BG26526A3 - METHOD FOR THE PREPARATION OF 1-(BENZAZOLYLALKYL)PIPERIDINE DERIVATIVES - Google Patents
METHOD FOR THE PREPARATION OF 1-(BENZAZOLYLALKYL)PIPERIDINE DERIVATIVESInfo
- Publication number
- BG26526A3 BG26526A3 BG033791A BG3379176A BG26526A3 BG 26526 A3 BG26526 A3 BG 26526A3 BG 033791 A BG033791 A BG 033791A BG 3379176 A BG3379176 A BG 3379176A BG 26526 A3 BG26526 A3 BG 26526A3
- Authority
- BG
- Bulgaria
- Prior art keywords
- benzazolylalkyl
- preparation
- piperidine derivatives
- piperidine
- derivatives
- Prior art date
Links
- NQRYJNQNLNOLGT-UHFFFAOYSA-N Piperidine Chemical class C1CCNCC1 NQRYJNQNLNOLGT-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/56—Nitrogen atoms
- C07D211/58—Nitrogen atoms attached in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/26—Oxygen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Hospice & Palliative Care (AREA)
- Pharmacology & Pharmacy (AREA)
- Otolaryngology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US59779375A | 1975-07-21 | 1975-07-21 | |
US05/687,139 US4066772A (en) | 1975-07-21 | 1976-05-17 | 1,3-Dihydro-1-[3-(1-piperidinyl)propyl]-2H-benzimidazol-2-ones and related compounds |
KR7601697A KR810000334B1 (en) | 1975-07-21 | 1976-07-12 | Process for preparation 1-(benzazolylalkyl)-piperidine derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
BG26526A3 true BG26526A3 (en) | 1979-04-12 |
Family
ID=27348142
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BG033791A BG26526A3 (en) | 1975-07-21 | 1976-07-20 | METHOD FOR THE PREPARATION OF 1-(BENZAZOLYLALKYL)PIPERIDINE DERIVATIVES |
Country Status (25)
Country | Link |
---|---|
JP (1) | JPS5217475A (en) |
AT (1) | AT364358B (en) |
AU (1) | AU511027B2 (en) |
BG (1) | BG26526A3 (en) |
CA (1) | CA1085852A (en) |
CH (1) | CH623820A5 (en) |
CS (1) | CS202550B2 (en) |
DE (1) | DE2632870A1 (en) |
DK (1) | DK154950C (en) |
ES (3) | ES449740A1 (en) |
FI (1) | FI62667C (en) |
GB (1) | GB1542514A (en) |
HK (1) | HK14180A (en) |
IE (1) | IE43496B1 (en) |
IT (1) | IT1062614B (en) |
KE (1) | KE3215A (en) |
LU (1) | LU75354A1 (en) |
MY (1) | MY8100017A (en) |
NL (1) | NL187442C (en) |
NZ (1) | NZ181256A (en) |
PH (1) | PH13710A (en) |
PT (1) | PT65387B (en) |
RO (1) | RO70566A (en) |
SE (2) | SE426490B (en) |
YU (1) | YU39969B (en) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4501749A (en) * | 1983-10-31 | 1985-02-26 | Merck & Co., Inc. | Peripherally selective dopamine antagonists in the treatment of ocular hypertension |
JPS6248684A (en) * | 1985-08-26 | 1987-03-03 | Sumitomo Chem Co Ltd | Novel iodobutyrophenone derivative and production thereof |
JPS62251313A (en) * | 1986-04-25 | 1987-11-02 | 信越ポリマー株式会社 | Bundling device |
FR2723091B1 (en) * | 1994-07-29 | 1996-11-08 | Esteve Labor Dr | TETRAHYDROPYRIDINE- (6,4-HYDROXYPIPERIDINE) ALKYLAZOLES |
US6355659B1 (en) | 1994-07-29 | 2002-03-12 | Laboratorios Del Dr. Esteve, S.A. | 4-(4-Chlorophenyl)-1236-tetrahydro-1(1H-124-triazol-1-yl)butty)pyrideine and salts thereof; pharmaceutical compositions and method of treating psychoses utilizing same |
