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BR112014027231A2 - comprimido contendo 5-hidróxi-1h-imidazola-4-carboxamida - Google Patents

comprimido contendo 5-hidróxi-1h-imidazola-4-carboxamida

Info

Publication number
BR112014027231A2
BR112014027231A2 BR112014027231A BR112014027231A BR112014027231A2 BR 112014027231 A2 BR112014027231 A2 BR 112014027231A2 BR 112014027231 A BR112014027231 A BR 112014027231A BR 112014027231 A BR112014027231 A BR 112014027231A BR 112014027231 A2 BR112014027231 A2 BR 112014027231A2
Authority
BR
Brazil
Prior art keywords
carboxamide
imidazole
hydroxy
tablet containing
tablet
Prior art date
Application number
BR112014027231A
Other languages
English (en)
Inventor
Yamasaki Yasuomi
Original Assignee
Fujifilm Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fujifilm Corp filed Critical Fujifilm Corp
Publication of BR112014027231A2 publication Critical patent/BR112014027231A2/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2095Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2009Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Inorganic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

resumo “comprimido contendo 5-hidróxi-1h-imidazola-4-carboxamida” trata-se de um comprimido contendo (1) 5-hidróxi-1h-imidazola-4-carboxamida, um sal, ou um hidrato da mesma, e (2) dióxido de silício, em que o teor de 5-hidróxi-1h-imidazola-4-carboxamida, sal, ou hidrato da mesma é alto. o comprimido tem um tamanho que torna fácil a ação de tomar o mesmo, e é excelente em termos de capacidade de liberação.
BR112014027231A 2013-01-15 2014-01-15 comprimido contendo 5-hidróxi-1h-imidazola-4-carboxamida BR112014027231A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2013004995 2013-01-15
PCT/JP2014/050591 WO2014112530A1 (ja) 2013-01-15 2014-01-15 5-ヒドロキシ-1h-イミダゾール-4-カルボキサミドを含有する錠剤

Publications (1)

Publication Number Publication Date
BR112014027231A2 true BR112014027231A2 (pt) 2017-06-27

Family

ID=51209619

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112014027231A BR112014027231A2 (pt) 2013-01-15 2014-01-15 comprimido contendo 5-hidróxi-1h-imidazola-4-carboxamida

Country Status (17)

Country Link
US (1) US9248102B2 (pt)
EP (1) EP2946780B1 (pt)
JP (1) JP5805891B2 (pt)
CN (1) CN104271134B (pt)
BR (1) BR112014027231A2 (pt)
CY (1) CY1119159T1 (pt)
DK (1) DK2946780T3 (pt)
ES (1) ES2622568T3 (pt)
HR (1) HRP20170571T1 (pt)
LT (1) LT2946780T (pt)
PL (1) PL2946780T3 (pt)
PT (1) PT2946780T (pt)
RS (1) RS56032B1 (pt)
RU (1) RU2654703C2 (pt)
SI (1) SI2946780T1 (pt)
SM (1) SMT201700220T1 (pt)
WO (1) WO2014112530A1 (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2937365C (en) 2016-03-29 2018-09-18 F. Hoffmann-La Roche Ag Granulate formulation of 5-methyl-1-phenyl-2-(1h)-pyridone and method of making the same
WO2018051971A1 (ja) * 2016-09-13 2018-03-22 富士フイルム株式会社 Mll関連白血病の予防または治療のための医薬、方法、使用及び化合物
WO2019082898A1 (ja) 2017-10-27 2019-05-02 富士フイルム株式会社 5-ヒドロキシ-1h-イミダゾール-4-カルボキサミド・3/4水和物の製造方法
RU2018134165A (ru) * 2018-09-03 2020-04-01 Фуджифилм Корпорэйшн Комбинированное фармацевтическое, профилактическое или супрессивное средство для подавления резистентности к пиримидиновому антиметаболиту и способ лечения заболевания

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS604802B2 (ja) 1976-09-07 1985-02-06 住友化学工業株式会社 制癌剤
US4181731A (en) * 1976-09-07 1980-01-01 Sumitomo Chemical Company, Limited Novel therapeutic application of 4-carbamoyl-5-hydroxyimidazole
JPS5824569A (ja) 1981-08-05 1983-02-14 Sumitomo Chem Co Ltd イミダゾ−ル誘導体の精製方法
JPS60185727A (ja) 1984-03-05 1985-09-21 Sumitomo Chem Co Ltd 4−カルバモイルイミダゾリウム−5−オレ−ト製剤の安定化法
JPH048468A (ja) * 1990-04-27 1992-01-13 Sanshin:Kk ワーク研摩機
JPH09208468A (ja) * 1996-02-02 1997-08-12 Dainippon Pharmaceut Co Ltd p−クロロ−N−(2−モルホリノエチル)ベンズアミドを含有する錠剤
WO2006046623A1 (ja) * 2004-10-25 2006-05-04 Japan Tobacco Inc. 溶解性及び安定性の改善された固形製剤及びその製造方法
JP5021210B2 (ja) * 2006-01-16 2012-09-05 エスエス製薬株式会社 圧縮成型製剤
FR2903695B1 (fr) * 2006-07-13 2008-10-24 Merck Sante Soc Par Actions Si Utilisation de derives d'imidazole activateurs de l'ampk, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
JP5266010B2 (ja) 2007-09-14 2013-08-21 富士フイルム株式会社 4−カルバモイル−5−ヒドロキシ−イミダゾール誘導体のスルホン酸塩化合物
PT2407166E (pt) * 2009-03-13 2013-11-25 Toyama Chemical Co Ltd Comprimido e pó granulado que contêm 6-fluoro-3-hidroxi-2-pirazinacarboxamida

Also Published As

Publication number Publication date
JP5805891B2 (ja) 2015-11-10
EP2946780B1 (en) 2017-03-01
PL2946780T3 (pl) 2017-07-31
JPWO2014112530A1 (ja) 2017-01-19
DK2946780T3 (en) 2017-05-08
WO2014112530A1 (ja) 2014-07-24
CY1119159T1 (el) 2018-02-14
RU2654703C2 (ru) 2018-05-22
RS56032B1 (sr) 2017-09-29
CN104271134B (zh) 2016-06-29
SI2946780T1 (sl) 2017-05-31
US20150057324A1 (en) 2015-02-26
US9248102B2 (en) 2016-02-02
LT2946780T (lt) 2017-06-12
SMT201700220T1 (it) 2017-07-18
CN104271134A (zh) 2015-01-07
HRP20170571T1 (hr) 2017-08-11
EP2946780A1 (en) 2015-11-25
ES2622568T3 (es) 2017-07-06
RU2014143976A (ru) 2016-05-27
HK1205463A1 (zh) 2015-12-18
PT2946780T (pt) 2017-04-26
EP2946780A4 (en) 2016-06-08

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Legal Events

Date Code Title Description
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B06U Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette]
B11B Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements