DK159853C - Analogifremgangsmaade til fremstilling af 9-dihydro-11,12-o-isopropyliden-erythromycin a eller -4ae-epi-erythromycin a eller 2'-o-acylater deraf eller farmaceutisk acceptable syreadditionssalte deraf - Google Patents

Analogifremgangsmaade til fremstilling af 9-dihydro-11,12-o-isopropyliden-erythromycin a eller -4ae-epi-erythromycin a eller 2'-o-acylater deraf eller farmaceutisk acceptable syreadditionssalte deraf

Info

Publication number: DK159853C
Authority: DK; Denmark
Prior art keywords: acceptable; erythromycin; isopropylide; acylates; epi
Prior art date: 1982-03-01

Application number

DK096983A

Other languages

English (en)

Other versions

DK96983D0 (da

DK96983A (da

DK159853B (da

Inventor

James Robert Hauske

Frank Christian Sciavolino

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1982-03-01

Filing date

1983-02-28

Publication date

1991-05-13

1983-02-28 Application filed by Pfizer filed Critical Pfizer

1983-02-28 Publication of DK96983D0 publication Critical patent/DK96983D0/da

1983-09-02 Publication of DK96983A publication Critical patent/DK96983A/da

1990-12-17 Publication of DK159853B publication Critical patent/DK159853B/da

1991-05-13 Application granted granted Critical

1991-05-13 Publication of DK159853C publication Critical patent/DK159853C/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Biochemistry (AREA)
Biotechnology (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Saccharide Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

DK096983A 1982-03-01 1983-02-28 Analogifremgangsmaade til fremstilling af 9-dihydro-11,12-o-isopropyliden-erythromycin a eller -4ae-epi-erythromycin a eller 2'-o-acylater deraf eller farmaceutisk acceptable syreadditionssalte deraf DK159853C (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US35354882		1982-03-01
US06/353,548 US4382086A (en)	1982-03-01	1982-03-01	9-Dihydro-11,12-ketal derivatives of erythromycin A and epi-erythromycin A

Publications (4)

Publication Number	Publication Date
DK96983D0 DK96983D0 (da)	1983-02-28
DK96983A DK96983A (da)	1983-09-02
DK159853B DK159853B (da)	1990-12-17
DK159853C true DK159853C (da)	1991-05-13

Family

ID=23389607

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK096983A DK159853C (da)	1982-03-01	1983-02-28	Analogifremgangsmaade til fremstilling af 9-dihydro-11,12-o-isopropyliden-erythromycin a eller -4ae-epi-erythromycin a eller 2'-o-acylater deraf eller farmaceutisk acceptable syreadditionssalte deraf

Country Status (8)

Country	Link
US (1)	US4382086A (da)
EP (1)	EP0087916B1 (da)
JP (1)	JPS58159500A (da)
DE (1)	DE3361453D1 (da)
DK (1)	DK159853C (da)
GR (1)	GR77921B (da)
IE (1)	IE54431B1 (da)
YU (1)	YU42841B (da)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB8421429D0 (en) *	1984-08-23	1984-09-26	Beecham Group Plc	Chemical compounds
EP0184921A3 (en) *	1984-12-08	1986-10-29	Beecham Group Plc	Erythromycin derivatives
EP0201166B1 (en)	1985-03-12	1990-02-07	Beecham Group Plc	Erythromycin derivatives
US4640910A (en) *	1985-11-12	1987-02-03	Abbott Laboratories	Erythromycin A silylated compounds and method of use
US4681872A (en) *	1985-11-12	1987-07-21	Abbott Laboratories	Erythromycin A 11,12-carbonate and method of use
KR930702369A (ko) *	1990-10-15	1993-09-08	우에노 아키라	에리쓰로마이신 또는 그의 유도체의 2'위치 수식 화합물
US20050171342A1 (en) *	2002-02-15	2005-08-04	Michael Burnet	Conjugates of biologically active compounds, methods for their preparation and use, formulation and pharmaceutical applications thereof
WO2003070173A2 (en)	2002-02-15	2003-08-28	Sympore Gmbh	Conjugates of biologically active compounds, methods for their preparation and use, formulation and pharmaceutical applications thereof
AU2003211113B2 (en) *	2002-02-15	2007-08-09	Merckle Gmbh	Antibiotic conjugates
US6946482B2 (en) *	2002-08-29	2005-09-20	Kosan Biosciences, Inc.	Motilide compounds
US7211568B2 (en) *	2003-12-18	2007-05-01	Kosan Biosciences Incorporated	9-Desoxoerythromycin compounds as prokinetic agents
EP1907392A1 (en) *	2005-07-26	2008-04-09	Merckle Gmbh	Macrolide conjugates of pyrrolizine and indolizine compounds as inhibitors of 5-lipooxygenase and cyclooxygenase

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US2653899A (en) *	1952-04-14	1953-09-29	Lilly Co Eli	Erythromycin, its salts, and method of preparation
US3417077A (en) *	1966-05-16	1968-12-17	Lilly Co Eli	Erythromycin derivative and process for the preparation thereof
US3884903A (en) *	1973-06-21	1975-05-20	Abbott Lab	4{41 -Deoxy-4{41 -oxoerythromycin B derivatives
US3884904A (en) *	1973-06-21	1975-05-20	Abbott Lab	11-Substituted erythromycin B derivatives
US4150220A (en) *	1977-02-04	1979-04-17	Pfizer Inc.	Semi-synthetic 4"-erythromycin A derivatives

1982
- 1982-03-01 US US06/353,548 patent/US4382086A/en not_active Expired - Lifetime
1983
- 1983-02-23 EP EP83300937A patent/EP0087916B1/en not_active Expired
- 1983-02-23 GR GR70583A patent/GR77921B/el unknown
- 1983-02-23 DE DE8383300937T patent/DE3361453D1/de not_active Expired
- 1983-02-25 YU YU459/83A patent/YU42841B/xx unknown
- 1983-02-28 DK DK096983A patent/DK159853C/da not_active IP Right Cessation
- 1983-02-28 IE IE410/83A patent/IE54431B1/en not_active IP Right Cessation
- 1983-03-01 JP JP58033682A patent/JPS58159500A/ja active Granted

Also Published As

Publication number	Publication date
EP0087916A1 (en)	1983-09-07
YU42841B (en)	1988-12-31
EP0087916B1 (en)	1985-12-11
YU45983A (en)	1986-02-28
US4382086A (en)	1983-05-03
DK96983D0 (da)	1983-02-28
JPS58159500A (ja)	1983-09-21
DK96983A (da)	1983-09-02
JPH0142275B2 (da)	1989-09-11
IE54431B1 (en)	1989-10-11
GR77921B (da)	1984-09-25
DE3361453D1 (en)	1986-01-23
DK159853B (da)	1990-12-17
IE830410L (en)	1983-09-01

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Legal Events

Date	Code	Title	Description
2003-03-17	PUP	Patent expired