DK633289A - RETROVIRAL PROTEASE INHIBITORS - Google Patents

RETROVIRAL PROTEASE INHIBITORS Download PDF

Info

Publication number: DK633289A
Authority: DK; Denmark
Prior art keywords: protease inhibitors; retroviral protease; retroviral; inhibitors; protease
Prior art date: 1988-12-15

Application number

DK633289A

Other languages

Danish (da)

Other versions

DK633289D0 (en

Inventor

Alexander Faessler

Ernst Hungerbuehler

Heinrich Rueeger

Peter Schneider

Original Assignee

Ciba Geigy Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1988-12-15

Filing date

1989-12-14

Publication date

1990-06-16

1989-12-14 Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag

1989-12-14 Publication of DK633289D0 publication Critical patent/DK633289D0/en

1990-06-16 Publication of DK633289A publication Critical patent/DK633289A/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/02—Linear peptides containing at least one abnormal peptide link
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
- C07K5/0207—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -NH-(X)4-C(=0), e.g. 'isosters', replacing two amino acids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Biochemistry (AREA)
Biophysics (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Virology (AREA)
Pharmacology & Pharmacy (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Crystallography & Structural Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Peptides Or Proteins (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

DK633289A 1988-12-15 1989-12-14 RETROVIRAL PROTEASE INHIBITORS DK633289A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
CH464088		1988-12-15

Publications (2)

Publication Number	Publication Date
DK633289D0 DK633289D0 (en)	1989-12-14
DK633289A true DK633289A (en)	1990-06-16

Family

ID=4279903

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK633289A DK633289A (en)	1988-12-15	1989-12-14	RETROVIRAL PROTEASE INHIBITORS

Country Status (15)

Country	Link
EP (1)	EP0374098A3 (en)
JP (1)	JPH02300199A (en)
KR (1)	KR900009692A (en)
AU (1)	AU626361B2 (en)
CA (1)	CA2005340A1 (en)
DD (1)	DD290894A5 (en)
DK (1)	DK633289A (en)
FI (1)	FI895962A0 (en)
HU (1)	HUT52525A (en)
IL (1)	IL92672A0 (en)
MX (1)	MX18736A (en)
NO (1)	NO895026L (en)
NZ (1)	NZ231750A (en)
PT (1)	PT92554A (en)
ZA (1)	ZA899558B (en)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CA2010531A1 (en) *	1989-03-06	1990-09-06	Werner Neidhart	Amino acid derivatives
AU7732691A (en) *	1990-06-01	1991-12-05	Ciba-Geigy Ag	Hiv protease inhibitors and processes for their preparation
DE4126485A1 (en) *	1991-08-10	1993-02-11	Bayer Ag	TRIFLUOROMETHYL-CONTAINING PSEUDOPEPTIDE
US5643878A (en) *	1991-09-12	1997-07-01	Ciba-Geigy Corporation	5-amino-4-hydroxyhexanoic acid derivatives
ATE253050T1 (en)	1992-03-11	2003-11-15	Narhex Ltd	AMINE DERIVATIVES OF OXO- AND HYDROXY-SUBSTITUTED HYDROCARBONS
JPH07504654A (en)	1992-03-11	1995-05-25	ナルヘックス　リミテッド	Amine derivatives of oxo- and hydroxy-substituted hydrocarbons
US5888992A (en)	1992-03-11	1999-03-30	Narhex Limited	Polar substituted hydrocarbons
US6071895A (en)	1992-03-11	2000-06-06	Narhex Limited	Polar-substituted hydrocarbons
TW217410B (en) *	1992-04-01	1993-12-11	Ciba Geigy
US5559256A (en) *	1992-07-20	1996-09-24	E. R. Squibb & Sons, Inc.	Aminediol protease inhibitors
EP0626178A1 (en) *	1993-05-17	1994-11-30	Ciba-Geigy Ag	Use of inhibitors of HIV-protease for the treatment of tumorous diseases
DE4332395A1 (en) *	1993-09-23	1995-04-13	Horst Dr Lindhofer	Inhibitors for the zymogen-like liberation cleavage of HIV-1 protease
JP3771591B2 (en)	1997-02-26	2006-04-26	ファイザー・インク	Heteroarylhexanoic acid amide derivatives, processes for their preparation and their use as selective inhibitors of MIP-1α binding to the CCR1 receptor
JP2002538151A (en)	1999-03-02	2002-11-12	ベーリンガーインゲルハイムファーマシューティカルズインコーポレイテッド	Compounds useful as reversible inhibitors of cathepsin
US6420364B1 (en)	1999-09-13	2002-07-16	Boehringer Ingelheim Pharmaceuticals, Inc.	Compound useful as reversible inhibitors of cysteine proteases
EA200401099A1 (en) *	2000-02-04	2005-02-24	Пфайзер Продактс Инк.	Derivatives of Heterocyclic Amide
EP1498417A1 (en) *	2000-02-04	2005-01-19	Pfizer Products Inc.	Heterocyclic amide derivatives

