DK431586D0 - Benzimidazolderivater, fremgangsmaade til fremstilling deraf og laegemiddel indeholdende disse - Google Patents

Benzimidazolderivater, fremgangsmaade til fremstilling deraf og laegemiddel indeholdende disse

Info

Publication number: DK431586D0
Authority: DK; Denmark
Prior art keywords: procedures; preparing; product containing; medicinal product; benzimidazold
Prior art date: 1985-09-11

Application number

DK431586A

Other languages

English (en)

Other versions

DK431586A (da

DK170594B1 (da

Inventor

Philippe Manoury

Jean Binet

Gerard Defosse

Original Assignee

Synthelabo

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1985-09-11

Filing date

1986-09-10

Publication date

1986-09-10

1986-09-10 Application filed by Synthelabo filed Critical Synthelabo

1986-09-10 Publication of DK431586D0 publication Critical patent/DK431586D0/da

1987-03-12 Publication of DK431586A publication Critical patent/DK431586A/da

1995-11-06 Application granted granted Critical

1995-11-06 Publication of DK170594B1 publication Critical patent/DK170594B1/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Pulmonology (AREA)
Immunology (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

DK431586A 1985-09-11 1986-09-10 Benzimidazol- og imidazoderivater, fremgangsmåde til fremstilling deraf, lægemiddel samt farmaceutisk præparat indeholdende disse DK170594B1 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR8513453A FR2587029B1 (fr)	1985-09-11	1985-09-11	Derives de benzimidazole, leur preparation et leur application en therapeutique
FR8513453		1985-09-11

Publications (3)

Publication Number	Publication Date
DK431586D0 true DK431586D0 (da)	1986-09-10
DK431586A DK431586A (da)	1987-03-12
DK170594B1 DK170594B1 (da)	1995-11-06

Family

ID=9322797

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK431586A DK170594B1 (da)	1985-09-11	1986-09-10	Benzimidazol- og imidazoderivater, fremgangsmåde til fremstilling deraf, lægemiddel samt farmaceutisk præparat indeholdende disse

Country Status (24)

