DK216685A - BETA-CARBOLIN-3-CARBOXYLIC ACID DERIVATIVES AND METHOD FOR PREPARING THE SAME - Google Patents
BETA-CARBOLIN-3-CARBOXYLIC ACID DERIVATIVES AND METHOD FOR PREPARING THE SAME Download PDFInfo
- Publication number
- DK216685A DK216685A DK216685A DK216685A DK216685A DK 216685 A DK216685 A DK 216685A DK 216685 A DK216685 A DK 216685A DK 216685 A DK216685 A DK 216685A DK 216685 A DK216685 A DK 216685A
- Authority
- DK
- Denmark
- Prior art keywords
- denotes
- carbolin
- beta
- alkyl
- preparing
- Prior art date
Links
- ARLVFKCLBYUINL-UHFFFAOYSA-N 9h-pyrido[3,4-b]indole-3-carboxylic acid Chemical class N1C2=CC=CC=C2C2=C1C=NC(C(=O)O)=C2 ARLVFKCLBYUINL-UHFFFAOYSA-N 0.000 title abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 3
- 239000001257 hydrogen Substances 0.000 abstract 3
- 125000004178 (C1-C4) alkyl group Chemical group 0.000 abstract 2
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 2
- 125000003253 isopropoxy group Chemical group [H]C([H])([H])C([H])(O*)C([H])([H])[H] 0.000 abstract 2
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 2
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 abstract 1
- 125000006272 (C3-C7) cycloalkyl group Chemical group 0.000 abstract 1
- -1 C4-7-alkylcycloalkyl Chemical group 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000000596 cyclohexenyl group Chemical group C1(=CCCCC1)* 0.000 abstract 1
- 125000005745 ethoxymethyl group Chemical group [H]C([H])([H])C([H])([H])OC([H])([H])* 0.000 abstract 1
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 abstract 1
- 150000002431 hydrogen Chemical class 0.000 abstract 1
- 125000004184 methoxymethyl group Chemical group [H]C([H])([H])OC([H])([H])* 0.000 abstract 1
- 125000002568 propynyl group Chemical group [*]C#CC([H])([H])[H] 0.000 abstract 1
- 230000000506 psychotropic effect Effects 0.000 abstract 1
Landscapes
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Novel β-carboline-3-carboxylic esters of the general formula I: <IMAGE> where R<4> denotes methyl, ethyl or methoxymethyl, R<5> denotes hydrogen, -OR<8> (where R<8> denotes C1-4- alkyl, C3-7-cycloalkyl, C4-7-alkylcycloalkyl, propynyl or cyclohexenyl) or -CH2-OR<9>, where R<9> denotes C1-4-alkyl, R<6> denotes hydrogen, -OR<10> (where R<10> denotes branched C1-4-alkyl or C3-6-cycloalkyl) or -CH2-OR<9>, where R<9> has the previously mentioned meaning, provided that R<5> and R<6> are not both hydrogen, that R<5> is not isopropoxy when R<4> denotes H, and that R<5> is not isopropoxy or ethoxymethyl when R<4> denotes methyl. The novel compounds, which exhibit surprising psychotropic properties, are prepared by means of analogy processes.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DK216685A DK151964C (en) | 1984-05-15 | 1985-05-15 | BETA-CARBOLIN-3-CARBOXYLIC ACID DERIVATIVES AND PROCEDURES FOR THE PREPARATION OF THE SAME AND PHARMACEUTICAL PREPARATIONS |
Applications Claiming Priority (6)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DK2401/84A DK240184D0 (en) | 1984-05-15 | 1984-05-15 | BETA-CARBOLINE-3-CARBOXYLIC ACID DERIVATIVES AND METHOD OF PREPARING THE SAME |
| DK240084 | 1984-05-15 | ||
| DK2400/84A DK240084D0 (en) | 1984-05-15 | 1984-05-15 | NEW BETA-CARBOLINE-3-OXADIAZOLYL DERIVATIVES |
| DK240184 | 1984-05-15 | ||
| DK216685 | 1985-05-15 | ||
| DK216685A DK151964C (en) | 1984-05-15 | 1985-05-15 | BETA-CARBOLIN-3-CARBOXYLIC ACID DERIVATIVES AND PROCEDURES FOR THE PREPARATION OF THE SAME AND PHARMACEUTICAL PREPARATIONS |
Publications (4)
| Publication Number | Publication Date |
|---|---|
| DK216685D0 DK216685D0 (en) | 1985-05-15 |
| DK216685A true DK216685A (en) | 1985-11-16 |
| DK151964B DK151964B (en) | 1988-01-18 |
| DK151964C DK151964C (en) | 1988-07-18 |
Family
ID=27221519
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK216685A DK151964C (en) | 1984-05-15 | 1985-05-15 | BETA-CARBOLIN-3-CARBOXYLIC ACID DERIVATIVES AND PROCEDURES FOR THE PREPARATION OF THE SAME AND PHARMACEUTICAL PREPARATIONS |
Country Status (1)
| Country | Link |
|---|---|
| DK (1) | DK151964C (en) |
-
1985
- 1985-05-15 DK DK216685A patent/DK151964C/en not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| DK216685D0 (en) | 1985-05-15 |
| DK151964C (en) | 1988-07-18 |
| DK151964B (en) | 1988-01-18 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PBP | Patent lapsed |