CH544116A - Verfahren zur Herstellung von 2-(Thienyl-3 -amino)-1,3-diazacycloalkenen-(2) - Google Patents

Verfahren zur Herstellung von 2-(Thienyl-3 -amino)-1,3-diazacycloalkenen-(2)

Info

Publication number: CH544116A
Authority: CH; Switzerland
Prior art keywords: diazacycloalkenene; thienyl; amino; preparation
Prior art date: 1969-08-13

Application number

CH611473A

Other languages

English (en)

Inventor

Robert Dr Rippel

Ruschig Heinrich Dr Prof

Lindner Ernst Dr Prof

Manfred Dr Schorr

Original Assignee

Hoechst Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1969-08-13

Filing date

1970-08-13

Publication date

1973-12-28

1969-08-16 Priority claimed from DE19691941761 external-priority patent/DE1941761C3/de

1970-08-13 Application filed by Hoechst Ag filed Critical Hoechst Ag

1973-12-28 Publication of CH544116A publication Critical patent/CH544116A/de

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61C—DENTISTRY; APPARATUS OR METHODS FOR ORAL OR DENTAL HYGIENE
- A61C19/00—Dental auxiliary appliances
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
- G—PHYSICS
- G03—PHOTOGRAPHY; CINEMATOGRAPHY; ANALOGOUS TECHNIQUES USING WAVES OTHER THAN OPTICAL WAVES; ELECTROGRAPHY; HOLOGRAPHY
- G03B—APPARATUS OR ARRANGEMENTS FOR TAKING PHOTOGRAPHS OR FOR PROJECTING OR VIEWING THEM; APPARATUS OR ARRANGEMENTS EMPLOYING ANALOGOUS TECHNIQUES USING WAVES OTHER THAN OPTICAL WAVES; ACCESSORIES THEREFOR
- G03B17/00—Details of cameras or camera bodies; Accessories therefor
- G03B17/02—Bodies

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Epidemiology (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Oral & Maxillofacial Surgery (AREA)
Public Health (AREA)
Dentistry (AREA)
Physics & Mathematics (AREA)
General Physics & Mathematics (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Heterocyclic Compounds Containing Sulfur Atoms (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

CH611473A 1969-08-13 1970-08-13 Verfahren zur Herstellung von 2-(Thienyl-3 -amino)-1,3-diazacycloalkenen-(2) CH544116A (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE19691941575 DE1941575A1 (de)	1969-08-13	1969-08-13	Neue Nitrofurylpyrimidinderivate
DE19691941761 DE1941761C3 (de)		1969-08-16	2-(Thienyl-3 '-amino) -1.3-diazacyclopentene und Verfahren zu ihrer Herstellung

Publications (1)

Publication Number	Publication Date
CH544116A true CH544116A (de)	1973-12-28

Family

ID=25757797

Family Applications (4)

Application Number	Title	Priority Date	Filing Date
CH1215970A CH530415A (de)	1969-08-13	1970-08-13	Verfahren zur Herstellung von Pyrimidinderivaten
CH611573A CH554894A (de)	1969-08-13	1970-08-13	Verfahren zur herstellung von 2-(thienyl-3'-amino)-1,3diazacycloalkenen-(2).
CH611473A CH544116A (de)	1969-08-13	1970-08-13	Verfahren zur Herstellung von 2-(Thienyl-3 -amino)-1,3-diazacycloalkenen-(2)
CH1214570A CH555358A (de)	1969-08-13	1970-08-13	Verfahren zur herstellung von 2-(thienyl-3'-amino)-1,3diazacycloalkenen-(2).

Family Applications Before (2)

Application Number	Title	Priority Date	Filing Date
CH1215970A CH530415A (de)	1969-08-13	1970-08-13	Verfahren zur Herstellung von Pyrimidinderivaten
CH611573A CH554894A (de)	1969-08-13	1970-08-13	Verfahren zur herstellung von 2-(thienyl-3'-amino)-1,3diazacycloalkenen-(2).

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
CH1214570A CH555358A (de)	1969-08-13	1970-08-13	Verfahren zur herstellung von 2-(thienyl-3'-amino)-1,3diazacycloalkenen-(2).

