DK1385515T3 - Spiropyrazole forbindelser - Google Patents

Spiropyrazole forbindelser

Info

Publication number: DK1385515T3
Authority: DK; Denmark
Prior art keywords: spiropyrazole; compounds; spiropyrazole compounds; whereinz; compound
Prior art date: 2001-04-18

Application number

DK02739163T

Other languages

English (en)

Inventor

Gary Lee

R Richard Goehring

Donald Kyle

Parviz Gharagozloo

Sam Victory

Original Assignee

Euro Celtique Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-04-18

Filing date

2002-04-18

Publication date

2008-10-27

2002-04-18 Application filed by Euro Celtique Sa filed Critical Euro Celtique Sa

2008-10-27 Application granted granted Critical

2008-10-27 Publication of DK1385515T3 publication Critical patent/DK1385515T3/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/10—Spiro-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Pain & Pain Management (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Rheumatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Dental Preparations (AREA)
Solid-Sorbent Or Filter-Aiding Compositions (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

DK02739163T 2001-04-18 2002-04-18 Spiropyrazole forbindelser DK1385515T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US28467501P	2001-04-18	2001-04-18
PCT/US2002/012376 WO2002085355A1 (en)	2001-04-18	2002-04-18	Spiropyrazole compounds

Publications (1)

Publication Number	Publication Date
DK1385515T3 true DK1385515T3 (da)	2008-10-27

Family

ID=23091099

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK02739163T DK1385515T3 (da)	2001-04-18	2002-04-18	Spiropyrazole forbindelser

Country Status (28)

Country	Link
US (2)	US6635653B2 (da)
EP (1)	EP1385515B1 (da)
JP (1)	JP4342181B2 (da)
KR (1)	KR100628292B1 (da)
CN (1)	CN1516584A (da)
AT (1)	ATE403429T1 (da)
AU (1)	AU2002311833B2 (da)
BR (1)	BR0209127A (da)
CA (1)	CA2444634C (da)
CY (1)	CY1108454T1 (da)
CZ (1)	CZ20032849A3 (da)
DE (1)	DE60228071D1 (da)
DK (1)	DK1385515T3 (da)
ES (1)	ES2312584T3 (da)
HK (1)	HK1062885A1 (da)
HU (1)	HUP0401333A3 (da)
IL (2)	IL158485A0 (da)
MX (1)	MXPA03009604A (da)
NO (1)	NO20034660L (da)
NZ (1)	NZ528978A (da)
PL (1)	PL367263A1 (da)
PT (1)	PT1385515E (da)
RU (1)	RU2299883C2 (da)
SI (1)	SI1385515T1 (da)
UA (1)	UA74439C2 (da)
WO (1)	WO2002085355A1 (da)
YU (1)	YU82403A (da)
ZA (1)	ZA200308103B (da)

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JP5727139B2 (ja)	2006-11-28	2015-06-03	ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプＪａｎｓｓｅｎＰｈａｒｍａｃｅｕｔｉｃａＮａａｍｌｏｚｅＶｅｎｎｏｏｔｓｃｈａｐ	３−（３−アミノ−２−（ｒ）−ヒドロキシ−プロピル）−１−（４−フルオロ−フェニル）−８−（８−メチル−ナフタレン−１−イルメチル）−１，３，８−トリアザ−スピロ［４．５］デカン−４−オンの塩
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MX2010002449A (es)	2007-08-31	2010-09-07	Purdue Pharma Lp	Compuestos de piperidina tipo quinoxalina sustituida y uso de los mismsos.
ES2393849T7 (es)	2008-07-21	2015-01-28	Purdue Pharma Lp	Compuestos de piperidina puenteada, de tipo quinoxalina sustituida, y usos de los mismos
UA107943C2 (xx) *	2009-11-16	2015-03-10	Lilly Co Eli	Сполуки спіропіперидину як антагоністи рецептора orl-1
ES2613631T3 (es)	2010-12-22	2017-05-25	Purdue Pharma L.P.	Compuestos de piperidina de tipo quinoxalina sustituidos con fósforo y usos de los mismos
US9290488B2 (en)	2011-12-01	2016-03-22	Purdue Pharma L.P.	Azetidine-substituted quinoxalines as opioid receptor like-1 modulators
US9085561B2 (en)	2012-07-30	2015-07-21	Purdue Pharma L.P.	Cyclic urea- or lactam-substituted quinoxaline-type piperidines as ORL-1 modulators
WO2014102589A1 (en)	2012-12-27	2014-07-03	Purdue Pharma L.P.	Quinazolin-4(3h)-one-type piperidine compounds and uses thereof
US9090618B2 (en)	2012-12-27	2015-07-28	Purdue Pharma L.P.	Substituted benzimidazole-type piperidine compounds and uses thereof
WO2014102592A2 (en)	2012-12-27	2014-07-03	Purdue Pharma L.P.	Oxime/substituted quinoxaline-type piperidine compounds and uses thereof
US10118927B2 (en)	2012-12-27	2018-11-06	Purdue Pharma L.P.	Substituted piperidin-4-amino-type compounds and uses thereof
WO2014102588A2 (en)	2012-12-27	2014-07-03	Purdue Pharma L.P.	Indole and indoline-type piperidine compounds and uses thereof
KR20240115925A (ko)	2016-07-29	2024-07-26	얀센 파마슈티카 엔브이	전립선암의 치료 방법
CN111825681A (zh) *	2020-07-07	2020-10-27	扬州大学	一种合成(e)-亚苄基螺吡唑吡咯嗪酮类化合物的方法

