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BR0110287A - Artigos de dosagem sólida e de liberação controlada, processo para a compressão direta de artigos de dosagem sólida, mistura diretamente compressìvel, e, processo para formar a mesma - Google Patents

Artigos de dosagem sólida e de liberação controlada, processo para a compressão direta de artigos de dosagem sólida, mistura diretamente compressìvel, e, processo para formar a mesma

Info

Publication number
BR0110287A
BR0110287A BR0110287-7A BR0110287A BR0110287A BR 0110287 A BR0110287 A BR 0110287A BR 0110287 A BR0110287 A BR 0110287A BR 0110287 A BR0110287 A BR 0110287A
Authority
BR
Brazil
Prior art keywords
articles
solid
release
controlled release
forming
Prior art date
Application number
BR0110287-7A
Other languages
English (en)
Inventor
William R Wilber
Jian-Hwa Guo
Edward S Greenberg
Original Assignee
Noveon Ip Holdings Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Noveon Ip Holdings Corp filed Critical Noveon Ip Holdings Corp
Publication of BR0110287A publication Critical patent/BR0110287A/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

"ARTIGOS DE DOSAGEM SóLIDA E DE LIBERAçãO CONTROLADA, PROCESSO PARA A COMPRESSãO DIRETA DE ARTIGOS DE DOSAGEM SóLIDA, MISTURA DIRETAMENTE COMPRESSìVEL E, PROCESSO PARA FORMAR A MESMA". Artigos de dosagem sólida tais como tabletes farmacêuticos para a liberação controlada de um composto desejado tal como um ingrediente ativo são diretamente comprimidos a partir de uma mistura fluível, compressível do ingrediente ativo, um polímero ou copolímero modificador de reologia, levemente reticulado e um ou mais excipientes. O polímero ou copolímero modificador de reologia é um pó granulado de tamanho de partícula adequado e são, no geral, fabricados a partir de um ou mais ácidos (di)carboxílicos insaturados, semi-éster destes e outros monómeros opcionais.
BR0110287-7A 2000-04-27 2001-04-17 Artigos de dosagem sólida e de liberação controlada, processo para a compressão direta de artigos de dosagem sólida, mistura diretamente compressìvel, e, processo para formar a mesma BR0110287A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US09/559,687 US6623756B1 (en) 2000-04-27 2000-04-27 Directly compressed solid dosage articles
PCT/US2001/012400 WO2001082894A2 (en) 2000-04-27 2001-04-17 Directly compressed solid dosage particles

Publications (1)

Publication Number Publication Date
BR0110287A true BR0110287A (pt) 2003-02-18

Family

ID=24234605

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0110287-7A BR0110287A (pt) 2000-04-27 2001-04-17 Artigos de dosagem sólida e de liberação controlada, processo para a compressão direta de artigos de dosagem sólida, mistura diretamente compressìvel, e, processo para formar a mesma

Country Status (13)

Country Link
US (1) US6623756B1 (pt)
EP (1) EP1276466B1 (pt)
JP (1) JP2003531848A (pt)
CN (1) CN1195498C (pt)
AT (1) ATE255886T1 (pt)
BR (1) BR0110287A (pt)
CA (1) CA2407140A1 (pt)
DE (1) DE60101468T2 (pt)
ES (1) ES2211796T3 (pt)
IL (2) IL152461A0 (pt)
MX (1) MXPA02010437A (pt)
WO (1) WO2001082894A2 (pt)
ZA (1) ZA200208571B (pt)

