DK454188A - 2-oxo-1-sulfonylaminocarbonyl-azetidiner samt fremgangsmaade til deres fremstilling - Google Patents
2-oxo-1-sulfonylaminocarbonyl-azetidiner samt fremgangsmaade til deres fremstillingInfo
- Publication number
- DK454188A DK454188A DK454188A DK454188A DK454188A DK 454188 A DK454188 A DK 454188A DK 454188 A DK454188 A DK 454188A DK 454188 A DK454188 A DK 454188A DK 454188 A DK454188 A DK 454188A
- Authority
- DK
- Denmark
- Prior art keywords
- sulphonylaminocarbonyl
- azetidines
- oxo
- procedures
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
- C07D205/085—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a nitrogen atom directly attached in position 3
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US07/085,050 US4777252A (en) | 1987-08-13 | 1987-08-13 | 2-oxo-1-[[(substituted sulfonyl)amino]-carbonyl]azetidines |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK454188D0 DK454188D0 (da) | 1988-08-12 |
| DK454188A true DK454188A (da) | 1989-02-14 |
Family
ID=22189148
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK454188A DK454188A (da) | 1987-08-13 | 1988-08-12 | 2-oxo-1-sulfonylaminocarbonyl-azetidiner samt fremgangsmaade til deres fremstilling |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US4777252A (da) |
| EP (1) | EP0303286A1 (da) |
| JP (1) | JPH0196181A (da) |
| AU (1) | AU2091988A (da) |
| DK (1) | DK454188A (da) |
| HU (1) | HU201547B (da) |
| NZ (1) | NZ225821A (da) |
| ZA (1) | ZA885998B (da) |
Families Citing this family (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR890700586A (ko) * | 1987-02-27 | 1989-04-25 | 로버어트 에이 아마테이지 | 피리돈 카르복실산 또는 산유도체를 함유하는 항균제 베타-락탐 |
| US4904775A (en) * | 1988-05-16 | 1990-02-27 | E. R. Squibb & Sons, Inc. | Heteroaroylhydrazide derivatives of monocyclic beta-lactam antibiotics |
| FR2653429B1 (fr) * | 1989-10-25 | 1991-12-20 | Adir | Nouveaux derives de l'azetidin-2-one, 1,3,4-trisubstitues, intermediaires utiles pour la synthese des beta-lactames, et leur procede de synthese asymetrique. |
| GB9008850D0 (en) * | 1990-04-19 | 1990-06-13 | Janssen Pharmaceutica Nv | Novel 2,9-disubstituted-4h-pyridol(1,2-a)pyrimidin-4-ones |
| IL99658A0 (en) * | 1990-10-15 | 1992-08-18 | Merck & Co Inc | Substituted azetidinones and pharmaceutical compositions containing them |
| CN1128790C (zh) * | 1997-12-22 | 2003-11-26 | 法玛西雅厄普约翰美国公司 | 用作抗病毒剂的4－羟基喹啉－3－甲酰胺和酰肼化合物 |
| ES2235883T3 (es) * | 1999-05-06 | 2005-07-16 | Neurogen Corporation | 4-oxo-quinolino-3-carboxamidas sustituidas: ligandos de receptores cerebrales gaba. |
| US20100074949A1 (en) | 2008-08-13 | 2010-03-25 | William Rowe | Pharmaceutical composition and administration thereof |
| US7056917B2 (en) * | 2001-04-26 | 2006-06-06 | Daiichi Pharmaceutical Co., Ltd. | Drug efflux pump inhibitor |
| US20050009843A1 (en) * | 2001-04-26 | 2005-01-13 | Kiyoshi Nakayama | Medicine for inhibiting drug elimination pump |
| PT2489659T (pt) | 2004-06-24 | 2018-03-07 | Vertex Pharma | Moduladores de transportadores de cassete de ligação a atp |
| US8354427B2 (en) | 2004-06-24 | 2013-01-15 | Vertex Pharmaceutical Incorporated | Modulators of ATP-binding cassette transporters |
