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CY1125395T1 - Αντιμικροβιακες συνθεσεις με αναβραζουσες ουσιες - Google Patents

Αντιμικροβιακες συνθεσεις με αναβραζουσες ουσιες

Info

Publication number
CY1125395T1
CY1125395T1 CY20211100955T CY211100955T CY1125395T1 CY 1125395 T1 CY1125395 T1 CY 1125395T1 CY 20211100955 T CY20211100955 T CY 20211100955T CY 211100955 T CY211100955 T CY 211100955T CY 1125395 T1 CY1125395 T1 CY 1125395T1
Authority
CY
Cyprus
Prior art keywords
compositions
antimicrobial compositions
effecting
substances
effecting substances
Prior art date
Application number
CY20211100955T
Other languages
English (en)
Inventor
Danping Li
Original Assignee
Melinta Subsidiary Corp.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=54868661&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CY1125395(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Melinta Subsidiary Corp. filed Critical Melinta Subsidiary Corp.
Publication of CY1125395T1 publication Critical patent/CY1125395T1/el

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4709Non-condensed quinolines and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0002Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0007Effervescent
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/133Amines having hydroxy groups, e.g. sphingosine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2009Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Inorganic Chemistry (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Communicable Diseases (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

Η παρούσα εφεύρεση αφορά σε φαρμακευτικές συνθέσεις, οι οποίες περιλαμβάνουν έναν αντιμικροβιακό παράγοντα παραγώγου του καρβοξυλικού οξέος της κινολόνης και μία αναβράζουσα ουσία. Οι εν λόγω συνθέσεις έχουν βελτιωμένη ανεκτικότητα από το γαστρεντερικό ή/και μειωμένη πιθανότητα να προκαλέσουν παρενέργειες στο γαστρεντερικό. Αυτές οι συνθέσεις είναι χρήσιμες για από του στόματος χορήγηση για τη θεραπευτική αντιμετώπιση, την πρόληψη ή τη μείωση του κινδύνου μικροβιακών λοιμώξεων.
CY20211100955T 2014-06-20 2021-11-04 Αντιμικροβιακες συνθεσεις με αναβραζουσες ουσιες CY1125395T1 (el)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201462014786P 2014-06-20 2014-06-20
PCT/US2015/036605 WO2015196027A1 (en) 2014-06-20 2015-06-19 Antimicrobial compositions with effervescent agents
EP15810507.2A EP3157510B1 (en) 2014-06-20 2015-06-19 Antimicrobial compositions with effervescent agents

Publications (1)

Publication Number Publication Date
CY1125395T1 true CY1125395T1 (el) 2023-03-24

Family

ID=54868661

Family Applications (2)

Application Number Title Priority Date Filing Date
CY20191100664T CY1121995T1 (el) 2014-06-20 2019-06-26 Αντιμικροβιακες συνθεσεις με αναβραζουσες ουσιες
CY20211100955T CY1125395T1 (el) 2014-06-20 2021-11-04 Αντιμικροβιακες συνθεσεις με αναβραζουσες ουσιες

Family Applications Before (1)

Application Number Title Priority Date Filing Date
CY20191100664T CY1121995T1 (el) 2014-06-20 2019-06-26 Αντιμικροβιακες συνθεσεις με αναβραζουσες ουσιες

Country Status (32)

Country Link
US (2) US20150366857A1 (el)
EP (3) EP3919057A1 (el)
JP (2) JP6995479B2 (el)
CN (2) CN106572982B9 (el)
AR (1) AR100920A1 (el)
AU (3) AU2015276954B2 (el)
BR (1) BR112016029761B1 (el)
CA (1) CA2952950C (el)
CL (2) CL2016003273A1 (el)
CR (2) CR20200565A (el)
CY (2) CY1121995T1 (el)
DK (2) DK3157510T3 (el)
EA (1) EA034152B1 (el)
EC (1) ECSP16095540A (el)
ES (2) ES2732865T3 (el)
HR (2) HRP20211685T1 (el)
HU (2) HUE044764T2 (el)
IL (1) IL249622A0 (el)
LT (2) LT3157510T (el)
MX (2) MX368940B (el)
PE (2) PE20210927A1 (el)
PH (2) PH12016502548B1 (el)
PL (2) PL3157510T3 (el)
PT (2) PT3157510T (el)
RS (2) RS62538B1 (el)
SI (2) SI3157510T1 (el)
SM (2) SMT202100618T1 (el)
SV (1) SV2016005349A (el)
TR (1) TR201909417T4 (el)
TW (2) TWI732337B (el)
UY (1) UY36184A (el)
WO (1) WO2015196027A1 (el)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2022240897A1 (en) * 2021-05-10 2022-11-17 Sepelo Therapeutics, Llc Pharmaceutical composition comprising delafloxacin for administration into the lung