Country Status (10)

Country	Link
US (2)	US3758476A (de)
AT (3)	AT310158B (de)
BE (2)	BE754935A (de)
CA (1)	CA1011738A (de)
CH (4)	CH530415A (de)
DE (1)	DE1941575A1 (de)
FR (2)	FR2068493B2 (de)
GB (2)	GB1324646A (de)
NL (2)	NL164859C (de)
SE (1)	SE368406B (de)

Families Citing this family (34)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4036972A (en) *	1973-02-23	1977-07-19	Boehringer Ingelheim Gmbh	2-(N-thienylmethyl-phenylamino)-imidazolines-(2) and salts thereof
DE2308883C3 (de) *	1973-02-23	1978-05-24	C.H. Boehringer Sohn, 6507 Ingelheim	2-Phenylamino-thienylmethyl-imidazoline-(2), Verfahren zur Herstellung derselben und diese enthaltene Arzneimittel
US3919225A (en) *	1974-04-26	1975-11-11	Universal Oil Prod Co	Preparation of N-vinyl substituted amidines
US3919231A (en) *	1974-06-17	1975-11-11	Morton Norwich Products Inc	Series of 5-aryl-2-furamidines
US3970648A (en) *	1974-09-06	1976-07-20	Diamond Shamrock Corporation	2-[2-(5-Nitro-2-furyl)vinyl]-4-(anilino)quinazolines
US4379926A (en) *	1978-05-08	1983-04-12	Ayerst, Mckenna & Harrison Ltd.	1,4,5,6-Tetrahydropyrimidine derivatives
EP0086428B1 (de) *	1979-08-23	1987-07-29	Beecham Group Plc	Veterinärmittel gegen Diarrhöe, seine Herstellung und dieses enthaltende orale Dosierungsvorrichtung
DE19514579A1 (de) *	1995-04-20	1996-10-24	Boehringer Ingelheim Kg	Verwendung von alpha¶1¶¶L¶-Agonisten zur Behandlung der Harninkontinenz
US7049333B2 (en) *	2002-06-04	2006-05-23	Sanofi-Aventis Deutschland Gmbh	Substituted thiophenes: compositions, processes of making, and uses in disease treatment and diagnosis
DE10224892A1 (de) *	2002-06-04	2003-12-18	Aventis Pharma Gmbh	Substituierte Thiophene, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament
US7763280B2 (en) *	2002-11-28	2010-07-27	Boehringer Ingelheim Pharma Gmbh & Co. Kg	Tiotropium containing powder formulation for inhalation
DE10341240A1 (de)	2003-09-08	2005-04-07	Aventis Pharma Deutschland Gmbh	Substituierte Thienoimidazole, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament
EP1797087A4 (de) *	2004-09-23	2009-06-03	Ulysses Pharmaceutical Product	Carbo- und heterocyclische antibiotika und deren anwendung
BRPI0707308A2 (pt) *	2006-01-27	2011-05-03	Hoffmann La Roche	uso de 2-imidazóis para o tratamento de distúrbios do snc
BRPI0717939A2 (pt) *	2006-10-19	2013-12-03	Hoffmann La Roche	Aminometil-4-imidazóis
CA2665255A1 (en) *	2006-10-19	2008-04-24	F. Hoffmann-La Roche Ag	Aminomethyl-2-imidazoles with affinity with the trace amine associated receptors
BRPI0718054A2 (pt) *	2006-11-02	2013-11-05	Hoffmann La Roche	2-imidazóis substituídos como moduladores de receptores associados à traços de aminas
JP2010510184A (ja) *	2006-11-16	2010-04-02	エフ．ホフマン−ラロシュアーゲー	置換４−イミダゾール類
BRPI0720047A2 (pt) *	2006-12-13	2013-12-24	Hoffmann La Roche	2-imidazóis como ligantes para receptores associados a aminas de traço (taar)
US20080146523A1 (en) *	2006-12-18	2008-06-19	Guido Galley	Imidazole derivatives
RU2473545C2 (ru) *	2007-02-02	2013-01-27	Ф.Хоффманн-Ля Рош Аг	Новые 2-аминооксазолины в качестве лигандов taar1 для заболеваний цнс
KR101222412B1 (ko)	2007-02-15	2013-01-15	에프. 호프만-라 로슈 아게	Ｔａａｒ1 리간드로서의 2-아미노옥사졸린
CA2691082A1 (en)	2007-07-02	2009-01-08	F. Hoffmann-La Roche Ag	2 -imidazolines having a good affinity to the trace amine associated receptors (taars)
WO2009003867A1 (en) *	2007-07-03	2009-01-08	F. Hoffmann-La Roche Ag	4-imidazolines and their use as antidepressants
AU2008281918A1 (en) *	2007-07-27	2009-02-05	F. Hoffmann-La Roche Ag	2-azetidinemethaneamines and 2-pyrrolidinemethaneamines as TAAR-ligands
JP2010535172A (ja) *	2007-08-02	2010-11-18	エフ．ホフマン−ラロシュアーゲー	Ｃｎｓ障害の処置のためのベンズアミド誘導体の使用
CA2695331A1 (en) *	2007-08-03	2009-02-12	F. Hoffmann-La Roche Ag	Pyridinecarboxamide and benzamide derivatives as taar1 ligands
US8242153B2 (en) *	2008-07-24	2012-08-14	Hoffmann-La Roche Inc.	4,5-dihydro-oxazol-2YL derivatives
JP5547187B2 (ja) *	2008-07-24	2014-07-09	エフ．ホフマン−ラロシュアーゲー	４，５−ジヒドロ−オキサゾール−２−イル誘導体
US20100311798A1 (en) *	2009-06-05	2010-12-09	Decoret Guillaume	2-aminooxazolines as taar1 ligands
US8354441B2 (en) *	2009-11-11	2013-01-15	Hoffmann-La Roche Inc.	Oxazoline derivatives
US9452980B2 (en)	2009-12-22	2016-09-27	Hoffmann-La Roche Inc.	Substituted benzamides
SG11201807516UA (en)	2016-03-17	2018-09-27	Hoffmann La Roche	5-ethyl-4-methyl-pyrazole-3-carboxamide derivative having activity as agonist of taar
CN111686806B (zh) *	2020-05-29	2022-09-30	黑龙江大学	一种聚[2-(3-噻吩基)乙醇]/石墨相氮化碳复合可见光催化剂的制备方法及应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR5402E (fr) *	1905-06-10	1906-03-27	Camille Durey	Compteur automatique de mouvements d'organes chez les etres animés
DE1695849A1 (de) *	1967-06-23	1971-05-13	Schering Ag	Verfahren zur Herstellung neuer Pyrimidinderivate