PA8603801A1 (en) * | 2003-05-27 | 2004-12-16 | Janssen Pharmaceutica Nv | DERIVATIVES OF QUINAZOLINE |
CA2549869C (en) | 2003-12-18 | 2015-05-05 | Janssen Pharmaceutica N.V. | Pyrido- and pyrimidopyrimidine derivatives as anti- proliferative agents |
NI200700147A (en) | 2004-12-08 | 2019-05-10 | Janssen Pharmaceutica Nv | QUINAZOLINE DERIVATIVES KINE INHIBITORS TARGETING MULTIP |
CA2654583C (en) | 2006-07-13 | 2015-11-24 | Janssen Pharmaceutica N.V. | Mtki quinazoline derivatives |
EP1997805A1 (en) * | 2007-06-01 | 2008-12-03 | Commissariat à l'Energie Atomique | Compounds with antiparasitic activity, applications thereof to the treatment of infectious diseases caused by apicomplexans |
EP2185562B1 (en) | 2007-07-27 | 2015-12-02 | Janssen Pharmaceutica, N.V. | Pyrrolopyrimidines useful for the treatment of proliferative diseases |
MX2010002449A (en) | 2007-08-31 | 2010-09-07 | Purdue Pharma Lp | Substituted-quinoxaline-type-piperidine compounds and the uses thereof. |
US9090618B2 (en) | 2012-12-27 | 2015-07-28 | Purdue Pharma L.P. | Substituted benzimidazole-type piperidine compounds and uses thereof |
EP3411031B1 (en) * | 2016-02-04 | 2024-07-24 | CinDome Pharma, Inc. | Deuterated domperidone compositions and methods for therapy of disorders |
KR20240125702A (en) | 2017-06-30 | 2024-08-19 | 신돔 파마, 인크. | Deuterated domperidone compositions, methods, and preparation |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BE633495A (en) * | 1962-06-13 | |||
BE633914A (en) * | 1962-06-22 | |||
US3629267A (en) * | 1968-10-28 | 1971-12-21 | Smith Kline French Lab | Benzoheterocyclicalkyl derivatives of 4-(2-keto -1-benzimidazolinyl)-piperidine 4-(2-keto - 1 - benzimidazolinyl) -1 2 3 6 tetrahydropyridine 1 - phenyl - 1 3 8-triazaspiro(4 5)decan - 4 - one and 2 4 9-triazaspiro(5 5)undecan-1 3 5-trione |
AU4698672A (en) * | 1972-09-22 | 1972-11-09 | Ciba-Geigy Ag | Azacycloaliphatic compounds, process for their manufacture and compositions containing them |
FR2218100A1 (en) * | 1973-02-20 | 1974-09-13 | Janssen Pharmaceutica Nv | Neuroleptic tricyclic derivs. - of benzimidazolinones and triazaspiro-4,5-decan-4-ones |
US3989707A (en) * | 1974-06-21 | 1976-11-02 | Janssen Pharmaceutica N.V. | Benzimidazolinone derivatives |
-
1976
- 1976-06-23 NZ NZ181256A patent/NZ181256A/en unknown
- 1976-06-30 GB GB7627242A patent/GB1542514A/en not_active Expired
- 1976-07-07 RO RO7686860A patent/RO70566A/en unknown
- 1976-07-07 CA CA256,450A patent/CA1085852A/en not_active Expired
- 1976-07-08 PH PH18663A patent/PH13710A/en unknown
- 1976-07-09 ES ES449740A patent/ES449740A1/en not_active Expired
- 1976-07-09 LU LU75354A patent/LU75354A1/xx unknown
- 1976-07-16 AU AU15964/76A patent/AU511027B2/en not_active Expired
- 1976-07-16 CS CS764688A patent/CS202550B2/en unknown
- 1976-07-19 IT IT50499/76A patent/IT1062614B/en active
- 1976-07-19 JP JP51085216A patent/JPS5217475A/en active Granted
- 1976-07-20 BG BG033791A patent/BG26526A3/en unknown
- 1976-07-20 PT PT65387A patent/PT65387B/en unknown