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SI1385515T1 (sl) *	2001-04-18	2008-12-31	Euro Celtique Sa	Spiropirazolne spojine

2002
- 2002-04-18 SI SI200230748T patent/SI1385515T1/sl unknown
- 2002-04-18 WO PCT/US2002/012376 patent/WO2002085355A1/en not_active Application Discontinuation
- 2002-04-18 PL PL02367263A patent/PL367263A1/xx not_active Application Discontinuation
- 2002-04-18 MX MXPA03009604A patent/MXPA03009604A/es active IP Right Grant
- 2002-04-18 CA CA2444634A patent/CA2444634C/en not_active Expired - Fee Related
- 2002-04-18 NZ NZ528978A patent/NZ528978A/en not_active IP Right Cessation
- 2002-04-18 ES ES02739163T patent/ES2312584T3/es not_active Expired - Lifetime
- 2002-04-18 BR BRPI0209127-5A patent/BR0209127A/pt not_active Application Discontinuation
- 2002-04-18 JP JP2002582928A patent/JP4342181B2/ja not_active Expired - Fee Related
- 2002-04-18 DK DK02739163T patent/DK1385515T3/da active
- 2002-04-18 YU YU82403A patent/YU82403A/sh unknown
- 2002-04-18 AU AU2002311833A patent/AU2002311833B2/en not_active Ceased
- 2002-04-18 HU HU0401333A patent/HUP0401333A3/hu unknown
- 2002-04-18 US US10/126,506 patent/US6635653B2/en not_active Expired - Lifetime
- 2002-04-18 EP EP02739163A patent/EP1385515B1/en not_active Expired - Lifetime
- 2002-04-18 DE DE60228071T patent/DE60228071D1/de not_active Expired - Lifetime
- 2002-04-18 CZ CZ20032849A patent/CZ20032849A3/cs unknown
- 2002-04-18 CN CNA028121767A patent/CN1516584A/zh active Pending
- 2002-04-18 UA UA20031110381A patent/UA74439C2/uk unknown
- 2002-04-18 KR KR1020037013821A patent/KR100628292B1/ko not_active IP Right Cessation
- 2002-04-18 RU RU2003133455/04A patent/RU2299883C2/ru not_active IP Right Cessation
- 2002-04-18 PT PT02739163T patent/PT1385515E/pt unknown
- 2002-04-18 IL IL15848502A patent/IL158485A0/xx unknown
- 2002-04-18 AT AT02739163T patent/ATE403429T1/de active
2003
- 2003-06-19 US US10/601,174 patent/US20040087641A1/en not_active Abandoned
- 2003-10-17 NO NO20034660A patent/NO20034660L/no not_active Application Discontinuation
- 2003-10-17 ZA ZA200308103A patent/ZA200308103B/en unknown
- 2003-10-19 IL IL158485A patent/IL158485A/en not_active IP Right Cessation
2004
- 2004-08-03 HK HK04105726.6A patent/HK1062885A1/xx not_active IP Right Cessation
2008
- 2008-10-27 CY CY20081101206T patent/CY1108454T1/el unknown

