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Application filed by Hokuriku PharmaceuticalfiledCriticalHokuriku Pharmaceutical
Priority to DK43884ApriorityCriticalpatent/DK156832C/en
Publication of DK43884D0publicationCriticalpatent/DK43884D0/en
Publication of DK43884ApublicationCriticalpatent/DK43884A/en
Publication of DK156832BpublicationCriticalpatent/DK156832B/en
Application grantedgrantedCritical
Publication of DK156832CpublicationCriticalpatent/DK156832C/en
Pharmaceuticals Containing Other Organic And Inorganic Compounds
(AREA)
Pyrrole Compounds
(AREA)
Abstract
Novel 3-pyrrolidinepropiophenone derivatives of the formula: <IMAGE> in which R denotes an ethyl, propyl, isopropyl, butyl or isobutyl group or a cycloalkyl group having 5-7 carbon atoms, and pharmaceutically acceptable acid addition salts thereof, are prepared by reacting a propiophenone derivative of the formula: <IMAGE> in which R has the previously mentioned meaning, with a formaldehyde, or an equivalent thereto, and pyrrolidine, or a salt thereof. The novel compounds possess improved muscle-relaxing activity and greatly inhibit nicotine-induced convulsions and oxotremor-induced shivering. The compounds are of low toxicity.
DK43884A1984-01-311984-01-31
3-PYRROLIDINE PROPIOPHENON DERIVATIVES AND PHARMACEUTICAL PREPARATIONS CONTAINING THE SAME
DK156832C
(en)