DK1053240T3 - Glucocorticoid-selektiv antiinflammatoriske midler - Google Patents
Glucocorticoid-selektiv antiinflammatoriske midlerInfo
- Publication number
- DK1053240T3 DK1053240T3 DK99905971T DK99905971T DK1053240T3 DK 1053240 T3 DK1053240 T3 DK 1053240T3 DK 99905971 T DK99905971 T DK 99905971T DK 99905971 T DK99905971 T DK 99905971T DK 1053240 T3 DK1053240 T3 DK 1053240T3
- Authority
- DK
- Denmark
- Prior art keywords
- glucocorticoid
- mammal
- inflammatory agents
- selective anti
- compounds
- Prior art date
Links
- 229940121363 anti-inflammatory agent Drugs 0.000 title 1
- 239000002260 anti-inflammatory agent Substances 0.000 title 1
- 239000003862 glucocorticoid Substances 0.000 title 1
- 241000124008 Mammalia Species 0.000 abstract 3
- 208000023275 Autoimmune disease Diseases 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 208000026278 immune system disease Diseases 0.000 abstract 2
- 102000003676 Glucocorticoid Receptors Human genes 0.000 abstract 1
- 108090000079 Glucocorticoid Receptors Proteins 0.000 abstract 1
- 241000845077 Iare Species 0.000 abstract 1
- 230000003042 antagnostic effect Effects 0.000 abstract 1
- 230000001363 autoimmune Effects 0.000 abstract 1
- 208000027866 inflammatory disease Diseases 0.000 abstract 1
- 230000002401 inhibitory effect Effects 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 230000000754 repressing effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Cosmetics (AREA)
- Cephalosporin Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US09/023,913 US6380207B2 (en) | 1998-02-13 | 1998-02-13 | Glucocortiocoid-selective antiinflammatory agents |
| PCT/US1999/003210 WO1999041257A1 (en) | 1998-02-13 | 1999-02-15 | Glucocorticoid-selective antiinflammatory agents |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK1053240T3 true DK1053240T3 (da) | 2003-08-11 |
Family
ID=21817891
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK99905971T DK1053240T3 (da) | 1998-02-13 | 1999-02-15 | Glucocorticoid-selektiv antiinflammatoriske midler |
Country Status (24)
| Country | Link |
|---|---|
| US (1) | US6380207B2 (da) |
| EP (1) | EP1053240B1 (da) |
| JP (1) | JP2002503666A (da) |
| KR (1) | KR20010040940A (da) |
| CN (1) | CN1153771C (da) |
| AT (1) | ATE237620T1 (da) |
| AU (1) | AU760511B2 (da) |
| BG (1) | BG64213B1 (da) |
| BR (1) | BR9907847A (da) |
| CA (1) | CA2320911A1 (da) |
| DE (1) | DE69906938T2 (da) |
| DK (1) | DK1053240T3 (da) |
| ES (1) | ES2197618T3 (da) |
| HK (1) | HK1033309A1 (da) |
| HU (1) | HUP0100846A3 (da) |
| IL (1) | IL137509A0 (da) |
| NO (1) | NO20004052L (da) |
| NZ (1) | NZ506012A (da) |
| PL (1) | PL342999A1 (da) |
| PT (1) | PT1053240E (da) |
| SK (1) | SK284076B6 (da) |
| TR (1) | TR200002345T2 (da) |
| WO (1) | WO1999041257A1 (da) |
| ZA (1) | ZA99533B (da) |
Families Citing this family (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6566372B1 (en) * | 1999-08-27 | 2003-05-20 | Ligand Pharmaceuticals Incorporated | Bicyclic androgen and progesterone receptor modulator compounds and methods |
| ATE303369T1 (de) | 2000-10-30 | 2005-09-15 | Pfizer Prod Inc | Glucocorticoid rezeptor modulatoren |
| US7026484B2 (en) * | 2001-02-23 | 2006-04-11 | Ligand Pharmaceuticals Incorporated | Tricyclic androgen receptor modulator compounds and methods |
