[go: up one dir, main page]

BG26526A3 - METHOD FOR THE PREPARATION OF 1-(BENZAZOLYLALKYL)PIPERIDINE DERIVATIVES - Google Patents

METHOD FOR THE PREPARATION OF 1-(BENZAZOLYLALKYL)PIPERIDINE DERIVATIVES

Info

Publication number
BG26526A3
BG26526A3 BG033791A BG3379176A BG26526A3 BG 26526 A3 BG26526 A3 BG 26526A3 BG 033791 A BG033791 A BG 033791A BG 3379176 A BG3379176 A BG 3379176A BG 26526 A3 BG26526 A3 BG 26526A3
Authority
BG
Bulgaria
Prior art keywords
benzazolylalkyl
preparation
piperidine derivatives
piperidine
derivatives
Prior art date
Application number
BG033791A
Other languages
Bulgarian (bg)
Inventor
Jan Vandenberk
Ludo Edmond Kennis
Marcel Van
Albert M.
Original Assignee
Неизвестен
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/687,139 external-priority patent/US4066772A/en
Application filed by Неизвестен filed Critical Неизвестен
Publication of BG26526A3 publication Critical patent/BG26526A3/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56Nitrogen atoms
    • C07D211/58Nitrogen atoms attached in position 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/26Oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Otolaryngology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BG033791A 1975-07-21 1976-07-20 METHOD FOR THE PREPARATION OF 1-(BENZAZOLYLALKYL)PIPERIDINE DERIVATIVES BG26526A3 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US59779375A 1975-07-21 1975-07-21
US05/687,139 US4066772A (en) 1975-07-21 1976-05-17 1,3-Dihydro-1-[3-(1-piperidinyl)propyl]-2H-benzimidazol-2-ones and related compounds
KR7601697A KR810000334B1 (en) 1975-07-21 1976-07-12 Process for preparation 1-(benzazolylalkyl)-piperidine derivatives

Publications (1)

Publication Number Publication Date
BG26526A3 true BG26526A3 (en) 1979-04-12

Family

ID=27348142

Family Applications (1)

Application Number Title Priority Date Filing Date
BG033791A BG26526A3 (en) 1975-07-21 1976-07-20 METHOD FOR THE PREPARATION OF 1-(BENZAZOLYLALKYL)PIPERIDINE DERIVATIVES

Country Status (25)