0
- BE BE754820D patent/BE754820R/xx active
- BE BE754935D patent/BE754935A/xx not_active IP Right Cessation
1969
- 1969-08-13 DE DE19691941575 patent/DE1941575A1/de active Pending
1970
- 1970-08-06 US US00061853A patent/US3758476A/en not_active Expired - Lifetime
- 1970-08-07 NL NL7011708.A patent/NL164859C/xx not_active IP Right Cessation
- 1970-08-12 FR FR7029657A patent/FR2068493B2/fr not_active Expired
- 1970-08-12 US US00063336A patent/US3814758A/en not_active Expired - Lifetime
- 1970-08-12 NL NL7011933A patent/NL7011933A/xx unknown
- 1970-08-13 GB GB3899770A patent/GB1324646A/en not_active Expired
- 1970-08-13 CH CH1215970A patent/CH530415A/de not_active IP Right Cessation
- 1970-08-13 CH CH611573A patent/CH554894A/de not_active IP Right Cessation
- 1970-08-13 CH CH611473A patent/CH544116A/de not_active IP Right Cessation
- 1970-08-13 CH CH1214570A patent/CH555358A/de not_active IP Right Cessation
- 1970-08-14 AT AT167772A patent/AT310158B/de not_active IP Right Cessation
- 1970-08-14 GB GB3930370A patent/GB1312133A/en not_active Expired
- 1970-08-14 AT AT741970A patent/AT304535B/de not_active IP Right Cessation
- 1970-08-14 CA CA090,785A patent/CA1011738A/en not_active Expired
- 1970-08-14 AT AT167672A patent/AT310157B/de not_active IP Right Cessation
- 1970-08-14 SE SE11112/70A patent/SE368406B/xx unknown
- 1970-08-17 FR FR707030143A patent/FR2068505B1/fr not_active Expired

