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DE69518323D1 - OXABOROLE AND THEIR SALTS, AND THEIR USE AS BIOCIDES - Google Patents

OXABOROLE AND THEIR SALTS, AND THEIR USE AS BIOCIDES

Info

Publication number
DE69518323D1
DE69518323D1 DE69518323T DE69518323T DE69518323D1 DE 69518323 D1 DE69518323 D1 DE 69518323D1 DE 69518323 T DE69518323 T DE 69518323T DE 69518323 T DE69518323 T DE 69518323T DE 69518323 D1 DE69518323 D1 DE 69518323D1
Authority
DE
Germany
Prior art keywords
pct
oxaborole
biocides
salts
date dec
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE69518323T
Other languages
German (de)
Other versions
DE69518323T2 (en
Inventor
William Austin
Juan Kneale
Jelf Crowley
Martin CLOUGH
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Avecia Ltd
Original Assignee
Avecia Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Avecia Ltd filed Critical Avecia Ltd
Publication of DE69518323D1 publication Critical patent/DE69518323D1/en
Application granted granted Critical
Publication of DE69518323T2 publication Critical patent/DE69518323T2/en
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N55/00—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur
    • A01N55/08—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur containing boron
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N55/00—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds
    • C—CHEMISTRY; METALLURGY
    • C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08K—Use of inorganic or non-macromolecular organic substances as compounding ingredients
    • C08K5/00—Use of organic ingredients
    • C08K5/0008—Organic ingredients according to more than one of the "one dot" groups of C08K5/01 - C08K5/59
    • C08K5/0058—Biocides
    • C—CHEMISTRY; METALLURGY
    • C09—DYES; PAINTS; POLISHES; NATURAL RESINS; ADHESIVES; COMPOSITIONS NOT OTHERWISE PROVIDED FOR; APPLICATIONS OF MATERIALS NOT OTHERWISE PROVIDED FOR
    • C09D—COATING COMPOSITIONS, e.g. PAINTS, VARNISHES OR LACQUERS; FILLING PASTES; CHEMICAL PAINT OR INK REMOVERS; INKS; CORRECTING FLUIDS; WOODSTAINS; PASTES OR SOLIDS FOR COLOURING OR PRINTING; USE OF MATERIALS THEREFOR
    • C09D5/00—Coating compositions, e.g. paints, varnishes or lacquers, characterised by their physical nature or the effects produced; Filling pastes
    • C09D5/14—Paints containing biocides, e.g. fungicides, insecticides or pesticides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Zoology (AREA)
  • Agronomy & Crop Science (AREA)
  • Polymers & Plastics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Biodiversity & Conservation Biology (AREA)
  • Materials Engineering (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Catalysts (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

PCT No. PCT/GB95/01206 Sec. 371 Date Dec. 9, 1996 Sec. 102(e) Date Dec. 9, 1996 PCT Filed May 26, 1995 PCT Pub. No. WO95/33754 PCT Pub. Date Dec. 14, 1995A method for the protection of a medium by susceptible to microbial attack by the treatment of the medium with an oxaborale or a salt of an oxaborale.
DE69518323T 1994-06-09 1995-05-26 OXABOROLE AND THEIR SALTS, AND THEIR USE AS BIOCIDES Expired - Fee Related DE69518323T2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB9411587A GB9411587D0 (en) 1994-06-09 1994-06-09 Compound, composition and use
PCT/GB1995/001206 WO1995033754A1 (en) 1994-06-09 1995-05-26 Oxaboroles and salts thereof, and their use as biocides

Publications (2)

Publication Number Publication Date
DE69518323D1 true DE69518323D1 (en) 2000-09-14
DE69518323T2 DE69518323T2 (en) 2001-02-01

Family

ID=10756481

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69518323T Expired - Fee Related DE69518323T2 (en) 1994-06-09 1995-05-26 OXABOROLE AND THEIR SALTS, AND THEIR USE AS BIOCIDES

Country Status (14)

Country Link
US (1) US5880188A (en)
EP (1) EP0765331B1 (en)
JP (1) JPH10500983A (en)
KR (1) KR970703349A (en)
CN (1) CN1068005C (en)
AT (1) ATE195316T1 (en)
AU (1) AU681291B2 (en)
BR (1) BR9507966A (en)
CA (1) CA2190155A1 (en)
DE (1) DE69518323T2 (en)
GB (1) GB9411587D0 (en)
NO (1) NO965235L (en)
TW (1) TW368397B (en)
WO (1) WO1995033754A1 (en)

