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CY1113422T1 - Παραγωγα οξαδιαζολης και η χρηση τους ως ενισχυτων μεταβοτροπικου υποδοχεα γλουταμικου - 842 - Google Patents

Παραγωγα οξαδιαζολης και η χρηση τους ως ενισχυτων μεταβοτροπικου υποδοχεα γλουταμικου - 842

Info

Publication number
CY1113422T1
CY1113422T1 CY20121101132T CY121101132T CY1113422T1 CY 1113422 T1 CY1113422 T1 CY 1113422T1 CY 20121101132 T CY20121101132 T CY 20121101132T CY 121101132 T CY121101132 T CY 121101132T CY 1113422 T1 CY1113422 T1 CY 1113422T1
Authority
CY
Cyprus
Prior art keywords
oxadiasol
transitional
glutamic
receptors
products
Prior art date
Application number
CY20121101132T
Other languages
English (en)
Inventor
Joshua Clayton
Ian Egle
James Emplfield
James Folmer
Methvin Isaac
Fupeng Ma
Abdelmalik Slassi
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40093925&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CY1113422(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of CY1113422T1 publication Critical patent/CY1113422T1/el

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    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Psychology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hematology (AREA)
  • Rheumatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hospice & Palliative Care (AREA)
  • Anesthesiology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Epidemiology (AREA)

Abstract

Ενώσεις του Τύπου (I) όπου το R1 και το Q είναι όπως περιγράφονται στην περιγραφή, φαρμακευτικώς αποδεκτά άλατα, μέθοδοι για την παρασκευή, φαρμακευτικές συνθέσεις που τις περιέχουν και μέθοδοι για τη χρήση αυτών.
CY20121101132T 2007-06-07 2012-11-22 Παραγωγα οξαδιαζολης και η χρηση τους ως ενισχυτων μεταβοτροπικου υποδοχεα γλουταμικου - 842 CY1113422T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US94255307P 2007-06-07 2007-06-07
EP08779348.5A EP2167502B3 (en) 2007-06-07 2008-06-05 Oxadiazole derivatives and their use as metabotropic glutamate receptor potentiators - 842

Publications (1)

Publication Number Publication Date
CY1113422T1 true CY1113422T1 (el) 2016-06-22

Family

ID=40093925

Family Applications (2)

Application Number Title Priority Date Filing Date
CY20121101132T CY1113422T1 (el) 2007-06-07 2012-11-22 Παραγωγα οξαδιαζολης και η χρηση τους ως ενισχυτων μεταβοτροπικου υποδοχεα γλουταμικου - 842
CY20151100204T CY1116150T1 (el) 2007-06-07 2015-02-26 Παραγωγα οξαδιαζολης και η χρηση τους ως ενισχυτων μεταβοτροπικου υποδοχεα γλουταμικου - 842

Family Applications After (1)

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CY20151100204T CY1116150T1 (el) 2007-06-07 2015-02-26 Παραγωγα οξαδιαζολης και η χρηση τους ως ενισχυτων μεταβοτροπικου υποδοχεα γλουταμικου - 842

Country Status (34)

Country Link
US (2) US8377940B2 (el)
EP (2) EP2444399B1 (el)
JP (2) JP5416696B2 (el)
KR (2) KR20150116907A (el)
CN (2) CN101679403B (el)
AR (1) AR066882A1 (el)
AU (1) AU2008260717B2 (el)
BR (1) BRPI0812889A2 (el)
CA (1) CA2690856C (el)
CL (1) CL2008001667A1 (el)
CO (1) CO6251287A2 (el)
CY (2) CY1113422T1 (el)
DK (2) DK2444399T3 (el)
EC (1) ECSP109856A (el)
ES (2) ES2531443T3 (el)
HK (2) HK1142318A1 (el)
HR (2) HRP20120909T4 (el)
IL (1) IL202158A (el)
ME (1) ME01488B (el)
MX (1) MX2009013078A (el)
MY (1) MY158066A (el)
NZ (1) NZ582445A (el)
PE (1) PE20090328A1 (el)
PL (2) PL2444399T3 (el)
PT (2) PT2167502E (el)
RS (2) RS53845B1 (el)
RU (2) RU2470931C2 (el)
SA (1) SA08290344B1 (el)
SI (2) SI2167502T1 (el)
TW (1) TWI417100B (el)
UA (1) UA99129C2 (el)
UY (1) UY31124A1 (el)
WO (1) WO2008150233A1 (el)
ZA (1) ZA200908285B (el)

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