| WO2003061651A1 (en) | 2002-01-22 | 2003-07-31 | The Regents Of The University Of California | Non-steroidal ligands for the glucocorticoid receptor, compositions and uses thereof |
| KR100492913B1 (ko) * | 2002-08-23 | 2005-06-03 | 주식회사 태평양 | 피부 감작 및 자극을 완화하는 피부 외용제 조성물 |
| US20040138187A1 (en) | 2002-08-28 | 2004-07-15 | Reading Christopher L. | Therapeutic treatment methods |
| US20040220153A1 (en) * | 2002-09-24 | 2004-11-04 | Jost-Price Edward Roydon | Methods and reagents for the treatment of diseases and disorders associated with increased levels of proinflammatory cytokines |
| MXPA05003800A (es) * | 2002-10-11 | 2005-06-08 | Ligand Pharm Inc | 5-(1¦,1¦-cicloalquil/alquenil)metiliden 1,2-dihidro-5h- cromeno[3,4f]quinolinas como compuestos moduladores de receptor de progesterona selectivos. |
| DE20301728U1 (de) * | 2002-10-11 | 2004-03-11 | Ligand Pharmaceuticals, Inc., San Diego | 5-substituierte 7,9-Difluor-5H-Chromeno(3,4-f) -Chinolin-Verbindungen als selektive Progesteronrezeptormodulator-Verbindungen |
| EP1551845A1 (en) * | 2002-10-11 | 2005-07-13 | Ligand Pharmaceuticals, Inc. | 5-CYCLOALKENYL 5 i H /i -CHROMENO 3,4-F QUINOLINE DERIV ATIVES AS SELECTIVE PROGESTERONE RECEPTOR MODULATOR COMPOUNDS |
| US7235662B2 (en) * | 2003-06-11 | 2007-06-26 | Bristol-Myers Squibb Company | Modulators of the glucocorticoid receptor and method |
| BRPI0413820A (pt) | 2003-08-22 | 2006-10-24 | Ligand Pharm Inc | derivados de 6-cicloamino-2-quinolinona como compostos moduladores de receptor de androgênio |
| TW200517114A (en) | 2003-10-15 | 2005-06-01 | Combinatorx Inc | Methods and reagents for the treatment of immunoinflammatory disorders |
| AU2004292445B2 (en) | 2003-11-21 | 2010-02-04 | Zalicus Inc. | Methods and reagents for the treatment of inflammatory disorders |
| US8519158B2 (en) * | 2004-03-12 | 2013-08-27 | Ligand Pharmaceuticals Incorporated | Androgen receptor modulator compounds and methods |
| US8193357B2 (en) | 2005-06-17 | 2012-06-05 | Ligand Pharmaceuticals Incorporated | Androgen receptor modulator compounds |
| EP1916896A4 (en) | 2005-08-26 | 2010-08-11 | Univ California | NOT STEROID-antiandrogens |
| US20070225217A1 (en) | 2005-11-09 | 2007-09-27 | Combinatorx, Incorporated | Methods, compositions, and kits for the treatment of medical conditions |
| CN101326169B (zh) * | 2005-12-09 | 2011-11-16 | 霍夫曼-拉罗奇有限公司 | 作为抗炎剂的糖皮质激素受体调节剂 |
| WO2007065821A1 (en) * | 2005-12-09 | 2007-06-14 | F. Hoffmann-La Roche Ag | Propionamide compounds as antiinflammatory agents |
| US8269612B2 (en) | 2008-07-10 | 2012-09-18 | Black & Decker Inc. | Communication protocol for remotely controlled laser devices |
| US20100092479A1 (en) * | 2008-08-18 | 2010-04-15 | Combinatorx (Singapore) Pte. Ltd. | Compositions and methods for treatment of viral diseases |
| US9908182B2 (en) | 2012-01-30 | 2018-03-06 | Black & Decker Inc. | Remote programming of a power tool |
| US8919456B2 (en) | 2012-06-08 | 2014-12-30 | Black & Decker Inc. | Fastener setting algorithm for drill driver |
| US10011006B2 (en) | 2013-08-08 | 2018-07-03 | Black & Decker Inc. | Fastener setting algorithm for drill driver |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5696127A (en) | 1994-12-22 | 1997-12-09 | Ligand Pharmaceuticals Incorporated | Steroid receptor modulator compounds and methods |