Country Link
JP (1) JPS5217475A (en)
AT (1) AT364358B (en)
AU (1) AU511027B2 (en)
BG (1) BG26526A3 (en)
CA (1) CA1085852A (en)
CH (1) CH623820A5 (en)
CS (1) CS202550B2 (en)
DE (1) DE2632870A1 (en)
DK (1) DK154950C (en)
ES (3) ES449740A1 (en)
FI (1) FI62667C (en)
GB (1) GB1542514A (en)
HK (1) HK14180A (en)
IE (1) IE43496B1 (en)
IT (1) IT1062614B (en)
KE (1) KE3215A (en)
LU (1) LU75354A1 (en)
MY (1) MY8100017A (en)
NL (1) NL187442C (en)
NZ (1) NZ181256A (en)
PH (1) PH13710A (en)
PT (1) PT65387B (en)
RO (1) RO70566A (en)
SE (2) SE426490B (en)
YU (1) YU39969B (en)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4501749A (en) * 1983-10-31 1985-02-26 Merck & Co., Inc. Peripherally selective dopamine antagonists in the treatment of ocular hypertension
JPS6248684A (en) * 1985-08-26 1987-03-03 Sumitomo Chem Co Ltd Novel iodobutyrophenone derivative and production thereof
JPS62251313A (en) * 1986-04-25 1987-11-02 信越ポリマー株式会社 Bundling device
FR2723091B1 (en) * 1994-07-29 1996-11-08 Esteve Labor Dr TETRAHYDROPYRIDINE- (6,4-HYDROXYPIPERIDINE) ALKYLAZOLES
US6355659B1 (en) 1994-07-29 2002-03-12 Laboratorios Del Dr. Esteve, S.A. 4-(4-Chlorophenyl)-1236-tetrahydro-1(1H-124-triazol-1-yl)butty)pyrideine and salts thereof; pharmaceutical compositions and method of treating psychoses utilizing same
PA8603801A1 (en) * 2003-05-27 2004-12-16 Janssen Pharmaceutica Nv DERIVATIVES OF QUINAZOLINE
CA2549869C (en) 2003-12-18 2015-05-05 Janssen Pharmaceutica N.V. Pyrido- and pyrimidopyrimidine derivatives as anti- proliferative agents
NI200700147A (en) 2004-12-08 2019-05-10 Janssen Pharmaceutica Nv QUINAZOLINE DERIVATIVES KINE INHIBITORS TARGETING MULTIP
CA2654583C (en) 2006-07-13 2015-11-24 Janssen Pharmaceutica N.V. Mtki quinazoline derivatives
EP1997805A1 (en) * 2007-06-01 2008-12-03 Commissariat à l'Energie Atomique Compounds with antiparasitic activity, applications thereof to the treatment of infectious diseases caused by apicomplexans
EP2185562B1 (en) 2007-07-27 2015-12-02 Janssen Pharmaceutica, N.V. Pyrrolopyrimidines useful for the treatment of proliferative diseases
MX2010002449A (en) 2007-08-31 2010-09-07 Purdue Pharma Lp Substituted-quinoxaline-type-piperidine compounds and the uses thereof.
US9090618B2 (en) 2012-12-27 2015-07-28 Purdue Pharma L.P. Substituted benzimidazole-type piperidine compounds and uses thereof
EP3411031B1 (en) * 2016-02-04 2024-07-24 CinDome Pharma, Inc. Deuterated domperidone compositions and methods for therapy of disorders
KR20240125702A (en) 2017-06-30 2024-08-19 신돔 파마, 인크. Deuterated domperidone compositions, methods, and preparation

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE633495A (en) * 1962-06-13
BE633914A (en) * 1962-06-22
US3629267A (en) * 1968-10-28 1971-12-21 Smith Kline French Lab Benzoheterocyclicalkyl derivatives of 4-(2-keto -1-benzimidazolinyl)-piperidine 4-(2-keto - 1 - benzimidazolinyl) -1 2 3 6 tetrahydropyridine 1 - phenyl - 1 3 8-triazaspiro(4 5)decan - 4 - one and 2 4 9-triazaspiro(5 5)undecan-1 3 5-trione
AU4698672A (en) * 1972-09-22 1972-11-09 Ciba-Geigy Ag Azacycloaliphatic compounds, process for their manufacture and compositions containing them
FR2218100A1 (en) * 1973-02-20 1974-09-13 Janssen Pharmaceutica Nv Neuroleptic tricyclic derivs. - of benzimidazolinones and triazaspiro-4,5-decan-4-ones
US3989707A (en) * 1974-06-21 1976-11-02 Janssen Pharmaceutica N.V. Benzimidazolinone derivatives

Also Published As

Publication number Publication date
ES449740A1 (en) 1978-02-16
JPS5217475A (en) 1977-02-09
FI762086A (en) 1977-01-22
CS202550B2 (en) 1981-01-30
RO70566A (en) 1982-10-11
MY8100017A (en) 1981-12-31
AT364358B (en) 1981-10-12
GB1542514A (en) 1979-03-21
ATA534776A (en) 1981-03-15
JPS6131109B2 (en) 1986-07-17
FI62667C (en) 1983-02-10
NL187442B (en) 1991-05-01
SE8008713L (en) 1980-12-11
NL187442C (en) 1991-10-01
SE426490B (en) 1983-01-24
DE2632870C2 (en) 1989-02-16
DK154950C (en) 1989-05-29
DE2632870A1 (en) 1977-02-10
ES461631A1 (en) 1978-12-01
IT1062614B (en) 1984-10-20
DK327576A (en) 1977-01-22
PT65387B (en) 1978-06-09
SE7608265L (en) 1977-01-22
PT65387A (en) 1976-08-01
YU39969B (en) 1985-06-30
NZ181256A (en) 1978-04-28
IE43496L (en) 1977-01-21
PH13710A (en) 1980-09-09
DK154950B (en) 1989-01-09
CA1085852A (en) 1980-09-16
YU179476A (en) 1983-01-21
KE3215A (en) 1982-07-09
IE43496B1 (en) 1981-03-11
NL7608023A (en) 1977-01-25
AU511027B2 (en) 1980-07-24
HK14180A (en) 1980-03-28
SE435621B (en) 1984-10-08
FI62667B (en) 1982-10-29
AU1596476A (en) 1978-01-19
ES461630A1 (en) 1978-06-16
LU75354A1 (en) 1977-02-28
CH623820A5 (en) 1981-06-30