| JP2006131568A (ja) * | 2004-11-08 | 2006-05-25 | Ueno Seiyaku Oyo Kenkyusho:Kk | ヒドロキシナフトエ酸ヒドラジドおよびその誘導体ならびにその製造方法 |
| CN101374849A (zh) * | 2005-12-24 | 2009-02-25 | 沃泰克斯药物股份有限公司 | 作为abc转运蛋白调控剂的喹啉-4-酮衍生物 |
| SI3219705T1 (sl) | 2005-12-28 | 2020-08-31 | Vertex Pharmaceuticals Incorporated | Farmacevtski sestavki amorfne oblike N-(2,4-bis(1,1-dimetiletil)-5- hidroksifenil)-1,4-dihidro-4-oksokinolin-3-karboksamid |
| EP2379546A1 (en) * | 2008-12-19 | 2011-10-26 | Pfizer Inc. | Monocarbams |
| SG193156A1 (en) | 2009-03-20 | 2013-09-30 | Vertex Pharma | Process for making modulators of cystic fibrosis transmembrane conductance regulator |
| DK2493871T3 (da) | 2009-10-30 | 2014-11-10 | Prestwick Chemical Sas | Nye oximderivater samt deres anvendelse som allosteriske modulatorer af metabotropiske glutamatreceptorer |
| US8802700B2 (en) | 2010-12-10 | 2014-08-12 | Vertex Pharmaceuticals Incorporated | Modulators of ATP-Binding Cassette transporters |
| CN109966264A (zh) | 2012-02-27 | 2019-07-05 | 沃泰克斯药物股份有限公司 | 药物组合物及其施用 |
| RU2672569C2 (ru) | 2014-08-27 | 2018-11-16 | Прекстон Терапьютикс Са | Новое производное оксима хромона и его использование в качестве аллостерического модулятора метаботропных рецепторов глутамата |
| ES2702288T3 (es) | 2014-10-07 | 2019-02-28 | Vertex Pharma | Co-cristales de moduladores de regulador de conductancia transmembrana de la fibrosis quística |
| CN108349993A (zh) | 2015-08-27 | 2018-07-31 | 普雷克斯顿医疗股份公司 | 用于左旋多巴诱导的运动障碍疗法的脑-穿透剂色酮肟衍生物 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4587047A (en) * | 1981-04-09 | 1986-05-06 | E. R. Squibb & Sons, Inc. | 2-oxo-1-[[(substituted sulfonyl)amino]-carbonyl]azetidines |
| NZ199981A (en) * | 1981-04-09 | 1985-08-16 | Squibb & Sons Inc | 2-oxo-1-(((substituted sulphonyl)amino)carbonyl)azetidines |
| EG18314A (en) * | 1985-09-26 | 1993-02-28 | Squibb & Sons Inc | Process for preparing of 2-oxo-1((substituted sulfonyl)amino)carbonyl)-azitidines |
| EP0308416A1 (en) * | 1986-05-23 | 1989-03-29 | The Upjohn Company | N-1 substituted sulfonylaminocarbonyl, c-4 substituted monobactams |
| US4801705A (en) * | 1986-06-23 | 1989-01-31 | E. R. Squibb & Sons, Inc. | 2-oxo-1-(((substituted sulfonyl)amino)-carbonyl)azetidines |
-
1987
- 1987-08-13 US US07/085,050 patent/US4777252A/en not_active Expired - Fee Related
-
1988
- 1988-08-12 NZ NZ225821A patent/NZ225821A/en unknown
- 1988-08-12 AU AU20919/88A patent/AU2091988A/en not_active Abandoned
- 1988-08-12 JP JP63202599A patent/JPH0196181A/ja active Pending
- 1988-08-12 DK DK454188A patent/DK454188A/da not_active Application Discontinuation
- 1988-08-12 HU HU884349A patent/HU201547B/hu not_active IP Right Cessation
- 1988-08-12 ZA ZA885998A patent/ZA885998B/xx unknown
- 1988-08-12 EP EP88113156A patent/EP0303286A1/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| AU2091988A (en) | 1989-02-16 |
| EP0303286A1 (en) | 1989-02-15 |
| HUT48235A (en) | 1989-05-29 |
| JPH0196181A (ja) | 1989-04-14 |
| NZ225821A (en) | 1990-11-27 |
| HU201547B (en) | 1990-11-28 |
| ZA885998B (en) | 1989-04-26 |
| DK454188D0 (da) | 1988-08-12 |
| US4777252A (en) | 1988-10-11 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| AHB | Application shelved due to non-payment |