| PT800519E (pt) | 1994-12-22 | 2004-03-31 | Ligand Pharm Inc | Compostos moduladores de receptores de esteroides e metodos |
| US5693133A (en) | 1995-05-10 | 1997-12-02 | Akzo Nobel Nv | Asbestos free roof coatings |
-
1998
- 1998-02-13 US US09/023,913 patent/US6380207B2/en not_active Expired - Fee Related
-
1999
- 1999-01-25 ZA ZA9900533A patent/ZA99533B/xx unknown
- 1999-02-15 NZ NZ506012A patent/NZ506012A/xx unknown
- 1999-02-15 SK SK1196-2000A patent/SK284076B6/sk unknown
- 1999-02-15 ES ES99905971T patent/ES2197618T3/es not_active Expired - Lifetime
- 1999-02-15 CA CA002320911A patent/CA2320911A1/en not_active Abandoned
- 1999-02-15 PL PL99342999A patent/PL342999A1/xx unknown
- 1999-02-15 TR TR2000/02345T patent/TR200002345T2/xx unknown
- 1999-02-15 KR KR1020007008857A patent/KR20010040940A/ko not_active Application Discontinuation
- 1999-02-15 WO PCT/US1999/003210 patent/WO1999041257A1/en not_active Application Discontinuation
- 1999-02-15 JP JP2000531450A patent/JP2002503666A/ja not_active Withdrawn
- 1999-02-15 PT PT99905971T patent/PT1053240E/pt unknown
- 1999-02-15 DE DE69906938T patent/DE69906938T2/de not_active Expired - Fee Related
- 1999-02-15 AT AT99905971T patent/ATE237620T1/de not_active IP Right Cessation
- 1999-02-15 CN CNB998050342A patent/CN1153771C/zh not_active Expired - Fee Related
- 1999-02-15 BR BR9907847-3A patent/BR9907847A/pt not_active IP Right Cessation
- 1999-02-15 DK DK99905971T patent/DK1053240T3/da active
- 1999-02-15 AU AU26003/99A patent/AU760511B2/en not_active Ceased
- 1999-02-15 EP EP99905971A patent/EP1053240B1/en not_active Expired - Lifetime
- 1999-02-15 HU HU0100846A patent/HUP0100846A3/hu unknown
- 1999-02-15 IL IL13750999A patent/IL137509A0/xx unknown
-
2000
- 2000-08-11 NO NO20004052A patent/NO20004052L/no not_active Application Discontinuation
- 2000-08-17 BG BG104698A patent/BG64213B1/bg unknown
-
2001
- 2001-04-19 HK HK01102795A patent/HK1033309A1/xx not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| ES2197618T3 (es) | 2004-01-01 |
| CN1153771C (zh) | 2004-06-16 |
| EP1053240B1 (en) | 2003-04-16 |
| AU760511B2 (en) | 2003-05-15 |
| PT1053240E (pt) | 2003-09-30 |
| HK1033309A1 (en) | 2001-08-24 |
| IL137509A0 (en) | 2001-07-24 |
| HUP0100846A3 (en) | 2003-03-28 |
| EP1053240A1 (en) | 2000-11-22 |
| NO20004052D0 (no) | 2000-08-11 |
| TR200002345T2 (tr) | 2000-11-21 |
| NZ506012A (en) | 2003-03-28 |
| PL342999A1 (en) | 2001-07-16 |
| ZA99533B (en) | 1999-07-26 |
| JP2002503666A (ja) | 2002-02-05 |
| BG104698A (en) | 2001-05-31 |
| BG64213B1 (bg) | 2004-05-31 |
| KR20010040940A (ko) | 2001-05-15 |
| BR9907847A (pt) | 2001-01-09 |
| ATE237620T1 (de) | 2003-05-15 |
| NO20004052L (no) | 2000-10-12 |
| CA2320911A1 (en) | 1999-08-19 |
| SK11962000A3 (sk) | 2001-03-12 |
| HUP0100846A2 (hu) | 2001-09-28 |
| DE69906938D1 (de) | 2003-05-22 |
| DE69906938T2 (de) | 2004-02-26 |
| CN1297451A (zh) | 2001-05-30 |
| US20010049377A1 (en) | 2001-12-06 |
| SK284076B6 (sk) | 2004-09-08 |
| US6380207B2 (en) | 2002-04-30 |
| AU2600399A (en) | 1999-08-30 |
| WO1999041257A1 (en) | 1999-08-19 |
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