Also Published As

Publication number	Publication date
NL7011708A (de)	1971-02-18
BE754820R (fr)	1971-02-15
US3758476A (en)	1973-09-11
NL164859B (nl)	1980-09-15
DE1941761A1 (de)	1971-02-25
GB1312133A (en)	1973-04-04
AT304535B (de)	1973-01-10
AT310157B (de)	1973-09-25
US3814758A (en)	1974-06-04
DE1941575A1 (de)	1971-03-04
DE1941761B2 (de)	1976-01-08
FR2068493B2 (de)	1973-12-21
FR2068505B1 (de)	1973-08-10
NL164859C (nl)	1981-02-16
CH554894A (de)	1974-10-15
CH530415A (de)	1972-11-15
CA1011738A (en)	1977-06-07
CH555358A (de)	1974-10-31
FR2068505A1 (de)	1971-08-27
AT310158B (de)	1973-09-25
GB1324646A (en)	1973-07-25
SE368406B (de)	1974-07-01
BE754935A (fr)	1971-02-17
NL7011933A (de)	1971-02-16
FR2068493A2 (de)	1971-08-27

Publication	Publication Date	Title
CH544116A (de)	1973-12-28	Verfahren zur Herstellung von 2-(Thienyl-3 -amino)-1,3-diazacycloalkenen-(2)
AT299142B (de)	1972-06-12	Verfahren zur Herstellung von 2,2-Dimethylpropandiol-(1,3)
CH525183A (de)	1972-07-15	Verfahren zur Herstellung von 3,4-Dihydronaphthalino-noxy-2-hydroxypropylaminen
CH532611A (de)	1973-01-15	Verfahren zur Herstellung von 4 ,a-1 -Demethyl-7-halogen-7-desoxy-lincomycinen
CH550176A (de)	1974-06-14	Verfahren zur herstellung von substituierten n-aminoalkylarylamino-imidazolinen-(2).
CH526618A (de)	1972-08-15	Verfahren zur Herstellung von 1,3,2-Oxazaboriniden
CH553181A (de)	1974-08-30	Verfahren zur herstellung von 4-heterosubstituierten azetidinonen-(2).
CH542801A (de)	1973-10-15	Verfahren zur Herstellung von 1,1-Dihydroperfluoralkanolen
CH531523A (de)	1972-12-15	Verfahren zur Herstellung von 2,6-Dichlor-4-heterocyclyl-pyridin-3,5-dicarbonitrilen
CH529083A (de)	1972-10-15	Verfahren zur Herstellung von Tricyclo-(4,3,1,13,8)-undecan-4-on
AT287665B (de)	1971-02-10	Verfahren zur Herstellung von 2,2-Dimethyl-3-hydroxypropanal
CH527185A (de)	1972-08-31	Verfahren zur Herstellung von 6,7-Dihydro-5H-pyrrolizinen
CH517110A (de)	1971-12-31	Verfahren zur Herstellung von 2,1,3-Benzothiadiazolen
CH539015A (de)	1973-07-15	Verfahren zur Herstellung von 1,3-Diacetoxy-2-methylen-propan
CH524556A (de)	1972-06-30	Verfahren zur Herstellung von 2,3,6-Trimethylhydrochinon
CH520143A (de)	1972-03-15	Verfahren zur Herstellung von 4,5,6,7-Tetrahydrobenzimidazolen
CH537968A (de)	1973-06-15	Verfahren zur Herstellung von 2,2'-Diacylamino-1,1'-dianthrachinonylen
CH516564A (de)	1971-12-15	Verfahren zur Herstellung von 4,5,6-Tri-chlorpyrimidinen
CH535760A (de)	1973-04-15	Verfahren zur Herstellung von 4,5,6,7-Tetrahydro-cyclopenta-1,3-dioxinonen-(4)
CH536854A (de)	1973-05-15	Verfahren zur Herstellung von 6,7 Methylendioxycinnolin-3-carbonitrilen
CH532572A (de)	1973-01-15	Verfahren zur Herstellung von 2,5-Diphenylpyrrolen
CH514568A (de)	1971-10-31	Verfahren zur Herstellung von 6,7-Epoxy-citronellal
CH515253A (de)	1971-11-15	Verfahren zur Herstellung von 2,4-Diamino-6-alkylthio-s-triazinen
CH528537A (de)	1972-09-30	Verfahren zur Herstellung von 3-(1,2,4-Triazolyl-(1))-7-aryltriazolyl-cumarinen
CH517088A (de)	1971-12-31	Verfahren zur Herstellung von 3B,14BB-Dihydroxy-carda-4,20(22)-dienoliden

Legal Events

Date	Code	Title	Description
1989-04-28	PL	Patent ceased