DK1313740T3 - Prodrugs af imidazopyridinderivater - Google Patents
Prodrugs af imidazopyridinderivaterInfo
- Publication number
- DK1313740T3 DK1313740T3 DK01933769T DK01933769T DK1313740T3 DK 1313740 T3 DK1313740 T3 DK 1313740T3 DK 01933769 T DK01933769 T DK 01933769T DK 01933769 T DK01933769 T DK 01933769T DK 1313740 T3 DK1313740 T3 DK 1313740T3
- Authority
- DK
- Denmark
- Prior art keywords
- prodrugs
- imidazopyridine derivatives
- imidazopyridine
- derivatives
- substituents
- Prior art date
Links
- 125000004857 imidazopyridinyl group Chemical class N1C(=NC2=C1C=CC=N2)* 0.000 title 1
- 229940002612 prodrug Drugs 0.000 title 1
- 239000000651 prodrug Substances 0.000 title 1
- 208000018522 Gastrointestinal disease Diseases 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
- C07D491/14—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/07—Optical isomers
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP00106695 | 2000-03-29 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK1313740T3 true DK1313740T3 (da) | 2006-04-03 |
Family
ID=8168271
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK01933769T DK1313740T3 (da) | 2000-03-29 | 2001-03-28 | Prodrugs af imidazopyridinderivater |
Country Status (25)
| Country | Link |
|---|---|
| US (2) | US20030125327A1 (da) |
| EP (1) | EP1313740B1 (da) |
| JP (1) | JP2003528878A (da) |
| KR (1) | KR100860627B1 (da) |
| CN (1) | CN1214030C (da) |
| AT (1) | ATE311389T1 (da) |
| AU (1) | AU783633B2 (da) |
| BR (1) | BR0109483A (da) |
| CA (1) | CA2404474A1 (da) |
| CZ (1) | CZ20023194A3 (da) |
| DE (1) | DE60115466T2 (da) |
| DK (1) | DK1313740T3 (da) |
| EA (1) | EA005597B1 (da) |
| ES (1) | ES2253376T3 (da) |
| HR (1) | HRP20020854A2 (da) |
| HU (1) | HUP0302331A2 (da) |
| IL (2) | IL151200A0 (da) |
| MX (1) | MXPA02009551A (da) |
| NO (1) | NO20024662L (da) |
| NZ (1) | NZ520837A (da) |
| PL (1) | PL365116A1 (da) |
| SI (1) | SI1313740T1 (da) |
| SK (1) | SK286850B6 (da) |
| WO (1) | WO2001072756A1 (da) |
| ZA (1) | ZA200207637B (da) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BR0109542A (pt) * | 2000-03-29 | 2003-06-10 | Altana Pharma Ag | Derivados de imidazopirina alquilados |
| MXPA03003706A (es) | 2000-10-25 | 2005-01-25 | Altana Pharma Ag | Imidazopiridinas polisustituidas, como inhibidores de secrecion gastrica. |
| US20050020637A1 (en) * | 2001-11-19 | 2005-01-27 | Wolfgang-Alexander Simon | Agents for the treatment of airway disorders |
| AU2003206879A1 (en) | 2002-02-15 | 2003-09-04 | Altana Pharma Ag | Tricyclic n-acyl compounds |
| TWI295575B (en) * | 2002-04-24 | 2008-04-11 | Altana Pharma Ag | Nitrosated imidazopyridines |
| RS95304A (sr) * | 2002-05-07 | 2006-12-15 | Altana Pharma Ag. | Nova kombinacija za tretman oboljenja disajnih puteva |
| RS20050377A (sr) | 2002-11-19 | 2007-11-15 | Altana Pharma Ag., | 8-supstituisani imidazopiridini |
| RS20050449A (sr) * | 2002-12-20 | 2007-11-15 | Altana Pharma Ag., | 8-trialkisiloksi-2-metil-9-fenil-7- okso-7,8,9,10- tetrahidroimidazo /1,2h//1,7/naftiridini |
| HRP20050790A2 (en) * | 2003-02-17 | 2006-12-31 | Altana Pharma Ag | New combinations and new use of selected pharmaceutically active compounds |
| AR044129A1 (es) | 2003-05-06 | 2005-08-24 | Altana Pharma Ag | Compuestos intermedios de imidazopiridina. proceso de preparacion. |
| SA04250092B1 (ar) * | 2003-05-14 | 2008-05-04 | التانا فاروا ايه جي | مركب وسيط جديد لتحضير مركبات إيميدازوبيريدين imidazopyridines فعالة علاجياً |
| RS20050868A (sr) * | 2003-05-27 | 2007-08-03 | Altana Pharma Ag., | Farmaceutske kombinacije inhibotora protonske pumpe i jedinjenje koje modifikuje gastrointestinalni motilitet |
| US20080280944A1 (en) | 2003-11-03 | 2008-11-13 | Paula Fernstrom | Imidazo[1,2-A]Pyridine Derivatives For The Treatment Of Silent Gastro-Esophageal Reflux |
| AR046893A1 (es) * | 2003-12-16 | 2005-12-28 | Altana Pharma Ag | Bencimidazoles triciclicos |
| WO2005058894A1 (en) | 2003-12-19 | 2005-06-30 | Altana Pharma Ag | Intermediates for the preparation of tricyclic dihydropyrano -imidazo -pyridines derivatives |
