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DK104056C - Fremgangsmåde til fremstilling af 3-hydroxy-20α-(β-N,N-dimethylaminoethylamino)-19-nor-Δ<1,3,5(10)>-pregnatrien eller estere, ethere eller salte deraf. - Google Patents

Fremgangsmåde til fremstilling af 3-hydroxy-20α-(β-N,N-dimethylaminoethylamino)-19-nor-Δ<1,3,5(10)>-pregnatrien eller estere, ethere eller salte deraf.

Info

Publication number
DK104056C
DK104056C DK269763AA DK269763A DK104056C DK 104056 C DK104056 C DK 104056C DK 269763A A DK269763A A DK 269763AA DK 269763 A DK269763 A DK 269763A DK 104056 C DK104056 C DK 104056C
Authority
DK
Denmark
Prior art keywords
pregnatriene
dimethylaminoethylamino
ethers
hydroxy
esters
Prior art date
Application number
DK269763AA
Other languages
English (en)
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Application granted granted Critical
Publication of DK104056C publication Critical patent/DK104056C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051Estrane derivatives
    • C07J1/0059Estrane derivatives substituted in position 17 by a keto group
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0072Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the A ring of the steroid being aromatic
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0094Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 containing nitrile radicals, including thiocyanide radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J7/00Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms
    • C07J7/0005Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21
    • C07J7/001Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21 substituted in position 20 by a keto group
    • C07J7/0015Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21 substituted in position 20 by a keto group not substituted in position 17 alfa
    • C07J7/002Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21 substituted in position 20 by a keto group not substituted in position 17 alfa not substituted in position 16

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Toxicology (AREA)
  • Steroid Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK269763AA 1962-06-25 1963-06-07 Fremgangsmåde til fremstilling af 3-hydroxy-20α-(β-N,N-dimethylaminoethylamino)-19-nor-Δ<1,3,5(10)>-pregnatrien eller estere, ethere eller salte deraf. DK104056C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR901845A FR1380424A (fr) 1962-06-25 1962-06-25 Nouveaux aminostéroïdes et procédé de préparation
FR933795A FR57F (da) 1962-06-25 1963-05-06

Publications (1)

Publication Number Publication Date
DK104056C true DK104056C (da) 1966-03-28

Family

ID=26196314

Family Applications (1)

Application Number Title Priority Date Filing Date
DK269763AA DK104056C (da) 1962-06-25 1963-06-07 Fremgangsmåde til fremstilling af 3-hydroxy-20α-(β-N,N-dimethylaminoethylamino)-19-nor-Δ<1,3,5(10)>-pregnatrien eller estere, ethere eller salte deraf.

Country Status (10)

Country Link
US (1) US3156619A (da)
BE (1) BE634065A (da)
CH (1) CH405300A (da)
DE (1) DE1290141B (da)
DK (1) DK104056C (da)
ES (1) ES289304A1 (da)
FR (4) FR1380424A (da)
GB (2) GB1031906A (da)
NL (3) NL6603331A (da)
SE (1) SE311357B (da)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1061778A (en) * 1963-07-18 1967-03-15 Merck & Co Inc Indolyl acetic acid glucuronides
US3285935A (en) * 1963-07-18 1966-11-15 Merck & Co Inc Indolyl glucuronides
USRE35053E (en) * 1985-09-12 1995-10-10 The Upjohn Company Amines useful in producing pharmaceutically active CNS compounds
US5506354A (en) * 1985-09-12 1996-04-09 The Upjohn Company Imidazolylpiperazinyl steroids
US5099019A (en) * 1985-09-12 1992-03-24 Upjohn Company Amines useful in producing pharmaceutically active CNS compounds
US4939134A (en) * 1988-09-19 1990-07-03 New York University 26-aminocholesterol and derivatives and analogs thereof in the regulation of cholesterol accumulation in body tissue
US5274088A (en) * 1992-07-02 1993-12-28 New York University Method for the preparation of (25r)-26-aminocholesterol
FR2718138B1 (fr) * 1994-04-01 1996-04-26 Roussel Uclaf Nouveaux stéroïdes comportant en position 20 une chaîne aminosubstituée, procédé et intermédiaires de préparation, application comme médicaments et compositions pharmaceutiques les renfermant.
US6054446A (en) * 1997-12-24 2000-04-25 Sri International Anti-estrogenic steroids, and associated pharmaceutical compositions and methods of use

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3013008A (en) * 1961-01-09 1961-12-12 Searle & Co N-substituted 20-aminopregnan-3-ols, esters thereof, and deta-derivatives corresponding

Also Published As

Publication number Publication date
BE634065A (da) 1900-01-01
ES289304A1 (es) 1963-08-16
SE311357B (da) 1969-06-09
NL120952C (da) 1900-01-01
NL6603331A (da) 1966-06-27
FR1380424A (fr) 1964-12-04
DE1290141B (de) 1969-03-06
NL294517A (da) 1900-01-01
FR57F (da) 1964-10-16
GB1031905A (en) 1966-06-02
GB1031906A (en) 1966-06-02
FR90805E (fr) 1968-02-23
CH405300A (fr) 1966-01-15
FR2488M (fr) 1900-01-01
US3156619A (en) 1964-11-10

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