CH460792A - Verfahren zur Herstellung von Benzodiazepinderivaten - Google Patents
Verfahren zur Herstellung von BenzodiazepinderivatenInfo
- Publication number
- CH460792A CH460792A CH1330467A CH1330467A CH460792A CH 460792 A CH460792 A CH 460792A CH 1330467 A CH1330467 A CH 1330467A CH 1330467 A CH1330467 A CH 1330467A CH 460792 A CH460792 A CH 460792A
- Authority
- CH
- Switzerland
- Prior art keywords
- preparation
- benzodiazepine derivatives
- benzodiazepine
- derivatives
- Prior art date
Links
- 229940053197 benzodiazepine derivative antiepileptics Drugs 0.000 title 1
- 125000003310 benzodiazepinyl group Chemical class N1N=C(C=CC2=C1C=CC=C2)* 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
- C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms
-
- F—MECHANICAL ENGINEERING; LIGHTING; HEATING; WEAPONS; BLASTING
- F27—FURNACES; KILNS; OVENS; RETORTS
- F27D—DETAILS OR ACCESSORIES OF FURNACES, KILNS, OVENS OR RETORTS, IN SO FAR AS THEY ARE OF KINDS OCCURRING IN MORE THAN ONE KIND OF FURNACE
- F27D11/00—Arrangement of elements for electric heating in or on furnaces
- F27D11/08—Heating by electric discharge, e.g. arc discharge
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2603/00—Systems containing at least three condensed rings
- C07C2603/02—Ortho- or ortho- and peri-condensed systems
- C07C2603/04—Ortho- or ortho- and peri-condensed systems containing three rings
- C07C2603/06—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members
- C07C2603/10—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings
- C07C2603/12—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings only one five-membered ring
- C07C2603/18—Fluorenes; Hydrogenated fluorenes
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P10/00—Technologies related to metal processing
- Y02P10/10—Reduction of greenhouse gas [GHG] emissions
- Y02P10/143—Reduction of greenhouse gas [GHG] emissions of methane [CH4]
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Mechanical Engineering (AREA)
- General Engineering & Computer Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyridine Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (6)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US8828561A | 1961-02-10 | 1961-02-10 | |
US11530961A | 1961-06-07 | 1961-06-07 | |
US33986164A | 1964-01-24 | 1964-01-24 | |
US412335A US3262938A (en) | 1961-02-10 | 1964-11-19 | Carbocyclic substituted piperidyl dioxolanes |
US412325A US3215688A (en) | 1961-02-10 | 1964-11-19 | Certain benzodiazepine compounds |
US416602A US3256289A (en) | 1961-02-10 | 1964-12-07 | Carbocyclic substituted piperidyl dioxanes |
Publications (1)
Publication Number | Publication Date |
---|---|
CH460792A true CH460792A (de) | 1968-08-15 |
Family
ID=27557343
Family Applications (5)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CH166162A CH405310A (de) | 1961-02-10 | 1962-02-10 | Verfahren zur Herstellung neuer Dioxolane bzw. Dioxane |
CH1687064A CH446360A (de) | 1961-02-10 | 1964-12-30 | Verfahren zur Herstellung von Benzodiazepinderivaten |
CH1330467A CH460792A (de) | 1961-02-10 | 1964-12-30 | Verfahren zur Herstellung von Benzodiazepinderivaten |
CH962768A CH460794A (de) | 1961-02-10 | 1964-12-30 | Verfahren zur Herstellung von Benzodiazepinderivaten |
CH1585965A CH460774A (de) | 1961-02-10 | 1965-11-17 | Verfahren zur Herstellung neuer N-Aralkyl-piperidyl-1,3-dioxolane |
Family Applications Before (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CH166162A CH405310A (de) | 1961-02-10 | 1962-02-10 | Verfahren zur Herstellung neuer Dioxolane bzw. Dioxane |
CH1687064A CH446360A (de) | 1961-02-10 | 1964-12-30 | Verfahren zur Herstellung von Benzodiazepinderivaten |
Family Applications After (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CH962768A CH460794A (de) | 1961-02-10 | 1964-12-30 | Verfahren zur Herstellung von Benzodiazepinderivaten |
CH1585965A CH460774A (de) | 1961-02-10 | 1965-11-17 | Verfahren zur Herstellung neuer N-Aralkyl-piperidyl-1,3-dioxolane |
Country Status (10)
Country | Link |
---|---|
US (3) | US3215688A (de) |
BE (2) | BE658797A (de) |
CH (5) | CH405310A (de) |
DE (3) | DE1545929A1 (de) |
FR (3) | FR1812M (de) |
GB (3) | GB971661A (de) |
IL (1) | IL22721A (de) |
NL (1) | NL141780B (de) |
NO (1) | NO117366B (de) |
