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DK188486A - Glycopeptid-derivater og fremgangsmaade til fremstilling deraf - Google Patents

Glycopeptid-derivater og fremgangsmaade til fremstilling deraf Download PDF

Info

Publication number
DK188486A
DK188486A DK188486A DK188486A DK188486A DK 188486 A DK188486 A DK 188486A DK 188486 A DK188486 A DK 188486A DK 188486 A DK188486 A DK 188486A DK 188486 A DK188486 A DK 188486A
Authority
DK
Denmark
Prior art keywords
procedures
preparing
glycopeptide derivatives
glycopeptide
derivatives
Prior art date
Application number
DK188486A
Other languages
English (en)
Other versions
DK188486D0 (da
Inventor
Ramakrishnan Nagarajan
Amelia Apolinaria Schabel
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of DK188486D0 publication Critical patent/DK188486D0/da
Publication of DK188486A publication Critical patent/DK188486A/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C07K9/006—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
    • C07K9/008—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C09—DYES; PAINTS; POLISHES; NATURAL RESINS; ADHESIVES; COMPOSITIONS NOT OTHERWISE PROVIDED FOR; APPLICATIONS OF MATERIALS NOT OTHERWISE PROVIDED FOR
    • C09K—MATERIALS FOR MISCELLANEOUS APPLICATIONS, NOT PROVIDED FOR ELSEWHERE
    • C09K9/00—Tenebrescent materials, i.e. materials for which the range of wavelengths for energy absorption is changed as a result of excitation by some form of energy

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Materials Engineering (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)

Description

hvori R, Rj. Rj. R3 og Rt| kan have an række forskellige betydninger, fremstilles ud fra et glycopeptid-antibio-ticum valgt blandt vancomycin, A515B8A. A515BBB, MM3A ag MM3B ved omsætning med et aldehyd eller en keton, eventuelt efterfulgt af en reduktion.
Forbindelserne (1) inhiberer væksten af en lang række bakterier, især gr em-pos iti ve bakterier.
DK188486A 1985-04-25 1986-04-24 Glycopeptid-derivater og fremgangsmaade til fremstilling deraf DK188486A (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US72673185A 1985-04-25 1985-04-25
US72673185 1985-04-25

Publications (2)

Publication Number Publication Date
DK188486D0 DK188486D0 (da) 1986-04-24
DK188486A true DK188486A (da) 1986-10-26

Family

ID=24919774

Family Applications (1)

Application Number Title Priority Date Filing Date
DK188486A DK188486A (da) 1985-04-25 1986-04-24 Glycopeptid-derivater og fremgangsmaade til fremstilling deraf

Country Status (15)

Country Link
EP (1) EP0201251A3 (da)
JP (1) JPS61251699A (da)
KR (1) KR870001282B1 (da)
CN (1) CN86103330A (da)
AU (1) AU587615B2 (da)
DK (1) DK188486A (da)
ES (1) ES8706725A1 (da)
GR (1) GR861071B (da)
HU (1) HU204854B (da)
IL (1) IL78597A0 (da)
NZ (1) NZ215947A (da)
PH (1) PH23900A (da)
PT (1) PT82445B (da)
SU (1) SU1586521A3 (da)
ZA (1) ZA863091B (da)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8701872D0 (en) * 1987-01-28 1987-03-04 Lepetit Spa N15-alkyl & n15,n15-dialkyl derivatives
US5071749A (en) * 1987-04-16 1991-12-10 Shionogi & Co., Ltd. Glycopetide antibiotic pa-45052-b
GB8711066D0 (en) * 1987-05-11 1987-06-17 Lepetit Spa Teicoplanin derivatives
GB8817053D0 (en) * 1988-07-18 1988-08-24 Lepetit Spa Process for preparing n15 n15-dialkyl derivatives of teicoplanin compounds
NZ270387A (en) * 1994-01-28 1996-11-26 Lilly Co Eli Glycopeptide antibiotic, its production and compositions thereof
US5840684A (en) * 1994-01-28 1998-11-24 Eli Lilly And Company Glycopeptide antibiotic derivatives
WO1997002288A1 (en) * 1995-07-05 1997-01-23 Gruppo Lepetit S.P.A. Purification of dalbaheptide antibiotics by isoelectric focusing
EP1276759B1 (en) 2000-05-02 2008-07-30 Theravance, Inc. Reductive alkylation process on glycopeptides
TWI312785B (en) 2001-08-24 2009-08-01 Theravance Inc Process for preparing vancomycin derivatives
TWI275594B (en) 2001-08-24 2007-03-11 Theravance Inc Process for preparing vancomycin phosphonate derivatives
MX2007006319A (es) 2004-11-29 2007-07-25 Univ Nagoya Nat Univ Corp Derivados de monomeros de glicopeptico antibioticos.
TW200808818A (en) 2006-05-26 2008-02-16 Shionogi & Co Glycopeptide antibiotic derivatives
BRPI0821947A2 (pt) 2007-12-26 2015-09-22 Shionogi & Co derivados de antibiótico de glicopetídeo glicosilatado
CA2954653C (en) * 2014-07-10 2023-01-24 The Scripps Research Institute N-(hydrophobe-substituted)vancosaminyl [.psi.[c(=nh)nh]tpg4]vancomycin and [.psi.[ch2nh]tpg4]vancomycin
CN105985412A (zh) * 2015-02-28 2016-10-05 爱斯医药科技(南京)有限公司 万古霉素衍生物、制备方法及其应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4462942A (en) * 1982-07-30 1984-07-31 Eli Lilly And Company A47934 Antibiotic and process for production thereof
ZA839269B (en) * 1982-12-20 1985-07-31 Lilly Co Eli Antibiotic a51568 factors a and b
DE3572178D1 (en) * 1984-04-16 1989-09-14 Lilly Co Eli Improvements in and relating to antibiotics m43a, m43b, m43c and m43d

Also Published As

Publication number Publication date
SU1586521A3 (ru) 1990-08-15
AU5659886A (en) 1986-10-30
ES8706725A1 (es) 1987-07-01
EP0201251A2 (en) 1986-11-12
HU204854B (en) 1992-02-28
JPS61251699A (ja) 1986-11-08
CN86103330A (zh) 1986-10-29
GR861071B (en) 1986-08-21
PT82445B (pt) 1988-11-30
AU587615B2 (en) 1989-08-24
KR860008210A (ko) 1986-11-14
NZ215947A (en) 1988-10-28
HUT40683A (en) 1987-01-28
IL78597A0 (en) 1986-08-31
PH23900A (en) 1989-12-18
KR870001282B1 (ko) 1987-06-30
DK188486D0 (da) 1986-04-24
ZA863091B (en) 1987-12-30
ES554286A0 (es) 1987-07-01
EP0201251A3 (en) 1987-12-16
PT82445A (en) 1986-05-01

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