DK2519512T3 - N1-acyl-5-fluorpyrimidinonderivater - Google Patents

N1-acyl-5-fluorpyrimidinonderivater Download PDF

Info

Publication number: DK2519512T3
Authority: DK; Denmark
Prior art keywords: fluorpyrimidinonderivater; acyl
Prior art date: 2009-08-07

Application number

DK10807171.3T

Other languages

English (en)

Inventor

Timothy Boebel

Kristy Bryan

Beth Lorsbach

Timothy Martin

W Owen

Mark Pobanz

Scott Thornburgh

Jeffery Webster

Chenglin Yao

Original Assignee

Adama Makhteshim Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2009-08-07

Filing date

2010-08-05

Publication date

2019-05-27

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535292&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK2519512(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2010-08-05 Application filed by Adama Makhteshim Ltd filed Critical Adama Makhteshim Ltd

2019-05-27 Application granted granted Critical

2019-05-27 Publication of DK2519512T3 publication Critical patent/DK2519512T3/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Agronomy & Crop Science (AREA)
Pest Control & Pesticides (AREA)
Plant Pathology (AREA)
Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Dentistry (AREA)
General Health & Medical Sciences (AREA)
Wood Science & Technology (AREA)
Zoology (AREA)
Environmental Sciences (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Plural Heterocyclic Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

DK10807171.3T 2009-08-07 2010-08-05 N1-acyl-5-fluorpyrimidinonderivater DK2519512T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US23222309P	2009-08-07	2009-08-07
PCT/US2010/044576 WO2011017538A1 (en)	2009-08-07	2010-08-05	N1-acyl-5-fluoropyrimidinone derivatives

Publications (1)

Publication Number	Publication Date
DK2519512T3 true DK2519512T3 (da)	2019-05-27

Family

ID=43535292

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK10807171.3T DK2519512T3 (da)	2009-08-07	2010-08-05	N1-acyl-5-fluorpyrimidinonderivater

Country Status (34)

Country	Link
US (1)	US8470839B2 (da)
EP (1)	EP2519512B1 (da)
JP (1)	JP5748754B2 (da)
KR (1)	KR101792285B1 (da)
CN (1)	CN102548981B (da)
AU (1)	AU2010279402B2 (da)
BR (1)	BR112012002810B1 (da)
CA (1)	CA2768510C (da)
CL (1)	CL2012000316A1 (da)
CO (1)	CO6491117A2 (da)
CR (1)	CR20120030A (da)
CY (1)	CY1122115T1 (da)
DK (1)	DK2519512T3 (da)
EA (1)	EA023411B1 (da)
EC (1)	ECSP12011653A (da)
ES (1)	ES2728966T3 (da)
HK (1)	HK1172894A1 (da)
HN (1)	HN2012000269A (da)
HR (1)	HRP20190919T1 (da)
HU (1)	HUE045290T2 (da)
IL (1)	IL217952A (da)
IN (1)	IN2012DN00539A (da)
LT (1)	LT2519512T (da)
MX (1)	MX2012001620A (da)
NI (1)	NI201200022A (da)
NZ (1)	NZ597570A (da)
PE (1)	PE20120688A1 (da)
PL (1)	PL2519512T3 (da)
PT (1)	PT2519512T (da)
SI (1)	SI2519512T1 (da)
TR (1)	TR201908180T4 (da)
UA (1)	UA106889C2 (da)
WO (1)	WO2011017538A1 (da)
ZA (1)	ZA201200819B (da)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CN102574831B (zh) *	2009-08-07	2014-12-10	陶氏益农公司	N1-磺酰基-5-氟代嘧啶酮衍生物
UA113062C2 (xx) *	2011-08-17	2016-12-12		Похідні 5-фтор-4-іміно-3-(заміщеного)-3,4-дигідропіримідин-2(1h)ону
KR20150100869A (ko)	2012-12-28	2015-09-02	다우 아그로사이언시즈 엘엘씨	N-(치환된)-5-플루오로-4-이미노-3-메틸-2-옥소-3,4-디히드로피리미딘-1(2h)-카르복스아미드 유도체
CA2893778A1 (en)	2012-12-28	2014-07-03	Dow Agrosciences Llc	N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2h)-carboxylate derivatives
RU2656101C2 (ru) *	2012-12-28	2018-05-31	Адама Мактешим Лтд.	Производные 1-(замещенный бензоил)-5-фтор-4-имино-3-метил-3,4-дигидропиримидин-2(1h)-она
CN105007737A (zh)	2012-12-31	2015-10-28	美国陶氏益农公司	作为杀真菌剂的3-烷基-5-氟-4-取代的-亚氨基-3,4-二氢嘧啶-2(1h)-酮衍生物
AP2016009340A0 (en)	2013-12-31	2016-07-31	Adama Makhteshim Ltd	Synergistic fungicidal mixtures for fungal control in cereals
MX2016008759A (es)	2013-12-31	2017-05-09	Adama Makhteshim Ltd	5-fluor-4-imino-3-(alquil/alquilo sustituido)-1-(arilsulfonil)-3,4 -dihidropirimidin-2(1h)-ona y los procesos para su preparacion.
JP6734267B2 (ja)	2014-09-26	2020-08-05	ザケマーズカンパニーエフシーリミテッドライアビリティカンパニー	イソシアネート由来のオルガノシラン
CA3069619A1 (en)	2017-07-17	2019-02-28	Adama Makhteshim Ltd.	Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one