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US7838032B2 (en) * 2000-04-28 2010-11-23 Reckitt Benckiser Inc. Sustained release of guaifenesin
US8012504B2 (en) * 2000-04-28 2011-09-06 Reckitt Benckiser Inc. Sustained release of guaifenesin combination drugs
US6955821B2 (en) 2000-04-28 2005-10-18 Adams Laboratories, Inc. Sustained release formulations of guaifenesin and additional drug ingredients
US6623754B2 (en) * 2001-05-21 2003-09-23 Noveon Ip Holdings Corp. Dosage form of N-acetyl cysteine
US20030012820A1 (en) * 2001-06-12 2003-01-16 Upadhyay Ajay Hasmukhlal Compressible guaifenesin compositions, method for making same and method for making compressed guaifenesin dosage forms therefrom
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US20040185016A1 (en) * 2002-07-30 2004-09-23 Popp Karl F Compositions for treatment of hyperpigmentation and methods for making and using such compositions
US20040219210A1 (en) * 2003-05-01 2004-11-04 Jian-Hwa Guo Controlled release solid dosage nifedipine formulations
US20050202079A1 (en) * 2004-03-15 2005-09-15 Mylan Pharmaceuticals Inc. Novel orally administrable formulation of nitrofurantoin and a method for preparing said formulation
US7704522B2 (en) 2004-09-08 2010-04-27 Clyde Morgan Topical medicament
US20070077297A1 (en) 2004-09-30 2007-04-05 Scolr Pharma, Inc. Modified release ibuprofen dosage form
FI20080353A0 (fi) * 2008-05-09 2008-05-09 Atacama Labs Oy Prosessi erittäin korkean lääkepitoisuuden tabletin valmistamiseksi
FI20080355A0 (fi) * 2008-05-09 2008-05-09 Atacama Labs Oy Prosessi metforminia käsittävien tablettien valmistamiseksi
FI20080346A0 (fi) * 2008-05-09 2008-05-09 Atacama Labs Oy Prosessi lisäaineita sisältävän tabletin valmistamiseksi
US7749537B2 (en) * 2006-12-04 2010-07-06 Scolr Pharma, Inc. Method of forming a tablet
CN101467988B (zh) * 2007-12-27 2014-07-09 北京德众万全医药科技有限公司 一种含有氨酚伪麻的药用组合物及其制备方法
WO2010071577A1 (en) * 2008-12-17 2010-06-24 Astrazeneca Ab Method of providing a target dose, powder provider device and its use
EP2461811B1 (en) 2009-08-05 2016-04-20 Idenix Pharmaceuticals LLC. Macrocyclic serine protease inhibitors useful against viral infections, particularly hcv
WO2011056764A1 (en) 2009-11-05 2011-05-12 Ambit Biosciences Corp. Isotopically enriched or fluorinated imidazo[2,1-b][1,3]benzothiazoles
AU2010330862B2 (en) 2009-12-18 2015-06-25 Idenix Pharmaceuticals, Inc. 5,5-fused arylene or heteroarylene hepatitis C virus inhibitors
WO2011094890A1 (en) 2010-02-02 2011-08-11 Argusina Inc. Phenylalanine derivatives and their use as non-peptide glp-1 receptor modulators
WO2011112689A2 (en) 2010-03-11 2011-09-15 Ambit Biosciences Corp. Saltz of an indazolylpyrrolotriazine
ES2619850T3 (es) 2010-09-01 2017-06-27 Ambit Biosciences Corporation Sales de hidrobromuro de una pirazolilaminoquinazolina
JP5932794B2 (ja) 2010-09-01 2016-06-08 アムビト ビオスシエンセス コルポラチオン 光学活性のあるピラゾリルアミノキナゾリン及びその医薬組成物及び使用方法
CA2819859A1 (en) 2010-12-06 2012-06-14 Follica, Inc. Methods for treating baldness and promoting hair growth
WO2012080050A1 (en) 2010-12-14 2012-06-21 F. Hoffmann-La Roche Ag Solid forms of a phenoxybenzenesulfonyl compound
JP2014503597A (ja) 2011-01-31 2014-02-13 セルジーン コーポレイション シチジンアナログの医薬組成物及びその使用方法
AR085352A1 (es) 2011-02-10 2013-09-25 Idenix Pharmaceuticals Inc Inhibidores macrociclicos de serina proteasa, sus composiciones farmaceuticas y su uso para tratar infecciones por hcv
US20120252721A1 (en) 2011-03-31 2012-10-04 Idenix Pharmaceuticals, Inc. Methods for treating drug-resistant hepatitis c virus infection with a 5,5-fused arylene or heteroarylene hepatitis c virus inhibitor
AR092809A1 (es) 2012-03-16 2015-05-06 Axikin Pharmaceuticals Inc 3,5-diaminopirazol como inhibidor de quinasa
NZ631142A (en) 2013-09-18 2016-03-31 Axikin Pharmaceuticals Inc Pharmaceutically acceptable salts of 3,5-diaminopyrazole kinase inhibitors
EP3046924A1 (en) 2013-09-20 2016-07-27 IDENIX Pharmaceuticals, Inc. Hepatitis c virus inhibitors
US20170066779A1 (en) 2014-03-05 2017-03-09 Idenix Pharmaceuticals Llc Solid forms of a flaviviridae virus inhibitor compound and salts thereof
CN106536506A (zh) 2014-03-20 2017-03-22 卡佩拉医疗公司 苯并咪唑衍生物作为erbb酪氨酸激酶抑制剂用于治疗癌症
KR102409739B1 (ko) 2014-03-20 2022-06-17 카펠라 테라퓨틱스, 인크. 암 치료용의 ｅｒｂｂ 티로신 키나제 억제제로서의 벤즈이미다졸 유도체
AR103264A1 (es) 2014-12-23 2017-04-26 Axikin Pharmaceuticals Inc Derivados de 3,5-aminopirazol como inhibidores de quinasa rc
EP3364955B1 (en) 2015-10-09 2022-04-20 RB Health (US) LLC Pharmaceutical formulation
WO2020152304A1 (en) 2019-01-24 2020-07-30 Novo Nordisk A/S Roller compactor and method of dry granulation using a roller compactor
WO2021043971A1 (en) 2019-09-06 2021-03-11 Novo Nordisk A/S Method and equipment for fractionation of granules for use in pharmaceutical compositions