- 1976-07-20 SE SE7608265A patent/SE426490B/en not_active IP Right Cessation
- 1976-07-20 AT AT0534776A patent/AT364358B/en not_active IP Right Cessation
- 1976-07-20 IE IE1602/76A patent/IE43496B1/en not_active IP Right Cessation
- 1976-07-20 CH CH929176A patent/CH623820A5/en not_active IP Right Cessation
- 1976-07-20 DK DK327576A patent/DK154950C/en not_active IP Right Cessation
- 1976-07-20 FI FI762086A patent/FI62667C/en not_active IP Right Cessation
- 1976-07-20 NL NLAANVRAGE7608023,A patent/NL187442C/en not_active IP Right Cessation
- 1976-07-21 YU YU1794/76A patent/YU39969B/en unknown
- 1976-07-21 DE DE19762632870 patent/DE2632870A1/en active Granted
-
1977
- 1977-08-16 ES ES461631A patent/ES461631A1/en not_active Expired
- 1977-08-16 ES ES461630A patent/ES461630A1/en not_active Expired
-
1980
- 1980-03-20 HK HK141/80A patent/HK14180A/en unknown
- 1980-12-11 SE SE8008713A patent/SE435621B/en not_active IP Right Cessation
-
1981
- 1981-12-30 MY MY17/81A patent/MY8100017A/en unknown
-
1982
- 1982-05-21 KE KE3215A patent/KE3215A/en unknown
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
SE437022B (en) | PROCEDURE FOR THE PREPARATION OF N-SUBSTITUTED MORPHOLINE DERIVATIVES RESPECTIVE PIPERIDINE DERIVATIVES | |
SE434049B (en) | PROCEDURE FOR PREPARING 1,4-DIHYDROPYRIDINE DERIVATIVES | |
SE7610940L (en) | PROCEDURE FOR THE PREPARATION OF BENZHYDRYL SULFINYL DERIVATIVE | |
DK115376A (en) | KINOLON DERIVATIVES | |
BG26515A3 (en) | METHOD FOR OBTAINING ACYLAMINO DERIVATIVES | |
ZA764322B (en) | Novel 1-(benzazolyalkyl)piperidine derivatives | |
BG26518A3 (en) | METHOD FOR OBTAINING PHENYL-ALKANE DERIVATIVES | |
BG26526A3 (en) | METHOD FOR THE PREPARATION OF 1-(BENZAZOLYLALKYL)PIPERIDINE DERIVATIVES | |
BG27542A3 (en) | METHOD FOR THE PREPARATION OF 1-BENZAZOLYLALKYL-4-SUBSTITUTED PIPERIDINES | |
PL191647A1 (en) | METHOD OF THE PRODUCTION OF THENOPYRIDINE DERIVATIVES | |
SE433745B (en) | PROCEDURE FOR PREPARING TETRAHYDROISOKINOLIN DERIVATIVES | |
MX4118E (en) | PROCEDURE FOR PREPARING PIPERIDINE COMPOUND | |
SE423390B (en) | PROCEDURES FOR PREPARING EBURNAME DERIVATIVES | |
SE423902B (en) | PROCEDURE FOR PURINATE DERIVATIVES | |
IT1066655B (en) | PROCEDURE FOR DEPURING CAPROLATTAME | |
RO73050A (en) | PROCESS FOR PREPARATION OF SUBSTITUTED AMINOCHINESOLINE DERIVATIVES | |
BG26535A3 (en) | METHOD FOR OBTAINING INDOLQUINOLYSINES | |
SE7709402L (en) | PROCEDURE FOR THE PREPARATION OF TETRAHYDROPYRIDINE DERIVATIVES | |
BG26388A3 (en) | METHOD FOR OBTAINING DERIVATIVES OF XANTHENIC ACID | |
BG26534A4 (en) | METHOD FOR OBTAINING 2-METHYL-2-CYANOMETHYL-5-ISOPROPYLTETRAHYDROFURAN | |
IT1053899B (en) | PROCEDURE FOR PRODUCING OR PARAISOPROPENYLPHENOL DERIVATIVES | |
SE7608519L (en) | MORPHANTRIDINE DERIVATIVES | |
SE435291B (en) | PROCEDURE FOR PREPARING 7-ACYLAMINO-3 (1- (2-SULFAMINOETHYL) -TETRAZOL-5-YLTIOMETHYL) -3-CEFEM-4-CARBONIC ACID | |
DD122967A1 (en) | HYLAMIN DERIVATIVES | |
PL191309A1 (en) | METHOD OF MAKING NEW DERIVATIVES 1- (BENZAZOLYL-ALKYL) -PIPERIDINE |