CS242858B2 - Method of octahydro-1h-pyrrolo(2,3-g)-isoquinolines production - Google Patents

Method of octahydro-1h-pyrrolo(2,3-g)-isoquinolines production Download PDF

Info

Publication number: CS242858B2
Authority: CS; Czechoslovakia
Prior art keywords: alkyl; hydroxy; phenyl; compound; alkoxy
Prior art date: 1978-10-13

Application number

CS796945A

Other languages

Czech (cs)

English (en)

Other versions

CS694579A2 (en

Inventor

Leo Berger

Gary Lee Olson

Original Assignee

Hoffmann La Roche

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1978-10-13

Filing date

1979-10-12

Publication date

1986-05-15

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26754910&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CS242858(B2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1979-09-10 Priority claimed from US06/073,813 external-priority patent/US4260762A/en

1979-10-12 Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche

1979-10-12 Priority to CS796945A priority Critical patent/CS613979A2/cs

1979-10-12 Priority to CS796945A priority patent/CS614079A2/cs

1984-08-13 Priority to CS846139A priority patent/CS242899B2/cs

1984-08-13 Priority to CS846140A priority patent/CS242900B2/cs

1985-08-15 Publication of CS694579A2 publication Critical patent/CS694579A2/cs

1986-05-15 Publication of CS242858B2 publication Critical patent/CS242858B2/cs

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/02—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines
- C07D217/04—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines with hydrocarbon or substituted hydrocarbon radicals attached to the ring nitrogen atom
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Medicinal Chemistry (AREA)
Psychiatry (AREA)
Neurology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Biomedical Technology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Neurosurgery (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

CS796945A 1978-10-13 1979-10-12 Method of octahydro-1h-pyrrolo(2,3-g)-isoquinolines production CS242858B2 (en)

Priority Applications (4)

Application Number	Priority Date	Filing Date	Title
CS796945A CS613979A2 (en)	1978-10-13	1979-10-12	Zpusob vyroby oktahydro 1h pyrrolo l2,3 g p isochinolinu
CS796945A CS614079A2 (en)	1978-10-13	1979-10-12	Zpusob vyroby oktahydro-1h-pyrrolo(2,3-g)-isochinonolinu
CS846139A CS242899B2 (cs)	1978-10-13	1984-08-13	Způsob výroby oktahydro-1H-pyrrolo[2,3-g]Ísochinolinů
CS846140A CS242900B2 (cs)	1978-10-13	1984-08-13	Způsob výroby oktahydro-1H-pyrroio[2,3-g]isochinolinů

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US95094778A	1978-10-13	1978-10-13
US06/073,813 US4260762A (en)	1979-09-10	1979-09-10	Octahydro-1H-pyrrolo[2,3-g]isoquinolines

Publications (2)

Publication Number	Publication Date
CS694579A2 CS694579A2 (en)	1985-08-15
CS242858B2 true CS242858B2 (en)	1986-05-15

Family

ID=26754910

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CS796945A CS242858B2 (en)	1978-10-13	1979-10-12	Method of octahydro-1h-pyrrolo(2,3-g)-isoquinolines production

Country Status (18)

Country	Link
EP (1)	EP0010661B1 (es)
AR (2)	AR228244A1 (es)
AU (1)	AU528685B2 (es)
CA (1)	CA1132553A (es)
CS (1)	CS242858B2 (es)
DE (1)	DE2967215D1 (es)
DK (1)	DK430579A (es)
ES (2)	ES493015A0 (es)
FI (1)	FI67548C (es)
HU (1)	HU181883B (es)
IE (1)	IE48965B1 (es)
IL (1)	IL58438A (es)
MC (1)	MC1285A1 (es)
NO (1)	NO152873C (es)
NZ (1)	NZ191830A (es)
PH (1)	PH14835A (es)
PT (1)	PT70310A (es)
SU (3)	SU1014474A3 (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
MC1377A1 (fr) *	1980-02-28	1982-01-19	Hoffmann La Roche	Derives d'isoquinoleine
DE3363146D1 (en) *	1982-03-29	1986-05-28	Hoffmann La Roche	Process for the manufacture of isoquinoline diones
US4732902A (en) *	1986-05-23	1988-03-22	Hoffmann-La Roche Inc.	Pyrroloisoquinolinyl-dimethyloxoalkyl alkonoates and their use as antipsychotic agents
GB8828669D0 (en) *	1988-12-08	1989-01-11	Lilly Industries Ltd	Organic compounds
US6344589B1 (en)	1998-11-20	2002-02-05	Basf Aktiengesellschaft	Method and intermediate products for producing bis(oxime)monoethers