Similar Documents

Publication Publication Date Title
SE437022B (en) PROCEDURE FOR THE PREPARATION OF N-SUBSTITUTED MORPHOLINE DERIVATIVES RESPECTIVE PIPERIDINE DERIVATIVES
SE434049B (en) PROCEDURE FOR PREPARING 1,4-DIHYDROPYRIDINE DERIVATIVES
SE7610940L (en) PROCEDURE FOR THE PREPARATION OF BENZHYDRYL SULFINYL DERIVATIVE
DK115376A (en) KINOLON DERIVATIVES
BG26515A3 (en) METHOD FOR OBTAINING ACYLAMINO DERIVATIVES
ZA764322B (en) Novel 1-(benzazolyalkyl)piperidine derivatives
BG26518A3 (en) METHOD FOR OBTAINING PHENYL-ALKANE DERIVATIVES
BG26526A3 (en) METHOD FOR THE PREPARATION OF 1-(BENZAZOLYLALKYL)PIPERIDINE DERIVATIVES
BG27542A3 (en) METHOD FOR THE PREPARATION OF 1-BENZAZOLYLALKYL-4-SUBSTITUTED PIPERIDINES
PL191647A1 (en) METHOD OF THE PRODUCTION OF THENOPYRIDINE DERIVATIVES
SE433745B (en) PROCEDURE FOR PREPARING TETRAHYDROISOKINOLIN DERIVATIVES
MX4118E (en) PROCEDURE FOR PREPARING PIPERIDINE COMPOUND
SE423390B (en) PROCEDURES FOR PREPARING EBURNAME DERIVATIVES
SE423902B (en) PROCEDURE FOR PURINATE DERIVATIVES
IT1066655B (en) PROCEDURE FOR DEPURING CAPROLATTAME
RO73050A (en) PROCESS FOR PREPARATION OF SUBSTITUTED AMINOCHINESOLINE DERIVATIVES
BG26535A3 (en) METHOD FOR OBTAINING INDOLQUINOLYSINES
SE7709402L (en) PROCEDURE FOR THE PREPARATION OF TETRAHYDROPYRIDINE DERIVATIVES
BG26388A3 (en) METHOD FOR OBTAINING DERIVATIVES OF XANTHENIC ACID
BG26534A4 (en) METHOD FOR OBTAINING 2-METHYL-2-CYANOMETHYL-5-ISOPROPYLTETRAHYDROFURAN
IT1053899B (en) PROCEDURE FOR PRODUCING OR PARAISOPROPENYLPHENOL DERIVATIVES
SE7608519L (en) MORPHANTRIDINE DERIVATIVES
SE435291B (en) PROCEDURE FOR PREPARING 7-ACYLAMINO-3 (1- (2-SULFAMINOETHYL) -TETRAZOL-5-YLTIOMETHYL) -3-CEFEM-4-CARBONIC ACID
DD122967A1 (en) HYLAMIN DERIVATIVES
PL191309A1 (en) METHOD OF MAKING NEW DERIVATIVES 1- (BENZAZOLYL-ALKYL) -PIPERIDINE