DK51878A - SEMI-SYNTHETIC 4 "-ERYTHROMYCIN A DERIVATIVES PROCEDURE FOR THEIR PREPARATION AND INTERMEDIATE PRODUCTS - Google Patents

SEMI-SYNTHETIC 4 "-ERYTHROMYCIN A DERIVATIVES PROCEDURE FOR THEIR PREPARATION AND INTERMEDIATE PRODUCTS

Info

Publication number: DK51878A
Authority: DK; Denmark
Prior art keywords: erythromycin; semi; synthetic; preparation; intermediate products
Prior art date: 1977-02-04

Application number

DK51878A

Other languages

Danish (da)

Other versions

DK148036B (en

DK148036C (en

Inventor

F C Sciavolino

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1977-02-04

Filing date

1978-02-03

Publication date

1978-08-05

1977-12-01 Priority claimed from US05/856,479 external-priority patent/US4150220A/en

1978-02-03 Application filed by Pfizer filed Critical Pfizer

1978-08-05 Publication of DK51878A publication Critical patent/DK51878A/en

1985-02-11 Publication of DK148036B publication Critical patent/DK148036B/en

1985-07-15 Application granted granted Critical

1985-07-15 Publication of DK148036C publication Critical patent/DK148036C/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Oncology (AREA)
Animal Behavior & Ethology (AREA)
Communicable Diseases (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Engineering & Computer Science (AREA)
Biochemistry (AREA)
Biotechnology (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Saccharide Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

DK51878A 1977-02-04 1978-02-03 METHOD OF ANALOGUE FOR THE PREPARATION OF EPIMERE 4 '' - AMINO-ERYTHROMYCIN COMPOUNDS OR ACID ADDITION SALTS. DK148036C (en)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
US76548077A	1977-02-04	1977-02-04
US76548077		1977-02-04
US05/856,479 US4150220A (en)	1977-02-04	1977-12-01	Semi-synthetic 4"-erythromycin A derivatives
US85647977		1977-12-01

Publications (3)

Publication Number	Publication Date
DK51878A true DK51878A (en)	1978-08-05
DK148036B DK148036B (en)	1985-02-11
DK148036C DK148036C (en)	1985-07-15

Family

ID=27117613

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK51878A DK148036C (en)	1977-02-04	1978-02-03	METHOD OF ANALOGUE FOR THE PREPARATION OF EPIMERE 4 '' - AMINO-ERYTHROMYCIN COMPOUNDS OR ACID ADDITION SALTS.

Country Status (30)

Country	Link
JP (1)	JPS5827798B2 (en)
AR (1)	AR222147A1 (en)
AU (1)	AU501298B1 (en)
BG (2)	BG32718A3 (en)
CA (1)	CA1106367A (en)
CH (1)	CH628906A5 (en)
CS (1)	CS221801B2 (en)
DD (1)	DD140048A5 (en)
DE (1)	DE2804507C2 (en)
DK (1)	DK148036C (en)
ES (2)	ES466057A1 (en)
FI (1)	FI780354A (en)
FR (2)	FR2379550A1 (en)
GB (2)	GB1585316A (en)
GR (1)	GR68691B (en)
HU (1)	HU182559B (en)
IE (1)	IE46661B1 (en)
IL (2)	IL53968A0 (en)
IT (1)	IT1094209B (en)
LU (1)	LU79004A1 (en)
NL (1)	NL176174C (en)
NO (2)	NO146472C (en)
NZ (1)	NZ186385A (en)
PH (2)	PH14421A (en)
PL (1)	PL116228B1 (en)
PT (1)	PT67568B (en)
RO (4)	RO79686A7 (en)
SE (2)	SE445223B (en)
SU (1)	SU927122A3 (en)
YU (3)	YU40913B (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4133950A (en) *	1978-01-03	1979-01-09	Pfizer Inc.	4"-Deoxy-4"-carbamate and dithiocarbamate derivatives of oleandomycin and its esters
US4124755A (en) *	1978-01-03	1978-11-07	Pfizer Inc.	11-Alkanoyl-4"-deoxy-4"-isonitrilo-oleandomycin derivatives
US4382085A (en) *	1982-03-01	1983-05-03	Pfizer Inc.	4"-Epi erythromycin A and derivatives thereof as useful antibacterial agents
US4518590A (en) *	1984-04-13	1985-05-21	Pfizer Inc.	9α-Aza-9α-homoerythromycin compounds, pharmaceutical compositions and therapeutic method
HN1998000074A (en) *	1997-06-11	1999-01-08	Pfizer Prod Inc	DERIVATIVES FROM MACROLIDES C-4 SUBSTITUTED
US6407074B1 (en)	1997-06-11	2002-06-18	Pfizer Inc	C-4″-substituted macrolide derivatives

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3836519A (en) *	1973-05-04	1974-09-17	Abbott Lab	Sulfonyl derivatives of erythromycin
US3884903A (en) *	1973-06-21	1975-05-20	Abbott Lab	4{41 -Deoxy-4{41 -oxoerythromycin B derivatives