Country	Link
US (2)	US4820710A (da)
EP (1)	EP0217700B1 (da)
JP (1)	JPS6261979A (da)
KR (1)	KR930001411B1 (da)
AR (1)	AR243187A1 (da)
AT (1)	ATE103603T1 (da)
AU (1)	AU582894B2 (da)
CA (1)	CA1272486A (da)
CS (1)	CS357991A3 (da)
DE (2)	DE3689748T2 (da)
DK (1)	DK170594B1 (da)
ES (1)	ES2001782A6 (da)
FI (1)	FI87210C (da)
FR (1)	FR2587029B1 (da)
GR (1)	GR862318B (da)
HU (1)	HU196597B (da)
IE (1)	IE61607B1 (da)
IL (1)	IL79992A (da)
LU (1)	LU90085I2 (da)
NL (1)	NL970029I2 (da)
NO (2)	NO167026C (da)
NZ (1)	NZ217537A (da)
PT (1)	PT83355B (da)
ZA (1)	ZA866901B (da)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2618435B1 (fr) *	1987-07-23	1989-10-27	Synthelabo	Derives de benzimidazole, leur preparation et leur application en therapeutique
FR2637595B1 (fr) *	1988-10-11	1990-11-30	Synthelabo	Derives de benzimidazole, leur preparation et leur application en therapeutique
JPH02294758A (ja) *	1989-05-09	1990-12-05	Nec Corp	計算機使用時間管理方式
FR2658823B1 (fr) *	1990-02-27	1992-04-30	Adir	Nouveaux derives d'aminomethylpiperidine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent .
FR2666582B1 (fr) *	1990-09-07	1994-09-02	Synthelabo	Derives de benzimidazole, leur preparation et leur application en therapeutique.
FR2693194B1 (fr) *	1992-07-03	1994-09-23	Synthelabo	Dérivés d'alcanecarboxamide, leur préparation et leur application thérapeutique.
FR2745500B1 (fr) *	1996-03-04	1998-04-03	Synthelabo	Formulations pharmaceutiques a liberation prolongee contenant de la mizolastine
JPH10101564A (ja) *	1996-09-27	1998-04-21	Mitsubishi Chem Corp	鼻炎予防及び／又は治療剤
ATE238998T1 (de)	1997-02-25	2003-05-15	Us Gov Health & Human Serv	Substituierte benzimidazole als nicht-nucleoside reverse transcriptase inhibitore
FR2762214B1 (fr) *	1997-04-17	2000-10-06	Synthelabo	Utilisation de la mizolastine pour la preparation d'un medicament destine au traitement de l'inflammation
EP0958820A1 (en) *	1998-05-19	1999-11-24	Sanofi-Synthelabo	Use of an imidazol derivative for the manufacture of a medicament for treating auto-immunodiseases
ES2208098B1 (es) *	2002-10-02	2005-10-16	Ragactives, S.L.	Procedimiento e intermedios para la obtencion de derivados de 1-(1h-bencimidazol-2-il)-4-(2-aminopirimidin) piperidina.
TW200526637A (en) *	2003-09-30	2005-08-16	Janssen Pharmaceutica Nv	Benzoimidazole compounds
ES2245227B1 (es) *	2004-04-06	2007-03-01	Ragactives, S.L.	Formas cristalinas de mizolastina, procedimientos para su obtencion y composiciones farmaceuticas que las contienen.
JP5732453B2 (ja) *	2009-06-25	2015-06-10	アルカーメスファーマアイルランドリミテッド	Ｎｈ酸性化合物のプロドラッグ
US8431576B2 (en)	2009-06-25	2013-04-30	Alkermes Pharma Ireland Limited	Heterocyclic compounds for the treatment of neurological and psychological disorders
CN102140076A (zh) *	2010-02-03	2011-08-03	辽宁本源制药有限公司	咪唑斯汀中间体的制备
AU2012351747B2 (en)	2011-12-15	2016-05-12	Alkermes Pharma Ireland Limited	Prodrugs of secondary amine compounds
CA3092335A1 (en)	2018-03-05	2019-09-12	Alkermes Pharma Ireland Limited	Aripiprazole dosing strategy
CN114096247B (zh) *	2019-04-11	2024-04-26	帝人制药株式会社	苯并咪唑衍生物及其用途
WO2023107705A1 (en)	2021-12-10	2023-06-15	Incyte Corporation	Bicyclic amines as cdk12 inhibitors
CN116655596A (zh) *	2022-02-17	2023-08-29	济南同路医药科技发展有限公司	一种大粒径咪唑斯汀原料药制备方法
CN119707917B (zh) *	2024-12-24	2025-12-09	沈阳三九药业有限公司	一种咪唑斯汀中间体的制备方法
CN120441547B (zh) *	2025-05-06	2026-01-27	大连医科大学附属第二医院	一种脂肪酸酰胺水解酶（faah）抑制剂及其在疾病治疗中的应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4281005A (en) *	1979-03-05	1981-07-28	Merck & Co., Inc.	Novel 2-pyridylimidazole compounds
US4556660A (en) *	1982-07-12	1985-12-03	Janssen Pharmaceutica N.V.	N-(Bicyclic heterocyclyl)-4-piperidinamines
DE3484096D1 (de) *	1983-11-30	1991-03-14	Janssen Pharmaceutica Nv	Bizyklisches heterozyklyl aufveisende n-(bizyklisches heterozyklyl-4-piperidinamine.
PH23995A (en) *	1984-01-09	1990-02-09	Janssen Pharmaceutica Nv	4((bicycle heterocyclyl)-methyl and hetero)piperidines
US4588722A (en) *	1984-01-09	1986-05-13	Janssen Pharmaceutica N.V.	N-(4-piperidinyl) bicyclic condensed 2-imidazolamine derivatives