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CH421973A (de) *	1962-05-01	1966-10-15	Hoffmann La Roche	Verfahren zur Herstellung eines Cytosin-Derivates
US3309359A (en) *	1965-10-22	1967-03-14	Hoffmann La Roche	N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) *	1966-01-13	1968-02-13	Hoffmann La Roche	Controlling fungi with 5-fluorocytosine
US3868373A (en) *	1970-01-27	1975-02-25	Hoffmann La Roche	4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (da)	1973-09-07	1976-08-31	Hoffmann La Roche
FR2530636A1 (fr)	1982-07-23	1984-01-27	Rhone Poulenc Agrochimie	Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
EP0139613A1 (de)	1983-08-29	1985-05-02	Ciba-Geigy Ag	N-(2-Nitrophenyl)-4-aminopyrimidin-Derivate, deren Herstellung und Verwendung
US4845081A (en) *	1984-10-18	1989-07-04	University Of Florida	Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
ATE109776T1 (de)	1988-03-09	1994-08-15	Ciba Geigy Ag	Mittel zum schutz von pflanzen gegen krankheiten.
DE3821711A1 (de) *	1988-06-28	1990-02-08	Bayer Ag	Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3217191B2 (ja) *	1992-07-16	2001-10-09	ビーエーエスエフアクチェンゲゼルシャフト	ヘテロ芳香族化合物およびこれを含有する植物保護剤
ES2167586T3 (es) *	1995-07-05	2002-05-16	Du Pont	Pirimidinonas fungicidas.
EP0888359B1 (en) *	1996-03-11	2002-05-02	Syngenta Participations AG	Pyrimidin-4-one derivatives as pesticide
HRP970239B1 (en)	1997-05-09	2004-04-30	Inst Ru Er Bouekovic	Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) *	1998-11-06	2001-04-18		Novedosa pirimidin-4-enamina como fungicida.
US7914799B2 (en) *	2001-08-27	2011-03-29	Immunitor USA, Inc.	Anti-fungal composition
JPWO2005095419A1 (ja) *	2004-04-01	2008-02-21	武田薬品工業株式会社	チアゾロピリミジン誘導体
WO2008005303A2 (en) *	2006-06-30	2008-01-10	Janssen Pharmaceutica N.V.	Thiazolopyrimidine modulators of trpv1
ES2549046T3 (es) *	2008-01-22	2015-10-22	Dow Agrosciences, Llc	Derivados de N-ciano-4-amino-5-fluoro-pirimidina como fungicidas
RU2536492C2 (ru)	2008-08-01	2014-12-27	ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи	Применение 5-фторцитозина в качестве фунгицида
DK2389375T3 (da)	2009-01-23	2015-08-24	Euro Celtique Sa	Hydroxamsyrederivater
CN102574831B (zh) *	2009-08-07	2014-12-10	陶氏益农公司	N1-磺酰基-5-氟代嘧啶酮衍生物