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US4267103A (en) * 1978-12-07 1981-05-12 The B. F. Goodrich Company Solvent polymerization of carboxyl containing monomers
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US5288814A (en) * 1992-08-26 1994-02-22 The B. F. Goodrich Company Easy to disperse polycarboxylic acid thickeners
US5780055A (en) * 1996-09-06 1998-07-14 University Of Maryland, Baltimore Cushioning beads and tablet comprising the same capable of forming a suspension

Also Published As

Publication number Publication date
WO2001082894A3 (en) 2002-02-21
DE60101468D1 (de) 2004-01-22
IL152461A0 (en) 2003-05-29
IL152461A (en) 2007-08-19
MXPA02010437A (es) 2003-04-25
CA2407140A1 (en) 2001-11-08
CN1426297A (zh) 2003-06-25
ATE255886T1 (de) 2003-12-15
EP1276466A2 (en) 2003-01-22
EP1276466B1 (en) 2003-12-10
US6623756B1 (en) 2003-09-23
WO2001082894A2 (en) 2001-11-08
ZA200208571B (en) 2003-08-19
CN1195498C (zh) 2005-04-06
JP2003531848A (ja) 2003-10-28
DE60101468T2 (de) 2004-10-28
ES2211796T3 (es) 2004-07-16

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Owner name: NOVEON, INC. (US)

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B25D Requested change of name of applicant approved

Owner name: LUBRIZOL ADVANCED MATERIALS, INC. (US)

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B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B15K Others concerning applications: alteration of classification

Free format text: PARA INT.CL.: A61K 9/16, A61K 9/00

Ipc: A61K 9/16 (2010.01), A61K 9/00 (2010.01)

B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: INDEFIRO O PEDIDO DE ACORDO COM O(S) ARTIGO(S) 8O, 11, 13 E 25 DA LPI

B15K Others concerning applications: alteration of classification

Free format text: PARA:INT.CI 461K 9/16; A61K 9/00; A61P 29/00; A61P 11/11

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B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: MANTIDO O INDEFERIMENTO UMA VEZ QUE NAO FOI APRESENTADO RECURSO DENTRO DO PRAZO LEGAL.