DK129704B - Fremgangsmåde til fremstilling af 17α-klor-6α-fluor-16α-methylpregna-1,4-dien-3,20-dion-21-oler eller estere deraf. - Google Patents
Fremgangsmåde til fremstilling af 17α-klor-6α-fluor-16α-methylpregna-1,4-dien-3,20-dion-21-oler eller estere deraf.Info
- Publication number
- DK129704B DK129704B DK428471AA DK428471A DK129704B DK 129704 B DK129704 B DK 129704B DK 428471A A DK428471A A DK 428471AA DK 428471 A DK428471 A DK 428471A DK 129704 B DK129704 B DK 129704B
- Authority
- DK
- Denmark
- Prior art keywords
- methylpregna
- dione
- diene
- fluoro
- chloro
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J5/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE2047105A DE2047105C3 (de) | 1970-09-18 | 1970-09-18 | 17-Chlorsteroide und Verfahren zu ihrer Herstellung |
Publications (2)
Publication Number | Publication Date |
---|---|
DK129704B true DK129704B (da) | 1974-11-11 |
DK129704C DK129704C (da) | 1975-04-21 |
Family
ID=5783313
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK428471AA DK129704B (da) | 1970-09-18 | 1971-09-01 | Fremgangsmåde til fremstilling af 17α-klor-6α-fluor-16α-methylpregna-1,4-dien-3,20-dion-21-oler eller estere deraf. |
Country Status (13)
Country | Link |
---|---|
US (1) | US3723484A (da) |
JP (1) | JPS5527919B1 (da) |
AT (1) | AT303983B (da) |
BE (1) | BE772739A (da) |
CH (1) | CH589670A5 (da) |
CS (1) | CS164765B2 (da) |
DE (1) | DE2047105C3 (da) |
DK (1) | DK129704B (da) |
ES (1) | ES394772A1 (da) |
FR (1) | FR2106606B1 (da) |
GB (1) | GB1363472A (da) |
HU (1) | HU162495B (da) |
NL (1) | NL7112856A (da) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1536691A (en) * | 1975-02-01 | 1978-12-20 | Lark Spa | 16-methyl-17-bromo-1,4-pregnadien-21-ol-3,20-dione compounds |
CA2141492C (en) * | 1994-04-28 | 1999-07-27 | Bruce B. Randolph | Transportation of hydrogen fluoride |
DE4433374A1 (de) * | 1994-09-20 | 1996-03-21 | Hoechst Ag | 17-Desoxi-corticosteroid-21-/O/-Carbonsäure- ester, Verfahren zu deren Herstellung und diese enthaltende Arzneimittel |
EP2778158A1 (en) * | 2013-03-14 | 2014-09-17 | Advanced Technology Materials, Inc. | Sulfolane mixtures as ambient aprotic polar solvents |
MX2019005330A (es) | 2016-11-08 | 2019-09-11 | Regeneron Pharma | Esteroides y conjugados de proteinas de los mismos. |
MX2019013690A (es) | 2017-05-18 | 2020-01-27 | Regeneron Pharma | Conjugados de farmaco-proteina con ciclodextrina. |
KR20200085807A (ko) | 2017-11-07 | 2020-07-15 | 리제너론 파마슈티칼스 인코포레이티드 | 항체 약물 접합제용 친수성 링커 |
MA54673A1 (fr) | 2018-01-08 | 2022-08-31 | Regeneron Pharma | Stéroïdes et leurs conjugués-anticorps |
CA3098453A1 (en) | 2018-05-09 | 2019-11-14 | Regeneron Pharmaceuticals, Inc. | Anti-msr1 antibodies and methods of use thereof |
US20220411460A1 (en) * | 2021-06-29 | 2022-12-29 | Board Of Regents, The University Of Texas System | Modified glucocorticoids |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3290338A (en) * | 1959-06-01 | 1966-12-06 | Schering Corp | 16-alkylprogesterones and their 9alpha, 11beta-dihalogeno analogs |
US3312692A (en) * | 1959-12-22 | 1967-04-04 | Schering Corp | 16-alkylene progesterones and intermediates formed in the production thereof |
AT241702B (de) * | 1960-01-13 | 1965-08-10 | Ayerst Mckenna & Harrison | Verfahren zur Herstellung von 17α-Brom-6α-halogenprogesteronen |
US3519651A (en) * | 1964-09-29 | 1970-07-07 | Hoffmann La Roche | 3,5-seco-a-norpregnan-3-oic acid-3,11-lactones |
-
1970
- 1970-09-18 DE DE2047105A patent/DE2047105C3/de not_active Expired
-
1971
- 1971-08-23 GB GB3940371A patent/GB1363472A/en not_active Expired
- 1971-08-31 CS CS6225A patent/CS164765B2/cs unknown
- 1971-09-01 DK DK428471AA patent/DK129704B/da unknown
- 1971-09-02 CH CH1295271A patent/CH589670A5/xx not_active IP Right Cessation
- 1971-09-03 ES ES394772A patent/ES394772A1/es not_active Expired
- 1971-09-15 US US00180898A patent/US3723484A/en not_active Expired - Lifetime
- 1971-09-16 HU HUSC351A patent/HU162495B/hu unknown
- 1971-09-17 FR FR7133558A patent/FR2106606B1/fr not_active Expired
- 1971-09-17 AT AT809571A patent/AT303983B/de active
- 1971-09-17 BE BE772739A patent/BE772739A/xx unknown
- 1971-09-17 NL NL7112856A patent/NL7112856A/xx not_active Application Discontinuation
- 1971-09-18 JP JP7294371A patent/JPS5527919B1/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
DE2047105A1 (de) | 1972-03-23 |
ES394772A1 (es) | 1974-03-01 |
FR2106606A1 (da) | 1972-05-05 |
FR2106606B1 (da) | 1974-11-15 |
NL7112856A (da) | 1972-03-21 |
BE772739A (fr) | 1972-03-17 |
CH589670A5 (da) | 1977-07-15 |
HU162495B (da) | 1973-02-28 |
AT303983B (de) | 1972-12-27 |
DE2047105C3 (de) | 1979-02-15 |
DK129704C (da) | 1975-04-21 |
GB1363472A (en) | 1974-08-14 |
JPS5527919B1 (da) | 1980-07-24 |
DE2047105B2 (de) | 1978-05-11 |
CS164765B2 (da) | 1975-11-28 |
US3723484A (en) | 1973-03-27 |
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