1978
- 1978-01-10 SE SE7800270A patent/SE445223B/en not_active IP Right Cessation
- 1978-01-13 PH PH20662A patent/PH14421A/en unknown
- 1978-01-17 ES ES466057A patent/ES466057A1/en not_active Expired
- 1978-01-18 AR AR270752A patent/AR222147A1/en active
- 1978-01-18 YU YU73/78A patent/YU40913B/en unknown
- 1978-01-23 PT PT67568A patent/PT67568B/en unknown
- 1978-01-31 CH CH106178A patent/CH628906A5/en not_active IP Right Cessation
- 1978-02-02 CS CS78703A patent/CS221801B2/en unknown
- 1978-02-02 DE DE2804507A patent/DE2804507C2/en not_active Expired
- 1978-02-02 CA CA296,037A patent/CA1106367A/en not_active Expired
- 1978-02-02 GB GB34309/79A patent/GB1585316A/en not_active Expired
- 1978-02-02 GR GR55330A patent/GR68691B/el unknown
- 1978-02-02 GB GB4165/78A patent/GB1585315A/en not_active Expired
- 1978-02-02 RO RO78101650A patent/RO79686A7/en unknown
- 1978-02-02 RO RO78101651A patent/RO79687A7/en unknown
- 1978-02-02 RO RO7893080A patent/RO77345A/en unknown
- 1978-02-02 RO RO105255A patent/RO81622B/en unknown
- 1978-02-03 IL IL53968A patent/IL53968A0/en not_active IP Right Cessation
- 1978-02-03 BG BG038579A patent/BG32718A3/en unknown
- 1978-02-03 DK DK51878A patent/DK148036C/en not_active IP Right Cessation
- 1978-02-03 NZ NZ186385A patent/NZ186385A/en unknown
- 1978-02-03 BG BG040069A patent/BG33159A3/en unknown
- 1978-02-03 FR FR7803066A patent/FR2379550A1/en active Granted
- 1978-02-03 DD DD78203547A patent/DD140048A5/en unknown
- 1978-02-03 PL PL1978204428A patent/PL116228B1/en unknown
- 1978-02-03 SU SU782573754A patent/SU927122A3/en active
- 1978-02-03 IE IE239/78A patent/IE46661B1/en not_active IP Right Cessation
- 1978-02-03 HU HU78PI611A patent/HU182559B/en not_active IP Right Cessation
- 1978-02-03 NL NLAANVRAGE7801262,A patent/NL176174C/en not_active IP Right Cessation
- 1978-02-03 LU LU79004A patent/LU79004A1/en unknown
- 1978-02-03 JP JP53011352A patent/JPS5827798B2/en not_active Expired
- 1978-02-03 AU AU32990/78A patent/AU501298B1/en not_active Expired
- 1978-02-03 FI FI780354A patent/FI780354A/en not_active Application Discontinuation
- 1978-02-03 NO NO780389A patent/NO146472C/en unknown
- 1978-02-03 IT IT20005/78A patent/IT1094209B/en active
- 1978-07-07 FR FR7820334A patent/FR2385735A1/en active Granted
- 1978-08-08 ES ES472429A patent/ES472429A1/en not_active Expired
- 1978-09-01 PH PH21555A patent/PH16675A/en unknown
1981
- 1981-01-27 IL IL61997A patent/IL61997A0/en unknown
- 1981-06-05 NO NO811913A patent/NO150484C/en unknown
1983
- 1983-02-07 YU YU265/83A patent/YU40798B/en unknown
- 1983-02-16 SE SE8300870A patent/SE457086B/en not_active IP Right Cessation
- 1983-11-21 YU YU2279/83A patent/YU40799B/en unknown