Also Published As

Publication number	Publication date
PT1385515E (pt)	2008-09-15
CY1108454T1 (el)	2014-04-09
US6635653B2 (en)	2003-10-21
SI1385515T1 (sl)	2008-12-31
UA74439C2 (uk)	2005-12-15
US20040087641A1 (en)	2004-05-06
ATE403429T1 (de)	2008-08-15
MXPA03009604A (es)	2004-04-02
RU2299883C2 (ru)	2007-05-27
IL158485A0 (en)	2004-05-12
ZA200308103B (en)	2004-10-18
CA2444634C (en)	2011-06-07
NO20034660L (no)	2003-12-17
KR100628292B1 (ko)	2006-09-27
CN1516584A (zh)	2004-07-28
CA2444634A1 (en)	2002-10-31
HUP0401333A2 (hu)	2004-10-28
IL158485A (en)	2009-09-01
YU82403A (sh)	2006-08-17
JP2004531531A (ja)	2004-10-14
NZ528978A (en)	2004-06-25
EP1385515B1 (en)	2008-08-06
EP1385515A1 (en)	2004-02-04
RU2003133455A (ru)	2005-05-10
BR0209127A (pt)	2006-03-21
KR20040008159A (ko)	2004-01-28
HUP0401333A3 (en)	2004-11-29
WO2002085355A1 (en)	2002-10-31
NO20034660D0 (no)	2003-10-17
PL367263A1 (en)	2005-02-21
ES2312584T3 (es)	2009-03-01
EP1385515A4 (en)	2004-06-30
DE60228071D1 (de)	2008-09-18
US20030027834A1 (en)	2003-02-06
HK1062885A1 (en)	2004-12-03
AU2002311833B2 (en)	2005-04-28
CZ20032849A3 (en)	2004-03-17
JP4342181B2 (ja)	2009-10-14

Publication	Publication Date	Title
DK1385515T3 (da)	2008-10-27	Spiropyrazole forbindelser
RS51444B (sr)	2011-04-30	JEDINJENJA KOJA SADRŽE LAKTAM I NJIHOVI DERIVATI KAO INHIBITORI FAKTORA Xa
DE60214392D1 (de)	2006-10-12	1,4-disubstituierte benzokondensierte cycloalkyl harnstoffverbindungen
CY1113578T1 (el)	2016-06-22	2,3-διυδρο-6-νιτροϊμιδαζο 2,1 -b-οξαζολια
DK1385514T3 (da)	2009-01-19	Spiroinden- og spiroindanforbindelser
YU82303A (sh)	2006-03-03	Analozi nociceptina
CY1106247T1 (el)	2011-06-08	Θειοφαινο- και θειαζολοσουλφοναμιδες ως αντινεοπλαστικοι παραγοντες
WO2003006425A3 (en)	2003-11-27	Novel compounds as anti-inflammatory, immunomodulatory and anti-proliferatory agents
SE0004245D0 (sv)	2000-11-20	Novel compounds and their use
DK1385518T3 (da)	2008-10-27	Benzimidazolon-forbindelser
DK1531672T3 (da)	2011-08-29	Antimikrobielle sammensætninger
MXPA03009602A (es)	2004-04-02	Analogos de nociceptina.
SE0103710D0 (sv)	2001-11-07	Compounds
SV2003000981A (es)	2003-07-29	Fenil-heterociclil-eteres ref. pcs10973
DE60232289D1 (de)	2009-06-25	Photopolymerisierbare Verbindungen
TR199901017A2 (xx)	1999-12-21	B�cek ilac� terkibi.
DK1347984T3 (da)	2005-01-10	Fremgangsmåde til fremstilling af taxanderivater
ATE254099T1 (de)	2003-11-15	Trimethyldecen-verbindungen
SE9901062D0 (sv)	1999-03-23	Use for conifer sapling protection
SE0402734D0 (sv)	2004-11-10	Antimiicrobial compounds
ATE470655T1 (de)	2010-06-15	Substituierte 1,5-diaminopentan-3-ol-verbindungen