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CH545295A - Process for the preparation of substituted benzimidazoles - Google Patents

Process for the preparation of substituted benzimidazoles

Info

Publication number
CH545295A
CH545295A CH184171A CH184171A CH545295A CH 545295 A CH545295 A CH 545295A CH 184171 A CH184171 A CH 184171A CH 184171 A CH184171 A CH 184171A CH 545295 A CH545295 A CH 545295A
Authority
CH
Switzerland
Prior art keywords
preparation
substituted benzimidazoles
benzimidazoles
substituted
Prior art date
Application number
CH184171A
Other languages
German (de)
Inventor
D R Hoff
H Fisher
Richard Hoff Dale
Herbert Fisher Michael
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of CH545295A publication Critical patent/CH545295A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • EFIXED CONSTRUCTIONS
    • E21EARTH OR ROCK DRILLING; MINING
    • E21DSHAFTS; TUNNELS; GALLERIES; LARGE UNDERGROUND CHAMBERS
    • E21D11/00Lining tunnels, galleries or other underground cavities, e.g. large underground chambers; Linings therefor; Making such linings in situ, e.g. by assembling
    • E21D11/14Lining predominantly with metal
    • E21D11/28Longitudinal struts, i.e. longitudinal connections between adjoining arches

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Mining & Mineral Resources (AREA)
  • Epidemiology (AREA)
  • Civil Engineering (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Architecture (AREA)
  • Animal Behavior & Ethology (AREA)
  • Structural Engineering (AREA)
  • Medicinal Chemistry (AREA)
  • General Life Sciences & Earth Sciences (AREA)
  • Geochemistry & Mineralogy (AREA)
  • Geology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
CH184171A 1967-02-03 1968-02-02 Process for the preparation of substituted benzimidazoles CH545295A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US61374667A 1967-02-03 1967-02-03
US69649668A 1968-01-09 1968-01-09

Publications (1)

Publication Number Publication Date
CH545295A true CH545295A (en) 1974-01-31

Family

ID=27087090

Family Applications (5)

Application Number Title Priority Date Filing Date
CH159768A CH509318A (en) 1967-02-03 1968-02-02 Benzimidazole derivatives - as anthelmintics
CH184071A CH545294A (en) 1967-02-03 1968-02-02 Process for the preparation of substituted benzimidazoles
CH184271A CH545796A (en) 1967-02-03 1968-02-02
CH183971A CH545293A (en) 1967-02-03 1968-02-02 Process for the preparation of substituted benzimidazoles
CH184171A CH545295A (en) 1967-02-03 1968-02-02 Process for the preparation of substituted benzimidazoles

Family Applications Before (4)

Application Number Title Priority Date Filing Date
CH159768A CH509318A (en) 1967-02-03 1968-02-02 Benzimidazole derivatives - as anthelmintics
CH184071A CH545294A (en) 1967-02-03 1968-02-02 Process for the preparation of substituted benzimidazoles
CH184271A CH545796A (en) 1967-02-03 1968-02-02
CH183971A CH545293A (en) 1967-02-03 1968-02-02 Process for the preparation of substituted benzimidazoles

Country Status (19)

Country Link
AT (5) AT293378B (en)
BE (2) BE710081A (en)
CH (5) CH509318A (en)
CS (1) CS162651B2 (en)
CY (1) CY653A (en)
DE (2) DE1795711C3 (en)
DK (1) DK139940B (en)
ES (4) ES350083A1 (en)
FI (1) FI52859C (en)
FR (1) FR1580153A (en)
GB (2) GB1198942A (en)
IE (1) IE31812B1 (en)
IT (1) IT1044176B (en)
NL (1) NL157015B (en)
NO (1) NO126484B (en)
OA (1) OA04036A (en)
SE (1) SE346321B (en)
SU (1) SU540569A3 (en)
YU (1) YU33831B (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3711608A (en) * 1971-04-13 1973-01-16 Merck & Co Inc The treatment of pain, fever and inflammation with benzimidazoles
US3983130A (en) * 1972-06-02 1976-09-28 E. R. Squibb & Sons, Inc. Anthelmintic isothiocyanobenzoxazoles
US3985755A (en) * 1972-06-02 1976-10-12 E. R. Squibb & Sons, Inc. Pyridine containing isothiocyanobenzoxazoles
US3853894A (en) * 1972-06-02 1974-12-10 Squibb & Sons Inc Isothiocyanobenzimidazoles
MA19290A1 (en) * 1980-05-22 1982-04-01 Ciba Geigy Ag BENZOLE DERIVATIVES, THEIR PREPARATON AND THEIR THERAPEUTIC USES.
SE8604566D0 (en) * 1986-10-27 1986-10-27 Haessle Ab NOVEL COMPUNDS
US7622592B2 (en) 2002-11-01 2009-11-24 Merck & Co., Inc. Carbonylamino-benzimidazole derivatives as androgen receptor modulators
GB0324792D0 (en) 2003-10-23 2003-11-26 Sterix Ltd Compound
CA2540843A1 (en) * 2003-10-23 2005-05-12 Sterix Limited Phenyl carboxamide and sulfonamide derivatives for use as 11-beta-hydroxysteroid dehydrogenase

Also Published As

Publication number Publication date
AT301244B (en) 1972-08-25
AT289833B (en) 1971-05-10
OA04036A (en) 1979-09-30
CH509318A (en) 1971-06-30
CH545796A (en) 1974-02-15
DE1795711C3 (en) 1979-05-17
AT289828B (en) 1971-05-10
AT293378B (en) 1971-10-11
YU21268A (en) 1977-12-31
ES363760A1 (en) 1970-12-16
DE1795711A1 (en) 1974-02-28
ES350083A1 (en) 1969-11-16
YU33831B (en) 1978-06-30
NL6801482A (en) 1968-08-05
CH545294A (en) 1974-01-31
GB1198941A (en) 1970-07-15
FI52859B (en) 1977-08-31
FI52859C (en) 1977-12-12
NO126484B (en) 1973-02-12
CH545293A (en) 1974-01-31
ES363762A1 (en) 1970-12-16
CY653A (en) 1972-08-31
NL157015B (en) 1978-06-15
FR1580153A (en) 1969-09-05
AT289835B (en) 1971-05-10
DE1695545A1 (en) 1971-05-06
DK139940C (en) 1979-10-15
IE31812B1 (en) 1973-01-10
DE1695545B2 (en) 1978-08-31
BE710081A (en) 1968-07-30
IT1044176B (en) 1980-03-20
CS162651B2 (en) 1975-07-15
GB1198942A (en) 1970-07-15
BE735281A (en) 1969-12-29
SE346321B (en) 1972-07-03
DE1795711B2 (en) 1978-09-21
IE31812L (en) 1968-08-03
SU540569A3 (en) 1976-12-25
DE1695545C3 (en) 1979-05-03
DK139940B (en) 1979-05-21
ES363761A1 (en) 1970-12-16

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Legal Events

Date Code Title Description
PL Patent ceased