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US6184363B1 (en) 1997-06-13 2001-02-06 Northwestern University Inhibitors of β-lactamases and uses therefor
JP2002504122A (en) 1997-06-13 2002-02-05 ノースウエスタン ユニバーシティー Beta-lactamase inhibitors and methods of use
MXPA05013848A (en) * 2003-06-16 2006-09-04 Anacor Pharmaceuticals Inc Hydrolytically-resistant boron-containing therapeutics and methods of use.
KR20050047699A (en) * 2003-11-18 2005-05-23 주식회사 엘지생명과학 Fungicidal aqueous suspension concentrate
HUE054365T2 (en) * 2005-02-16 2021-09-28 Anacor Pharmaceuticals Inc Boronophthalides for therapeutic use
AU2006333527B2 (en) 2005-12-30 2013-08-01 Anacor Pharmaceuticals, Llc Boron-containing small molecules
CN102532180B (en) * 2005-12-30 2016-06-29 安纳考尔医药公司 The little molecule of boracic
DK2719388T3 (en) * 2006-02-16 2019-05-13 Anacor Pharmaceuticals Inc Boron-containing small molecules as anti-inflammatory agents
US20070197388A1 (en) * 2006-02-22 2007-08-23 Buckman Laboratories International, Inc. Haloperoxidase treatment to control algae
KR20080110812A (en) * 2006-03-16 2008-12-19 몰레악 피티이 엘티디 Combination Therapy for the Treatment of Patients with Neuropathy and Cerebral Infarction
EP2015757A4 (en) * 2006-05-02 2011-01-26 Anacor Pharmaceuticals Inc THERAPEUTIC SUBSTANCES CONTAINING HYDROLYSIS-RESISTANT BORON AND METHODS OF USE
EP1900378A1 (en) * 2006-08-31 2008-03-19 Novartis AG Pharmaceutical compositions for the treatment of fungal infections
JO3396B1 (en) 2007-06-20 2019-10-20 Anacor Pharmaceuticals Inc Boron-containing small molecules
JP5504454B2 (en) * 2007-12-06 2014-05-28 国立大学法人京都大学 Novel boron compounds, methods for producing them, and functional electronic devices using them
JP5745279B2 (en) * 2008-01-09 2015-07-08 アナコール ファーマシューティカルズ，インコーポレイテッド Boron-containing small molecules as anti-inflammatory agents
AU2009221793B2 (en) 2008-03-06 2015-02-19 Anacor Pharmaceuticals, Inc Boron-containing small molecules as anti-inflammatory agents
EP2285384A4 (en) * 2008-05-12 2012-04-25 Anacor Pharmaceuticals Inc SMALL MOLECULES CONTAINING BORON
EP2348863A4 (en) 2008-09-04 2012-03-07 Anacor Pharmaceuticals Inc SMALL MOLECULES CONTAINING BORON
US8461336B2 (en) 2008-09-04 2013-06-11 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
CA2739060C (en) 2008-10-15 2016-08-23 Kissei Pharmaceutical Co., Ltd. Fused-ring derivative and medical application of same
US9493489B2 (en) 2008-10-15 2016-11-15 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as anti-protozoal agents
PE20120052A1 (en) 2008-12-17 2012-02-13 Anacor Pharmaceuticals Inc (S) -3-AMINO-METHYL-7- (3-HYDROXY-PROPOXY) -3H-BENZO- [C] [1,2] -OXABOROL-1-OL POLYMORPHES
JP2013500974A (en) 2009-07-28 2013-01-10 アナコール ファーマシューティカルズ，インコーポレイテッド Trisubstituted boron-containing molecules
US9440994B2 (en) 2009-08-14 2016-09-13 Anacor Pharmaceuticals, Inc. Boron containing small molecules as antiprotozoal agents
US20110207701A1 (en) * 2009-08-19 2011-08-25 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as antiprotozoal agents
US9346834B2 (en) 2009-10-20 2016-05-24 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as antiprotozoal agents
US8461134B2 (en) 2009-11-11 2013-06-11 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
WO2011094450A1 (en) 2010-01-27 2011-08-04 Anacor Pharmaceuticals, Inc Boron-containing small molecules
WO2011116348A1 (en) 2010-03-19 2011-09-22 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as anti-protozoal agent
HUE059033T2 (en) 2010-09-07 2022-10-28 Anacor Pharmaceuticals Inc Benzoxaborole derivatives for the treatment of bacterial infections
AU2012320382B2 (en) * 2011-10-07 2015-11-26 Syngenta Participations Ag Method for protecting useful plants or plant propagation material
UY34367A (en) * 2011-10-07 2014-08-29 Syngenta Participations Ag ? METHOD TO PROTECT MATERIAL OF VEGETABLE PROPAGATION OR USEFUL PLANTS ?.
US11039617B2 (en) 2013-01-30 2021-06-22 Agrofresh Inc. Large scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness
US8669207B1 (en) 2013-01-30 2014-03-11 Dow Agrosciences, Llc. Compounds and compositions