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4727060A (en) *	1984-11-13	1988-02-23	Ciba-Geigy Corporation	Novel 5-amino-4-hydroxyvaleryl derivatives
HU204285B (en) *	1986-10-31	1991-12-30	Pfizer	Process for producing renin-inhibiting polypeptides of small molecule mass and pharmaceutical compositions containing them

1989
- 1989-12-06 EP EP19890810923 patent/EP0374098A3/en not_active Withdrawn
- 1989-12-13 CA CA002005340A patent/CA2005340A1/en not_active Abandoned
- 1989-12-13 PT PT92554A patent/PT92554A/en not_active Application Discontinuation
- 1989-12-13 DD DD89335619A patent/DD290894A5/en not_active IP Right Cessation
- 1989-12-13 NZ NZ231750A patent/NZ231750A/en unknown
- 1989-12-13 FI FI895962A patent/FI895962A0/en not_active Application Discontinuation
- 1989-12-13 IL IL92672A patent/IL92672A0/en unknown
- 1989-12-14 HU HU896611A patent/HUT52525A/en unknown
- 1989-12-14 ZA ZA899558A patent/ZA899558B/en unknown
- 1989-12-14 KR KR1019890018523A patent/KR900009692A/en not_active Application Discontinuation
- 1989-12-14 AU AU46784/89A patent/AU626361B2/en not_active Ceased
- 1989-12-14 NO NO89895026A patent/NO895026L/en unknown
- 1989-12-14 DK DK633289A patent/DK633289A/en not_active Application Discontinuation
- 1989-12-15 JP JP1324111A patent/JPH02300199A/en active Pending
- 1989-12-15 MX MX1873689A patent/MX18736A/en unknown

Also Published As

Publication number	Publication date
DD290894A5 (en)	1991-06-13
EP0374098A3 (en)	1991-05-02
NO895026L (en)	1990-06-18
KR900009692A (en)	1990-07-05
NO895026D0 (en)	1989-12-14
IL92672A0 (en)	1990-09-17
FI895962A0 (en)	1989-12-13
CA2005340A1 (en)	1990-06-15
JPH02300199A (en)	1990-12-12
EP0374098A2 (en)	1990-06-20
MX18736A (en)	1994-02-28
NZ231750A (en)	1992-08-26
AU626361B2 (en)	1992-07-30
HUT52525A (en)	1990-07-28
DK633289D0 (en)	1989-12-14
AU4678489A (en)	1990-06-21
ZA899558B (en)	1990-08-29
PT92554A (en)	1990-06-29

Publication	Publication Date	Title
DK674387A (en)	1988-06-23	protease inhibitors
IL90218A0 (en)	1989-12-15	Retroviral protease inhibitors
MX9100119A (en)	1992-02-28	RETROVIRAL PROTEASE INHIBITORS
DE3689314D1 (en)	1994-01-05	Peptide inhibitor.
DE3785615D1 (en)	1993-06-03	SERIN PROTEASE INHIBITORS.
DK317287D0 (en)	1987-06-22	Reductase inhibitors
EP0428849A3 (en)	1991-07-31	Retroviral protease inhibitors
DK633289D0 (en)	1989-12-14	RETROVIRAL PROTEASE INHIBITORS
NO934628D0 (en)	1993-12-15	Retroviral protease inhibitors
BR8907457A (en)	1991-04-02	INTERLEUCIN-1 INHIBITORS
MX9100120A (en)	1992-02-28	RETROVIRAL PROTEASE INHIBITORS
DK349586D0 (en)	1986-07-23	enzyme inhibitor
FI101796B1 (en)	1998-08-31	New-glucosidase inhibitors
DK174087A (en)	1987-10-08	ANGIOTENSIN CONVERTERING ENZYMIN INHIBITOR
DE68922014D1 (en)	1995-05-11	Protease.
DK69489A (en)	1989-08-17	ASPARTATTRANSCARBAMYLASE INHIBITORS
NO872985L (en)	1988-01-22	INHIBITOR FOR POLYURETHANPROPERGOLS.
BR8902293A (en)	1990-01-09	ABRASIVE
KR900004589U (en)	1990-03-07	long time
KR890023207U (en)	1989-12-02	Relationship
DK658489A (en)	1989-12-22	protease inhibitors
MX22596A (en)	1993-11-01	RETROVIRAL PROTEASE INHIBITORS.
IS3397A7 (en)	1989-02-15	Enzyme inhibitors (Protease Inhibitors)
IE894013L (en)	1990-06-15	Retroviral protease inhibitors
ATE88720T1 (en)	1993-05-15	SERIN PROTEASE INHIBITORS.

Legal Events

Date	Code	Title	Description
1994-08-22	AHB	Application shelved due to non-payment