Also Published As

Publication number	Publication date
NL176174B (en)	1984-10-01
AU501298B1 (en)	1979-06-14
DD140048A5 (en)	1980-02-06
DE2804507A1 (en)	1978-08-10
NO150484B (en)	1984-07-16
NO811913L (en)	1978-08-07
PH16675A (en)	1983-12-13
SE445223B (en)	1986-06-09
DK148036B (en)	1985-02-11
NL7801262A (en)	1978-08-08
RO81622B (en)	1983-04-30
YU26583A (en)	1984-02-29
FR2385735A1 (en)	1978-10-27
FR2379550B1 (en)	1980-07-04
ES472429A1 (en)	1979-04-01
IT7820005A0 (en)	1978-02-03
BG33159A3 (en)	1982-12-15
ES466057A1 (en)	1978-10-01
SU927122A3 (en)	1982-05-07
CS221801B2 (en)	1983-04-29
PH14421A (en)	1981-07-10
YU40799B (en)	1986-06-30
GB1585315A (en)	1981-02-25
JPS5827798B2 (en)	1983-06-11
PL116228B1 (en)	1981-05-30
SE8300870D0 (en)	1983-02-16
IE780239L (en)	1978-08-04
IL53968A0 (en)	1978-04-30
NL176174C (en)	1985-03-01
NO146472B (en)	1982-06-28
IT1094209B (en)	1985-07-26
YU7378A (en)	1983-04-30
HU182559B (en)	1984-02-28
GR68691B (en)	1982-02-01
NO146472C (en)	1982-10-06
DE2804507C2 (en)	1982-11-04
NO150484C (en)	1984-10-24
RO81622A (en)	1983-04-29
RO79686A7 (en)	1982-08-17
JPS53101337A (en)	1978-09-04
YU40913B (en)	1986-08-31
DK148036C (en)	1985-07-15
RO77345A (en)	1981-08-17
SE457086B (en)	1988-11-28
IL61997A0 (en)	1981-02-27
SE7800270L (en)	1978-08-05
BG32718A3 (en)	1982-09-15
AR222147A1 (en)	1981-04-30
CA1106367A (en)	1981-08-04
LU79004A1 (en)	1979-09-06
PT67568B (en)	1979-06-18
GB1585316A (en)	1981-02-25
YU227983A (en)	1984-04-30
FR2385735B1 (en)	1980-10-24
RO79687A7 (en)	1982-08-17
IE46661B1 (en)	1983-08-24
FI780354A (en)	1978-08-05
NO780389L (en)	1978-08-07
PT67568A (en)	1978-02-01
FR2379550A1 (en)	1978-09-01
YU40798B (en)	1986-06-30
NZ186385A (en)	1980-10-08
CH628906A5 (en)	1982-03-31
PL204428A1 (en)	1979-06-04
SE8300870L (en)	1983-02-16

Publication	Publication Date	Title
DK377678A (en)	1979-02-28	3,4,5-TRIHYDROXYPIPERIDINE DERIVATIVES THEIR PREPARATION AND USE
JPS53116356A (en)	1978-10-11	Derivative of chalcone and its preparation
NO783471L (en)	1979-04-18	XANTINE DERIVATIVES AND PROCEDURES FOR THEIR PREPARATION
DK522578A (en)	1979-05-26	G PROSTACYCLIN DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION
IL55555A0 (en)	1978-12-17	Novel 3-phenyl-azacycloalkane derivatives and their preparation
JPS545999A (en)	1979-01-17	Novel benzoquinolidine derivative and its preparation
DK313878A (en)	1979-01-14	CONTAINING DERIVATIVES AND PROCEDURE FOR THE PREPARATION THEREOF
DK495578A (en)	1979-05-09	QUINAZOLE DERIVATIVES AND METHODS OF PREPARATION
DK150778A (en)	1978-10-06	PROSTAND DERIVATIVES AND PROCEDURES FOR MANUFACTURE THEREOF
NZ186095A (en)	1979-03-28	Phenylcarbamoylpyrazoline derivatives and pesticidal compositions
NZ186096A (en)	1979-03-16	Phenylcarbamoyl-2-pyrazdine derivatives and pesticidal compositions
NO780800L (en)	1978-09-12	AZO COMPOUNDS AND PROCEDURES FOR THEIR PREPARATION
DK582578A (en)	1979-06-30	2,4-THIAZOLIDINDION DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION
DK331978A (en)	1979-01-30	NITROSOURIN INDUSTRIAL DERIVATIVES AND PROCEDURES FOR THE PREPARATION
GB2001630B (en)	1982-03-17	Inosadiamine derivatives and their preparation
DK355378A (en)	1979-02-13	4-HYDROXY-2-BENZIMIDAZONE DERIVATIVES AND PROCEDURES
DK308878A (en)	1979-02-19	AMINOGLYOSIDE DERIVATIVES AND PROCEDURES FOR THEIR PREPARATION
DK51878A (en)	1978-08-05	SEMI-SYNTHETIC 4 "-ERYTHROMYCIN A DERIVATIVES PROCEDURE FOR THEIR PREPARATION AND INTERMEDIATE PRODUCTS
DK63080A (en)	1980-08-16	25-HYDROXY-24-OXOCHLOSTANDER DERIVATIVES AND PROCEDURES FOR PREPARING THEREOF
IL54252A0 (en)	1978-06-15	Novel -aryl-acetamide derivatives and their preparation
DK416278A (en)	1979-03-23	2-OXAZOLIDON DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION
DK319478A (en)	1979-01-19	ANGIOTENSINPEPTIDES AND THEIR PREPARATION
ZA781598B (en)	1979-06-27	4-alkylthio-2-trifluoromethylalkanesulfonanilides and derivatives thereof
DK51778A (en)	1978-08-05	SEMI-SYNTHETIC 4 "AMINO-OLEANDOMYCIN DERIVATIVES AND THEIR MANUFACTURE
DK21579A (en)	1979-07-21	5-PHENETHYL-2-OXAZOLIDON DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION

Legal Events

Date	Code	Title	Description
1994-10-24	PBP	Patent lapsed