RU2595157C1 (en) 2013-01-30 2016-08-20 Агрофреш Инк. Use of benzoxaboroles as antimicrobial agents for treatment of meat products, plants or parts of plants
US9585396B2 (en) 2013-01-30 2017-03-07 Agrofresh Inc. Volatile applications against pathogens
US10070649B2 (en) 2013-01-30 2018-09-11 Agrofresh Inc. Volatile applications against pathogens
US20220125049A1 (en) * 2013-01-30 2022-04-28 Agrofresh Inc. Method and system for centralized management, monitoring, and controlled delivery of biological compounds to fruit storage rooms
WO2014147009A1 (en) * 2013-03-18 2014-09-25 Syngenta Participations Ag Novel microbiocides
WO2014173880A1 (en) 2013-04-22 2014-10-30 Syngenta Participations Ag Novel microbiocides
AU2014202928B1 (en) * 2013-06-05 2014-09-11 Agrofresh Inc. Compounds and compositions
US20170000133A1 (en) * 2013-12-23 2017-01-05 Syngenta Participations Ag Benzoxaborole fungicides
WO2015097237A1 (en) * 2013-12-23 2015-07-02 Syngenta Participations Ag Benzoxaborole fungicides
MA41495A (en) * 2015-02-12 2017-12-19 Anacor Pharmaceuticals Inc BENZOXABOROLE COMPOUNDS AND THEIR USES
WO2016130658A1 (en) * 2015-02-12 2016-08-18 Agrofresh Inc. Fungicidal compounds and compositions
CN107872956B (en) * 2015-04-09 2020-07-10 宾夕法尼亚州研究基金会 Synergistic antifungal composition containing benzoxaborole
WO2017024022A1 (en) * 2015-08-06 2017-02-09 The Penn State Research Foundation Benzoxaborole-containing coating resistant to cellulose-supportable fungus
WO2017031041A1 (en) * 2015-08-17 2017-02-23 Channel Therapeutics, Inc. Functionalized aminobenzoboroxoles
CN113563368A (en) * 2016-03-02 2021-10-29 比尔及梅琳达盖茨基金会 Boron-containing small molecules
NZ745681A (en) 2016-03-07 2022-05-27 Agrofresh Inc Synergistic methods of using benzoxaborole compounds and preservative gases as an antimicrobial for crops
WO2017155877A1 (en) 2016-03-07 2017-09-14 Agrofresh Inc. Vaporized administration of pesticides
US11447506B2 (en) 2016-05-09 2022-09-20 Anacor Pharmaceuticals, Inc. Crystal forms of crisaborole in free form and preparation method and use thereof
MA44968A (en) 2016-05-12 2019-03-20 Anacor Pharmaceuticals Inc OXABOROLE ESTERS AND THEIR USES
PL3704100T3 (en) 2017-11-02 2024-04-22 Halcyon Labs Private Limited Novel process for the preparation tavaborole and its intermediates
MX2020005464A (en) 2017-11-30 2020-12-03 Boragen Inc Benzoxaborole compounds and formulations thereof.
WO2019173814A1 (en) 2018-03-09 2019-09-12 University Of The Sciences Protective groups and methods for protecting benzoxaboroles or oxaboroles
MX2021001904A (en) * 2018-08-18 2021-05-27 Boragen Inc Solid forms of substituted benzoxaborole and compositions thereof.
SG11202102674RA (en) 2018-10-05 2021-04-29 Pfizer Boron containing pde4 inhibitors
US12065456B2 (en) 2019-07-25 2024-08-20 National Institutes Of Health (Nih), U.S. Dept. Of Health And Human Services (Dhhs), U.S. Government Boron-containing pharmacophore
AR120504A1 (en) 2019-11-22 2022-02-16 Agrofresh Inc COMPOSITION AND METHOD FOR TREATMENT OF PLANTS AND PARTS OF PLANTS WITH VOLATILE ASSETS FOR THE CONTROL OF DECOMPOSITION ORGANISMS
EP4100413A1 (en) * 2020-02-05 2022-12-14 AgroFresh Inc. Antimicrobial compounds and compositions
CN114644645B (en) * 2022-03-08 2023-05-26 南京农业大学 3-indole substituted phenylborozole compound and preparation method and application thereof

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GB1396904A (en) * 1972-08-11 1975-06-11 Ici Ltd Method for the control of micro-organisms

Also Published As

Publication number Publication date
NO965235D0 (en) 1996-12-06
CA2190155A1 (en) 1995-12-14
US5880188A (en) 1999-03-09
ATE195316T1 (en) 2000-08-15
AU2534895A (en) 1996-01-04
DE69518323T2 (en) 2001-02-01
EP0765331A1 (en) 1997-04-02
AU681291B2 (en) 1997-08-21
CN1068005C (en) 2001-07-04
KR970703349A (en) 1997-07-03
WO1995033754A1 (en) 1995-12-14
EP0765331B1 (en) 2000-08-09
TW368397B (en) 1999-09-01
CN1155286A (en) 1997-07-23
BR9507966A (en) 1997-09-02
NO965235L (en) 1997-01-21
GB9411587D0 (en) 1994-08-03
JPH10500983A (en) 1998-01-27

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Legal Events

Date Code Title Description
8339 Ceased/non-payment of the annual fee