SE (3) | SE335135B (de) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BE661945A (de) * | 1964-04-01 | |||
US3464997A (en) * | 1966-03-17 | 1969-09-02 | Us Army | Synthesis of 3-quinuclidinol |
US3760077A (en) * | 1969-02-18 | 1973-09-18 | Cutter Lab | Injectable compositions of the (plus)-optical isomer of the alpha racemate of 2-(2-ethyl-2-phenyl-1, -dioxolan-4-yl)piperidine and their use |
US3856963A (en) * | 1971-10-15 | 1974-12-24 | Cutter Lab | Use of injectable compositions of the ({30 )-optional isomer of the alpha racemate of 2-(2-ethyl-2-phenyl-1,3-dioxolan-4-yl) piperidine to control pain |
US3879406A (en) * | 1972-07-13 | 1975-04-22 | Hoffmann La Roche | Preparation of triazolobenzodiazepines |
US4044016A (en) * | 1975-01-13 | 1977-08-23 | Hoffmann-La Roche Inc. | Preparation of triazolo benzodiazepines and novel compounds |
DE19714041A1 (de) * | 1997-04-05 | 1998-10-08 | Henkel Kgaa | Phenonenketale |
WO2006015683A1 (en) * | 2004-08-10 | 2006-02-16 | Merck Patent Gmbh | Liquid crystal compounds, liquid crystal medium and liquid crystal display |
JP2008510742A (ja) * | 2004-08-24 | 2008-04-10 | ビーエーエスエフ ソシエタス・ヨーロピア | 高純度の第4級アンモニウム化合物の製造方法 |
JP2008001596A (ja) * | 2004-09-03 | 2008-01-10 | Astellas Pharma Inc | ナトリウムチャネル阻害剤 |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2606909A (en) * | 1947-08-01 | 1952-08-12 | Univ Michigan | Basic dioxolanes |
US2606907A (en) * | 1949-08-04 | 1952-08-12 | Univ Michigan | Basic dioxanes |
DE1099540B (de) * | 1954-09-10 | 1961-02-16 | Bayer Ag | Verfahren zur Herstellung von Kondensationsprodukten |
FR1186192A (fr) * | 1957-02-26 | 1959-08-17 | Rhone Poulenc Sa | Nouveaux pipéridyl-2 dioxolannes et leur préparation |
US3070596A (en) * | 1959-03-23 | 1962-12-25 | Aerojet General Co | 1, 1'-biaziridine compounds and the process of preparation |
US3121103A (en) * | 1961-10-20 | 1964-02-11 | Hoffmann La Roche | Aminobenzophenones |
-
0
- BE BE412325D patent/BE412325A/xx unknown
-
1962
- 1962-01-23 GB GB2462/62A patent/GB971661A/en not_active Expired
- 1962-02-07 FR FR887227A patent/FR1812M/fr active Active
- 1962-02-10 CH CH166162A patent/CH405310A/de unknown
- 1962-04-27 FR FR895864A patent/FR1818M/fr active Active
-
1964
- 1964-11-19 US US412325A patent/US3215688A/en not_active Expired - Lifetime
- 1964-11-19 US US412335A patent/US3262938A/en not_active Expired - Lifetime
- 1964-12-07 US US416602A patent/US3256289A/en not_active Expired - Lifetime
- 1964-12-30 CH CH1687064A patent/CH446360A/de unknown
- 1964-12-30 CH CH1330467A patent/CH460792A/de unknown
- 1964-12-30 CH CH962768A patent/CH460794A/de unknown
-
1965
- 1965-01-04 DE DE19651545929 patent/DE1545929A1/de active Pending
- 1965-01-04 IL IL22721A patent/IL22721A/en unknown
- 1965-01-18 NL NL656500594A patent/NL141780B/xx unknown
- 1965-01-21 GB GB2614/65A patent/GB1043049A/en not_active Expired
- 1965-01-22 SE SE18131/67A patent/SE335135B/xx unknown
- 1965-01-22 FR FR2857A patent/FR4166M/fr not_active Expired
- 1965-01-22 SE SE18130/67A patent/SE335134B/xx unknown
- 1965-01-22 SE SE857/65A patent/SE315595B/xx unknown
- 1965-01-23 NO NO65156482A patent/NO117366B/no unknown
- 1965-01-25 BE BE658797D patent/BE658797A/xx unknown
- 1965-11-11 GB GB47936/65A patent/GB1077800A/en not_active Expired
- 1965-11-17 DE DE19651545714 patent/DE1545714A1/de active Pending
- 1965-11-17 DE DE19651545713 patent/DE1545713A1/de active Pending
- 1965-11-17 CH CH1585965A patent/CH460774A/de unknown
Also Published As
Publication number | Publication date |
---|---|
GB1077800A (en) | 1967-08-02 |
DE1545713A1 (de) | 1969-12-18 |
NO117366B (de) | 1969-08-04 |
NL141780B (nl) | 1974-04-16 |
FR1818M (de) | 1963-05-13 |
US3256289A (en) | 1966-06-14 |
CH460774A (de) | 1968-08-15 |
CH446360A (de) | 1967-11-15 |
DE1545929A1 (de) | 1969-12-18 |
US3215688A (en) | 1965-11-02 |
GB1043049A (en) | 1966-09-21 |
US3262938A (en) | 1966-07-26 |
DE1445558B2 (de) | 1975-06-05 |
SE315595B (de) | 1969-10-06 |
FR1812M (de) | 1963-05-13 |
CH460794A (de) | 1968-08-15 |
FR4166M (de) | 1966-05-16 |
BE658797A (de) | 1965-07-26 |
DE1545714A1 (de) | 1969-06-26 |
GB971661A (en) | 1964-09-30 |
SE335135B (de) | 1971-05-17 |
BE412325A (de) | 1900-01-01 |
NL6500594A (de) | 1965-07-26 |
IL22721A (en) | 1968-09-26 |
DE1445558A1 (de) | 1972-04-20 |
SE335134B (de) | 1971-05-17 |
CH405310A (de) | 1966-01-15 |
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