077A (fr) 1986-03-01
PT82077B (fr) 1987-09-25
NZ215282A (en) 1989-08-29
KR860006487A (ko) 1986-09-11
EP0214209A1 (fr) 1987-03-18
ES8900018A1 (es) 1988-11-16
AU587426B2 (en) 1989-08-17
DK89286A (da) 1986-08-27
GR860532B (en) 1986-06-24
ES552407A0 (es) 1988-11-16
WO1986004901A1 (fr) 1986-08-28

Similar Documents

Publication Publication Date Title
NO850817L (no) Fremgangsmaate for aa bevare effektiviteten til bakteriepreparater
ES556042A0 (es) Procedimiento para la obtencion de preparados de poliisocianato dispersables en agua
ES557643A0 (es) Procedimiento para la obtencion de derivados de acidos benzoheterociclilalcanoicos
DK110886D0 (da) Hidtil ukendte sulfonylaminoforbindelser, fremgangsmaader til deres fremstilling, og farmaceutiske praeparater, der indeholder forbindelserne
NO863061D0 (no) Fremgangsmaate for fremstilling av fysiologisk aktive fenoksyeddiksyrederivater.
DK213085A (da) Aminotetralinderivater, laegemidler indeholdende disse og fremgangsmaade til forbindelsernes fremstilling
NO864425L (no) Fremgangsmaate for fremstilling av terapeutisk aktive heterocyklyl-oksoftalazinyl-eddiksyre-derivater
NO165143C (no) Fremgangsmaate til fremstilling av hydrokloridet av fenyl-1-dietylaminokarbonyl-1-aminometyl-2-cyklopropan (z).
IT8522564A0 (it) Procedimento per la preparazione di idroalofluoroalcani.
NO862373D0 (no) Fremgangsmaate for fremstilling av terapeutisk aktive tienopyridoner.
NO870049D0 (no) Fremgangsmaate for fremstilling av terapeutisk aktive aminosyrederivater.
DK241585D0 (da) 8-chlor-quinolincarboxylsyre-derivater, fremgangsmaade til fremstilling deraf og farmaceutiske praeparater indeholdende saadanne forbindelser
IT8421622A1 (it) Procedimento per la preparazione di peptidi
DK89286D0 (da) Renininhiberende peptid-aminoalkoholderivater, som ogsaa inhiberer sure proteaser, fremgangsmaade til fremstilling deraf og derivaternes terapeutiske anvendelse
NO863373D0 (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive aminosyre derivater.
NO861584L (no) Fremgangsmaate til fremstilling av terapeutisk aktive cyklopentyletere.
IT1200400B (it) Procedimento per la preparazione di 2-alchil ciclopent-2-enoni
IT1183883B (it) Procedimento per la preparazione di amminoidrossicefamcarbossilati
IT1200594B (it) Procedimento per la preparazione di alfa-omega-aloperfluorocarburi
IT1191806B (it) Procedimento per la preparazione di 2-bromo-alfa-ergocriptina
IT1190358B (it) Procedimento per la preparazione di l-carnitina
DK515686A (da) Dopamin-beta-hydroxylase-inhibitorer og fremgangsmaade til fremstillingderaf
DK182186D0 (da) Ethanobenzazepiner, fremgangsmaade og mellemprodukter til deres fremstilling og deres anvendelse som laegemidler
DK164453C (da) Dibenzooeb,daathiopyran-6-carboxylsyreforbindelser, fremgangsmaade til fremstilling heraf og farmaceutiske praeparater indeholdende disse forbindelser
NO864689D0 (no) Fremgangsmaate for fremstilling av terapeutisk aktive peptider.

Legal Events

Date Code Title Description
AHB Application shelved due to non-payment