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DK76378A - F SOMOTOSTATINAL ANALOGUE AND METHOD OF MANUFACTURE THEREOF - Google Patents

F SOMOTOSTATINAL ANALOGUE AND METHOD OF MANUFACTURE THEREOF

Info

Publication number
DK76378A
DK76378A DK76378A DK76378A DK76378A DK 76378 A DK76378 A DK 76378A DK 76378 A DK76378 A DK 76378A DK 76378 A DK76378 A DK 76378A DK 76378 A DK76378 A DK 76378A
Authority
DK
Denmark
Prior art keywords
somotostatinal
analogue
manufacture
somotostatinal analogue
Prior art date
Application number
DK76378A
Other languages
Danish (da)
Other versions
DK150618C (en
DK150618B (en
Inventor
D Sarantakis
Original Assignee
American Home Prod
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/778,517 external-priority patent/US4077952A/en
Priority claimed from US05/830,930 external-priority patent/US4104267A/en
Priority claimed from US05/864,173 external-priority patent/US4190575A/en
Application filed by American Home Prod filed Critical American Home Prod
Publication of DK76378A publication Critical patent/DK76378A/en
Publication of DK150618B publication Critical patent/DK150618B/en
Application granted granted Critical
Publication of DK150618C publication Critical patent/DK150618C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10Tetrapeptides
    • C07K5/1002Tetrapeptides with the first amino acid being neutral
    • C07K5/1005Tetrapeptides with the first amino acid being neutral and aliphatic
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/02Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575Hormones
    • C07K14/655Somatostatins
    • C07K14/6555Somatostatins at least 1 amino acid in D-form
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Diabetes (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Endocrinology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Toxicology (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
DK076378A 1977-02-22 1978-02-21 ANALOGUE PROCEDURE FOR PREPARING SOMATOSTATIN ANALOGUE OR PHARMACEUTICAL ACCEPTABLE SALTS THEREOF DK150618C (en)

Applications Claiming Priority (10)

Application Number Priority Date Filing Date Title
US77095377A 1977-02-22 1977-02-22
US77095377 1977-02-22
US77851777 1977-03-17
US05/778,517 US4077952A (en) 1977-03-17 1977-03-17 Somatostatin analogs
US83093077 1977-09-06
US05/830,930 US4104267A (en) 1977-02-22 1977-09-06 Somatostatin analogs
GB4047177 1977-09-29
GB4047177 1977-09-29
US05/864,173 US4190575A (en) 1977-12-27 1977-12-27 Polypeptides related to somatostatin
US86417377 1977-12-27

Publications (3)

Publication Number Publication Date
DK76378A true DK76378A (en) 1978-08-23
DK150618B DK150618B (en) 1987-04-21
DK150618C DK150618C (en) 1987-10-19

Family

ID=27516344

Family Applications (1)

Application Number Title Priority Date Filing Date
DK076378A DK150618C (en) 1977-02-22 1978-02-21 ANALOGUE PROCEDURE FOR PREPARING SOMATOSTATIN ANALOGUE OR PHARMACEUTICAL ACCEPTABLE SALTS THEREOF

Country Status (5)

Country Link
DE (1) DE2807403A1 (en)
DK (1) DK150618C (en)
FR (1) FR2382433A1 (en)
IE (1) IE46462B1 (en)
SE (1) SE447482B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE7810156L (en) * 1977-12-13 1979-06-14 American Home Prod SOMATOSTATINAL ANALOGES
LU80207A1 (en) * 1978-09-07 1980-04-21 H Kalbacher NEW SUBSTITUTED CARBONIC ESTERS AND URETHANE, METHOD FOR THE PRODUCTION AND USE THEREOF
US4225472A (en) * 1979-05-29 1980-09-30 American Home Products Corporation Truncated somatostatin analogs

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4061608A (en) * 1976-07-13 1977-12-06 American Home Products Corporation Arg 4 -somatostatin and analogues thereof

Also Published As

Publication number Publication date
IE46462B1 (en) 1983-06-15
DE2807403A1 (en) 1978-08-31
SE447482B (en) 1986-11-17
DE2807403C2 (en) 1990-11-29
DK150618C (en) 1987-10-19
FR2382433B1 (en) 1983-12-09
FR2382433A1 (en) 1978-09-29
SE7802015L (en) 1978-10-16
IE780348L (en) 1978-08-22
DK150618B (en) 1987-04-21

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