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BG98887A - Халогениране чрез използване на халогенен реагент на вилсмайер - Google Patents

Халогениране чрез използване на халогенен реагент на вилсмайер Download PDF

Info

Publication number
BG98887A
BG98887A BG98887A BG9888794A BG98887A BG 98887 A BG98887 A BG 98887A BG 98887 A BG98887 A BG 98887A BG 9888794 A BG9888794 A BG 9888794A BG 98887 A BG98887 A BG 98887A
Authority
BG
Bulgaria
Prior art keywords
reagent
wilsmeier
halogen
chloride
bromide
Prior art date
Application number
BG98887A
Other languages
Bulgarian (bg)
English (en)
Inventor
Neil Baine
Donald Klein
Richard Mewshaw
Lillian Owings
Original Assignee
Smithkline Beecham Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Corporation filed Critical Smithkline Beecham Corporation
Publication of BG98887A publication Critical patent/BG98887A/bg

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J9/00Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J43/00Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J3/00Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
    • C07J3/005Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom the carbon atom being part of a carboxylic function
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0066Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the 17-beta position being substituted by a carbon atom forming part of an amide group

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BG98887A 1992-01-06 1994-07-05 Халогениране чрез използване на халогенен реагент на вилсмайер BG98887A (bg)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US81717992A 1992-01-06 1992-01-06
US94134892A 1992-09-04 1992-09-04
PCT/US1993/000079 WO1993014106A1 (en) 1992-01-06 1993-01-06 Halogenation using halo-vilsmeier reagent

Publications (1)

Publication Number Publication Date
BG98887A true BG98887A (bg) 1995-05-31

Family

ID=27124147

Family Applications (1)

Application Number Title Priority Date Filing Date
BG98887A BG98887A (bg) 1992-01-06 1994-07-05 Халогениране чрез използване на халогенен реагент на вилсмайер

Country Status (23)

Country Link
EP (1) EP0643723A4 (pt)
JP (1) JPH07505138A (pt)
KR (1) KR940703849A (pt)
CN (1) CN1077201A (pt)
AP (1) AP370A (pt)
AU (1) AU666167B2 (pt)
BG (1) BG98887A (pt)
BR (1) BR9305786A (pt)
CA (1) CA2127272A1 (pt)
CZ (1) CZ161994A3 (pt)
FI (1) FI943214L (pt)
HU (1) HUT68273A (pt)
IL (1) IL104302A (pt)
MA (1) MA22761A1 (pt)
MX (1) MX9300025A (pt)
NO (1) NO942535L (pt)
NZ (1) NZ246788A (pt)
OA (1) OA09961A (pt)
RU (1) RU94038223A (pt)
SI (1) SI9300006A (pt)
SK (1) SK80094A3 (pt)
TW (1) TW300226B (pt)
WO (1) WO1993014106A1 (pt)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5641765A (en) * 1992-11-18 1997-06-24 Smithkline Beecham Corporation 17-αand 17-βsubstituted acyl-3-carboxy-3,5-dienes and use in inhibiting 5-α-reductase
US5683995A (en) * 1992-11-18 1997-11-04 Smithkline Beecham Corporation 17 substituted acyl-3-carboxy 3,5-diene steroidals as α-reductase inhibitors
US8143428B2 (en) 2004-06-08 2012-03-27 Temple University-Of The Commonwealth System Of Higher Education Heteroaryl sulfones and sulfonamides and therapeutic uses thereof

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA883034B (en) * 1987-04-29 1989-03-29 Smithkline Beckman Corp Steroid 5-alpha-reductase inhibitors

Also Published As

Publication number Publication date
FI943214A0 (fi) 1994-07-05
BR9305786A (pt) 1997-02-18
FI943214L (fi) 1994-07-05
OA09961A (en) 1995-12-11
NO942535D0 (no) 1994-07-05
KR940703849A (ko) 1994-12-12
JPH07505138A (ja) 1995-06-08
CA2127272A1 (en) 1993-07-22
HUT68273A (en) 1995-06-28
NZ246788A (en) 1996-11-26
IL104302A0 (en) 1993-05-13
TW300226B (pt) 1997-03-11
SI9300006A (en) 1993-09-30
CN1077201A (zh) 1993-10-13
CZ161994A3 (en) 1995-03-15
NO942535L (no) 1994-07-05
AP370A (en) 1994-11-10
MA22761A1 (fr) 1993-10-01
EP0643723A1 (en) 1995-03-22
EP0643723A4 (en) 1995-05-10
AP9300473A0 (en) 1993-01-31
MX9300025A (es) 1994-01-31
IL104302A (en) 1998-02-22
HU9402030D0 (en) 1994-09-28
WO1993014106A1 (en) 1993-07-22
AU3434893A (en) 1993-08-03
RU94038223A (ru) 1997-04-20
SK80094A3 (en) 1994-12-07
AU666167B2 (en) 1996-02-01

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