1985
- 1985-09-11 FR FR8513453A patent/FR2587029B1/fr not_active Expired
1986
- 1986-09-02 AT AT86401928T patent/ATE103603T1/de active
- 1986-09-02 DE DE3689748T patent/DE3689748T2/de not_active Expired - Lifetime
- 1986-09-02 DE DE1997175081 patent/DE19775081I2/de active Active
- 1986-09-02 EP EP86401928A patent/EP0217700B1/fr not_active Expired - Lifetime
- 1986-09-09 IL IL79992A patent/IL79992A/xx not_active IP Right Cessation
- 1986-09-10 KR KR1019860007594A patent/KR930001411B1/ko not_active Expired - Lifetime
- 1986-09-10 GR GR862318A patent/GR862318B/el unknown
- 1986-09-10 NZ NZ217537A patent/NZ217537A/xx unknown
- 1986-09-10 NO NO863608A patent/NO167026C/no not_active IP Right Cessation
- 1986-09-10 ZA ZA866901A patent/ZA866901B/xx unknown
- 1986-09-10 HU HU863907A patent/HU196597B/hu unknown
- 1986-09-10 IE IE241686A patent/IE61607B1/en not_active IP Right Cessation
- 1986-09-10 ES ES8601773A patent/ES2001782A6/es not_active Expired
- 1986-09-10 DK DK431586A patent/DK170594B1/da not_active IP Right Cessation
- 1986-09-10 PT PT83355A patent/PT83355B/pt unknown
- 1986-09-10 CA CA000517916A patent/CA1272486A/en not_active Expired - Lifetime
- 1986-09-10 AR AR86305197A patent/AR243187A1/es active
- 1986-09-10 JP JP61214978A patent/JPS6261979A/ja active Granted
- 1986-09-10 US US06/906,279 patent/US4820710A/en not_active Expired - Lifetime
- 1986-09-10 AU AU62552/86A patent/AU582894B2/en not_active Expired
- 1986-09-10 FI FI863661A patent/FI87210C/fi not_active IP Right Cessation
1988
- 1988-12-12 US US07/283,468 patent/US4912219A/en not_active Expired - Lifetime
1991
- 1991-11-25 CS CS913579A patent/CS357991A3/cs unknown
1997
- 1997-07-25 NL NL970029C patent/NL970029I2/nl unknown
- 1997-07-30 LU LU90085C patent/LU90085I2/fr unknown
2001
- 2001-10-15 NO NO2001017C patent/NO2001017I1/no unknown

Also Published As

Publication number	Publication date
LU90085I2 (fr)	1997-09-25
US4820710A (en)	1989-04-11
AU6255286A (en)	1987-03-12
AR243187A1 (es)	1993-07-30
FI87210B (fi)	1992-08-31
PT83355A (fr)	1986-10-01
NO167026C (no)	1991-09-25
NO2001017I1 (no)	2001-11-05
NO863608D0 (no)	1986-09-10
HU196597B (en)	1988-12-28
NO863608L (no)	1987-03-12
CS357991A3 (en)	1992-06-17
GR862318B (en)	1987-01-19
ES2001782A6 (es)	1988-06-16
PT83355B (pt)	1989-05-12
ZA866901B (en)	1987-04-29
KR870003100A (ko)	1987-04-15
DE19775081I2 (de)	2002-08-29
IE61607B1 (en)	1994-11-16
NO167026B (no)	1991-06-17
US4912219A (en)	1990-03-27
NZ217537A (en)	1988-11-29
EP0217700B1 (fr)	1994-03-30
HUT41771A (en)	1987-05-28
IE862416L (en)	1987-03-11
HK1005592A1 (en)	1999-01-15
FR2587029A1 (fr)	1987-03-13
ATE103603T1 (de)	1994-04-15
CA1272486A (en)	1990-08-07
FI863661A0 (fi)	1986-09-10
DE3689748D1 (de)	1994-05-05
KR930001411B1 (ko)	1993-02-27
NL970029I1 (nl)	1997-10-01
FI87210C (fi)	1992-12-10
JPS6261979A (ja)	1987-03-18
IL79992A0 (en)	1986-12-31
FR2587029B1 (fr)	1987-10-30
DE3689748T2 (de)	1994-08-11
DK431586A (da)	1987-03-12
JPH0460596B2 (da)	1992-09-28
FI863661L (fi)	1987-03-12
DK170594B1 (da)	1995-11-06
AU582894B2 (en)	1989-04-13
IL79992A (en)	1990-07-12
EP0217700A1 (fr)	1987-04-08
NL970029I2 (nl)	1998-04-01

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Legal Events

Date	Code	Title	Description
1995-11-06	B1	Patent granted (law 1993)
1998-04-06	CTFF	Application for supplementary protection certificate (spc) filed	Free format text: CA 1997 00043, 971031
1998-05-25	CTFG	Supplementary protection certificate (spc) issued	Free format text: CA 1997 00043, 971031, EXPIRES: 20101121
2006-09-25	PUP	Patent expired