2010
- 2010-05-08 UA UAA201202731A patent/UA106889C2/uk unknown
- 2010-08-05 EP EP10807171.3A patent/EP2519512B1/en active Active
- 2010-08-05 DK DK10807171.3T patent/DK2519512T3/da active
- 2010-08-05 KR KR1020127005927A patent/KR101792285B1/ko active IP Right Grant
- 2010-08-05 BR BR112012002810-3A patent/BR112012002810B1/pt active IP Right Grant
- 2010-08-05 PT PT10807171T patent/PT2519512T/pt unknown
- 2010-08-05 TR TR2019/08180T patent/TR201908180T4/tr unknown
- 2010-08-05 CN CN201080045370.7A patent/CN102548981B/zh active Active
- 2010-08-05 WO PCT/US2010/044576 patent/WO2011017538A1/en active Application Filing
- 2010-08-05 PE PE2012000169A patent/PE20120688A1/es not_active Application Discontinuation
- 2010-08-05 ES ES10807171T patent/ES2728966T3/es active Active
- 2010-08-05 PL PL10807171T patent/PL2519512T3/pl unknown
- 2010-08-05 MX MX2012001620A patent/MX2012001620A/es active IP Right Grant
- 2010-08-05 SI SI201031893T patent/SI2519512T1/sl unknown
- 2010-08-05 US US12/851,236 patent/US8470839B2/en active Active - Reinstated
- 2010-08-05 NZ NZ597570A patent/NZ597570A/en unknown
- 2010-08-05 IN IN539DEN2012 patent/IN2012DN00539A/en unknown
- 2010-08-05 HU HUE10807171A patent/HUE045290T2/hu unknown
- 2010-08-05 AU AU2010279402A patent/AU2010279402B2/en not_active Ceased
- 2010-08-05 CA CA2768510A patent/CA2768510C/en not_active Expired - Fee Related
- 2010-08-05 EA EA201270253A patent/EA023411B1/ru not_active IP Right Cessation
- 2010-08-05 LT LTEP10807171.3T patent/LT2519512T/lt unknown
- 2010-08-05 JP JP2012523950A patent/JP5748754B2/ja active Active
2012
- 2012-01-18 CR CR20120030A patent/CR20120030A/es unknown
- 2012-02-02 HN HN2012000269A patent/HN2012000269A/es unknown
- 2012-02-02 ZA ZA2012/00819A patent/ZA201200819B/en unknown
- 2012-02-03 NI NI201200022A patent/NI201200022A/es unknown
- 2012-02-05 IL IL217952A patent/IL217952A/en active IP Right Grant
- 2012-02-06 CO CO12019954A patent/CO6491117A2/es active IP Right Grant
- 2012-02-06 CL CL2012000316A patent/CL2012000316A1/es unknown
- 2012-02-07 EC ECSP12011653 patent/ECSP12011653A/es unknown
- 2012-12-31 HK HK12113559.2A patent/HK1172894A1/xx unknown
2019
- 2019-05-17 HR HRP20190919TT patent/HRP20190919T1/hr unknown
- 2019-06-06 CY CY20191100603T patent/CY1122115T1/el unknown

Also Published As

Publication number	Publication date
TR201908180T4 (tr)	2019-06-21
HUE045290T2 (hu)	2019-12-30
EA023411B1 (ru)	2016-06-30
JP2013501723A (ja)	2013-01-17
EP2519512B1 (en)	2019-03-20
MX2012001620A (es)	2012-04-11
HN2012000269A (es)	2015-04-27
ECSP12011653A (es)	2012-03-30
EA201270253A1 (ru)	2012-07-30
BR112012002810B1 (pt)	2018-12-11
ZA201200819B (en)	2013-05-29
IL217952A0 (en)	2012-03-29
NZ597570A (en)	2014-04-30
HK1172894A1 (en)	2013-05-03
EP2519512A1 (en)	2012-11-07
NI201200022A (es)	2012-05-22
CY1122115T1 (el)	2020-11-25
AU2010279402B2 (en)	2015-04-16
SI2519512T1 (sl)	2019-09-30
AU2010279402A1 (en)	2012-02-02
PT2519512T (pt)	2019-06-04
CL2012000316A1 (es)	2014-06-27
KR20120041786A (ko)	2012-05-02
IN2012DN00539A (da)	2015-06-12
JP5748754B2 (ja)	2015-07-15
PE20120688A1 (es)	2012-06-06
PL2519512T3 (pl)	2019-09-30
KR101792285B1 (ko)	2017-10-31
CN102548981A (zh)	2012-07-04
ES2728966T3 (es)	2019-10-29
EP2519512A4 (en)	2013-01-16
US20110034490A1 (en)	2011-02-10
CR20120030A (es)	2012-03-28
CA2768510C (en)	2018-05-15
IL217952A (en)	2017-11-30
LT2519512T (lt)	2019-07-25
CN102548981B (zh)	2015-05-13
HRP20190919T1 (hr)	2019-09-20
WO2011017538A1 (en)	2011-02-10
CA2768510A1 (en)	2011-02-10
CO6491117A2 (es)	2012-07-31
BR112012002810A2 (pt)	2015-09-15
US8470839B2 (en)	2013-06-25
UA106889C2 (uk)	2014-10-27

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