| CN101027277A (zh) * | 2004-07-23 | 2007-08-29 | 帝斯曼知识产权资产管理有限公司 | (2r,3r)-2-羟基-3-氨基-3-芳基-丙酰胺和(2r,3r)-2-羟基-3-氨基-3-芳基-丙酸烷基酯的制备方法 |
| CA2582256A1 (en) * | 2004-10-01 | 2006-04-13 | Altana Pharma Ag | Substituted tricyclic benzimidazoles |
| RU2586276C2 (ru) | 2009-07-09 | 2016-06-10 | Раквалиа Фарма Инк. | Антагонист кислотного насоса для лечения заболеваний, связанных с патологическим нарушением моторики желудочно-кишечного тракта |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4468400A (en) * | 1982-12-20 | 1984-08-28 | Schering Corporation | Antiulcer tricyclic imidazo [1,2-a]pyridines |
| US4673679A (en) * | 1986-05-14 | 1987-06-16 | E. I. Du Pont De Nemours And Company | Use of prodrugs of 3-hydroxymorphinans to prevent bitter taste upon buccal, nasal or sublingual administration |
| JPH06502659A (ja) * | 1991-05-31 | 1994-03-24 | ファイザー インク | 免疫抑制剤としてのラパマイシンプロドラッグの使用 |
| DE4308095A1 (de) * | 1993-03-13 | 1994-09-15 | Hoechst Ag | Prodrug-Derivate von Arzneimittelwirkstoffen mit Hydroxylgruppen, Verfahren zu deren Herstellung und ihre Verwendung |
| SE9401197D0 (sv) * | 1994-04-11 | 1994-04-11 | Astra Ab | Active compounds |
| US6073004A (en) | 1996-12-17 | 2000-06-06 | Ericsson Inc. | Emergency call initiator |
| ES2219890T3 (es) * | 1997-03-24 | 2004-12-01 | Altana Pharma Ag | Compuestos tetrahidropirido. |
| WO1998042707A1 (en) * | 1997-03-24 | 1998-10-01 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Tetrahydropyrido compounds |
| JP2001526703A (ja) * | 1997-05-28 | 2001-12-18 | ビイク グルデン ロンベルク ヒエーミツシエ フアブリーク ゲゼルシヤフト ミツト ベシユレンクテル ハフツング | 縮合ジヒドロピラン |
| PT1115725E (pt) * | 1998-09-23 | 2003-06-30 | Altana Pharma Ag | Tetra-hidropiridoeteres |
| WO2000026217A1 (en) * | 1998-11-03 | 2000-05-11 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Imidazonaphthyridines |
| BR0109542A (pt) | 2000-03-29 | 2003-06-10 | Altana Pharma Ag | Derivados de imidazopirina alquilados |
-
2001
- 2001-03-28 AT AT01933769T patent/ATE311389T1/de not_active IP Right Cessation
- 2001-03-28 DE DE60115466T patent/DE60115466T2/de not_active Expired - Fee Related
- 2001-03-28 AU AU60166/01A patent/AU783633B2/en not_active Ceased
- 2001-03-28 SI SI200130498T patent/SI1313740T1/sl unknown
- 2001-03-28 US US10/182,619 patent/US20030125327A1/en not_active Abandoned
- 2001-03-28 NZ NZ520837A patent/NZ520837A/en unknown
- 2001-03-28 EA EA200200875A patent/EA005597B1/ru not_active IP Right Cessation
- 2001-03-28 WO PCT/EP2001/003514 patent/WO2001072756A1/en not_active Ceased
- 2001-03-28 HU HU0302331A patent/HUP0302331A2/hu unknown
- 2001-03-28 EP EP01933769A patent/EP1313740B1/en not_active Expired - Lifetime
- 2001-03-28 HR HRP20020854 patent/HRP20020854A2/hr not_active Application Discontinuation
- 2001-03-28 JP JP2001570665A patent/JP2003528878A/ja not_active Withdrawn
- 2001-03-28 IL IL15120001A patent/IL151200A0/xx unknown
- 2001-03-28 PL PL01365116A patent/PL365116A1/xx not_active Application Discontinuation
- 2001-03-28 DK DK01933769T patent/DK1313740T3/da active
- 2001-03-28 CA CA002404474A patent/CA2404474A1/en not_active Abandoned
- 2001-03-28 MX MXPA02009551A patent/MXPA02009551A/es active IP Right Grant
- 2001-03-28 BR BR0109483-1A patent/BR0109483A/pt not_active Application Discontinuation
- 2001-03-28 CZ CZ20023194A patent/CZ20023194A3/cs unknown
- 2001-03-28 KR KR1020027012842A patent/KR100860627B1/ko not_active Expired - Fee Related
- 2001-03-28 SK SK1385-2002A patent/SK286850B6/sk not_active IP Right Cessation
- 2001-03-28 ES ES01933769T patent/ES2253376T3/es not_active Expired - Lifetime
- 2001-03-28 CN CNB018071635A patent/CN1214030C/zh not_active Expired - Fee Related
-
2002
- 2002-08-12 IL IL151200A patent/IL151200A/en not_active IP Right Cessation
- 2002-09-23 ZA ZA200207637A patent/ZA200207637B/en unknown
- 2002-09-27 NO NO20024662A patent/NO20024662L/no not_active Application Discontinuation
-
2004
- 2004-04-19 US US10/826,337 patent/US7189736B2/en not_active Expired - Fee Related
Also Published As
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