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS51118799A (en) *	1975-04-10	1976-10-18	Sankyo Co Ltd	Method for preparing pyridindole derivatives

1979
- 1979-09-27 CA CA336,495A patent/CA1132553A/en not_active Expired
- 1979-10-08 SU SU812819251K patent/SU1014474A3/ru active
- 1979-10-08 SU SU792819251A patent/SU1109052A3/ru active
- 1979-10-10 MC MC791409A patent/MC1285A1/xx unknown
- 1979-10-11 IL IL58438A patent/IL58438A/xx unknown
- 1979-10-11 DE DE7979103908T patent/DE2967215D1/de not_active Expired
- 1979-10-11 AU AU51697/79A patent/AU528685B2/en not_active Ceased
- 1979-10-11 DK DK430579A patent/DK430579A/da not_active Application Discontinuation
- 1979-10-11 EP EP79103908A patent/EP0010661B1/de not_active Expired
- 1979-10-11 NZ NZ191830A patent/NZ191830A/en unknown
- 1979-10-12 NO NO793301A patent/NO152873C/no unknown
- 1979-10-12 PH PH23160A patent/PH14835A/en unknown
- 1979-10-12 CS CS796945A patent/CS242858B2/cs unknown
- 1979-10-12 AR AR278488A patent/AR228244A1/es active
- 1979-10-12 IE IE1944/79A patent/IE48965B1/en unknown
- 1979-10-12 PT PT70310A patent/PT70310A/pt unknown
- 1979-10-12 FI FI793183A patent/FI67548C/fi not_active IP Right Cessation
- 1979-10-12 HU HU79HO2188A patent/HU181883B/hu not_active IP Right Cessation
1980
- 1980-07-02 ES ES493015A patent/ES493015A0/es active Granted
- 1980-07-02 ES ES493014A patent/ES493014A0/es active Granted
1981
- 1981-03-02 SU SU813250198A patent/SU1048985A3/ru active
- 1981-07-02 AR AR285961A patent/AR229096A1/es active

Also Published As

Publication number	Publication date
SU1014474A3 (ru)	1983-04-23
ES8104806A1 (es)	1981-05-16
FI793183A (fi)	1980-04-14
DE2967215D1 (en)	1984-10-18
AU528685B2 (en)	1983-05-12
NO152873C (no)	1985-12-04
FI67548C (fi)	1985-04-10
HU181883B (en)	1983-11-28
PT70310A (en)	1979-11-01
ES493015A0 (es)	1981-05-16
SU1048985A3 (ru)	1983-10-15
AU5169779A (en)	1980-04-17
AR229096A1 (es)	1983-06-15
DK430579A (da)	1980-04-14
ES8104805A1 (es)	1981-05-16
NZ191830A (en)	1984-09-28
ES493014A0 (es)	1981-05-16
IE791944L (en)	1980-04-13
EP0010661A3 (en)	1980-10-01
EP0010661A2 (de)	1980-05-14
MC1285A1 (fr)	1980-07-22
CA1132553A (en)	1982-09-28
PH14835A (en)	1981-12-16
NO152873B (no)	1985-08-26
NO793301L (no)	1980-04-15
IL58438A (en)	1982-12-31
CS694579A2 (en)	1985-08-15
AR228244A1 (es)	1983-02-15
FI67548B (fi)	1984-12-31
IE48965B1 (en)	1985-06-26
IL58438A0 (en)	1980-01-31
SU1109052A3 (ru)	1984-08-15
EP0010661B1 (de)	1984-09-12

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