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KR101900249B1 (ko) * 2011-01-14 2018-11-02 스페로 트리넴, 인코포레이티드 자이라제 억제제 (r)­1­에틸­3­[6­플루오로­5­[2­(1­하이드록시­1­메틸­에틸)피리미딘­5­일]­7­(테트라하이드로푸란­2­일)­1h­벤즈이미다졸­2­일]우레아의 고체 형태
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Also Published As

Publication number Publication date
AU2021286284B2 (en) 2024-02-29
HUE056298T2 (hu) 2022-02-28
HRP20191133T1 (hr) 2019-09-20
CA2952950A1 (en) 2015-12-23
TR201909417T4 (tr) 2019-07-22
PL3157510T3 (pl) 2019-12-31
BR112016029761A8 (pt) 2021-06-29
NZ727638A (en) 2023-08-25
CR20160592A (es) 2017-02-21
AU2015276954A1 (en) 2017-01-12
PH12016502548A1 (en) 2017-04-10
AU2020256457B2 (en) 2021-09-30
AR100920A1 (es) 2016-11-09
SMT201900348T1 (it) 2019-09-09
TWI705814B (zh) 2020-10-01
HUE044764T2 (hu) 2019-11-28
CA2952950C (en) 2023-11-14
DK3581180T3 (da) 2021-11-08
TW201625249A (zh) 2016-07-16
CL2020003153A1 (es) 2021-06-25
CL2016003273A1 (es) 2017-08-04
ES2897576T3 (es) 2022-03-01
PH12022550979A1 (en) 2023-06-26
HRP20211685T1 (hr) 2022-02-04
CY1121995T1 (el) 2020-10-14
AU2021286284A1 (en) 2022-01-06
EA201692532A1 (ru) 2017-05-31
RS62538B1 (sr) 2021-12-31
ECSP16095540A (es) 2017-03-31
DK3157510T3 (da) 2019-07-01
CN114831955B (zh) 2024-03-12
BR112016029761A2 (pt) 2017-08-22
EA034152B1 (ru) 2020-01-09
TWI732337B (zh) 2021-07-01
CN106572982B9 (zh) 2022-07-08
CN106572982A (zh) 2017-04-19
WO2015196027A1 (en) 2015-12-23
JP7149991B2 (ja) 2022-10-07
MX2019012608A (es) 2019-12-02
BR112016029761B1 (pt) 2023-03-07
MX368940B (es) 2019-10-21
CN106572982B (zh) 2022-06-03
SV2016005349A (es) 2017-08-31
US20200237744A1 (en) 2020-07-30
US20150366857A1 (en) 2015-12-24
PE20210927A1 (es) 2021-05-19
MX2016017350A (es) 2017-04-06
PH12016502548B1 (en) 2023-05-24
EP3581180B1 (en) 2021-08-04
EP3157510A4 (en) 2018-02-21
ES2732865T3 (es) 2019-11-26
SI3157510T1 (sl) 2019-09-30
LT3157510T (lt) 2019-09-25
EP3157510A1 (en) 2017-04-26
SMT202100618T1 (it) 2022-01-10
CN114831955A (zh) 2022-08-02
LT3581180T (lt) 2021-12-27
TW202005650A (zh) 2020-02-01
EP3919057A1 (en) 2021-12-08
JP6995479B2 (ja) 2022-01-14
PE20170304A1 (es) 2017-04-19
EP3581180A1 (en) 2019-12-18
PT3581180T (pt) 2021-11-09
AU2020256457A1 (en) 2020-11-12
PT3157510T (pt) 2019-06-21
PL3581180T3 (pl) 2022-02-07
IL249622A0 (en) 2017-02-28
EP3157510B1 (en) 2019-03-27
JP2020183415A (ja) 2020-11-12
CR20200565A (es) 2021-01-14
AU2015276954B2 (en) 2020-07-23
UY36184A (es) 2016-01-29
JP2017518349A (ja) 2017-07-06
RS59064B1 (sr) 2019-08-30
SI3581180T1 (sl) 2021-12-31

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